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高分子-抗癌药偶合体纳米靶向药物 纳米医学

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Jalilov, Almaz S.; Li, Gaoquan; Nelsen, Stephen F.; Guzei, Ilia A.; Wu, Qin, “Solution and solid-state studies of doubly trimethylene-bridged tetraalkyl p-phenylenediamine diradical dication conformations.” Journal of the American Chemical Society, Volume 132, Number 17, pages 6176-6182, 2010. Li, Gaoquan; Nelsen, Stephen F.; Jalilov, Almaz S.; Guzei, Ilia A., “O-capped heteroadamantyl-substituted hydrazines and their oxidation products.” Journal of Organic Chemistry, Volume 75, Number 8, pages 2445-2452, 2010. Nelsen, Stephen; Li, Gaoquan; Schultz, Kevin; Tran, Hieu Q.; Guzei, Ilia; Evans, Dennis H.; “Alkylated Trimethylene-Bridged Bis(p-phenylenediamines),” Journal of the American Chemical Society, Volume 130, Number 35, pages 11620-11622, 2008. Li, Gaoquan; Tao, Zhi-Fu; Tong, Yunsong; Przytulinska, Magdalena K.; Kovar, Peter; Merta, Philip; Chen, Zehan; Zhang, Haiying; Sowin, Thomas; Rosenberg, Saul H.; Lin, Nan-Horng; “Synthesis and In-Vitro Biological Activity of Macrocyclic Urea Chk1 Inhibitors,” Bioorganic and Medicinal Chemistry Letters, Volume 17, pages 6499-6504, 2007. Tao, Zhi-Fu; Li, Gaoquan; Tong, Yunsong; Stewart, Kent D.; Chen, Zehan; Bui, Mai-Ha; Merta, Philip; Park, Chang; Kovar, Peter; Zhang, Haiying; Sham, Hing L.; Rosenberg, Saul H.; Sowin, Thomas J.; Lin, Nan-Horng; “Discovery of 4’-(1,4-dihydro-indeno[1,2-c]pyrazol-3-yl)-benzonitriles and 4’-(1,4-dihydro-indeno[1,2-c]pyrazol-3-yl)-pyridine-2’- carbonitriles as Potent Checkpoint Kinase 1 (Chk1) Inhibitors,” Bioorganic and Medicinal Chemistry Letters, Volume 17, Number 21, pages 5944-5951, 2007. Tao, Zhi-Fu; Li, Gaoquan; Tong, Yunsong; Chen, Zehan; Merta, Philip; Kovar, Peter; Zhang, Haiying; Rosenberg, Saul H.; Sham, Hing L.; Sowin, Thomas J.; Lin, Nan-Horng; “Synthesis and Biological Evaluation of 4’-(6,7-disubstituted-2,4-dihydro-indeno[1,2-c]pyrazol-3-yl)-biphenyl-4-ol as potent Chk1 Inhibitors,” Bioorganic and Medicinal Chemistry Letters, Volume 17, Number 15, pages 4308-4315, 2007 Li, Gaoquan; Hasvold, Lisa A.; Tao, Zhi-Fu; Wang, Gary T.; Gwaltney II, Stephen L.; Patel, Jyoti; Kovar, Robert b. Credo, Zehan Chen, Haiying Zhang, Chang Park, Hing L. Sham, Thomas Sowin, Saul H. Rosenberg, Peter; Lin, Nan-Horng; “Synthesis and Biological Evaluation of 1-(2,4,5-trisubstitutedphenyl-3-(5-cyanopyrazin-2-yl)ureas as Potent Chk1 Kinase Inhibitors.” Bioorganic and Medicinal Chemistry Letters, Volume 16, Number 8, page 2293-2298, 2006. Wang, Gary T.; Li, Gaoquan; Mantei, Robert A.; Chen, Zehan; Kevar, Peter; Gu, Wendy; Zhang, Haiying; Sham, Hing L.; Sowin, Thomas; Rosenburg, Saul H.; Lin, Nan-Horng; “1-(5-Chloro-2-alkoxyphenyl)-3-(5-cyano-pyrazin-2-yl)ureas as Potent and Selective Inhibitors of Chk1 Kinase: Synthesis, Preliminary SAR, and Biological Activities,” Journal of Medicinal Chemistry, Volume 48, Number 9, pages 3118-3121, 2005. Nelsen, Stephen F.; Li, Gaoquan; Konradsson, Asgeir; “Twist-Dependent Electronic Couplings in an Organic Intervalence Radical Cation,” Organic Letters, Volume 3, Number 10, pages 1583-1586, 2001. Li, Gaoquan; Tan, Jian; Fu, Hejian; Ma, Hong; Chen, Deben; Zhou, Zhonghua; “Effect of the Polysilane Structure on its Solution Fluorescence Quenching,” Journal of Applied Polymer Science, Volume 78, Number 1, pages 133-139, 2000. Fu, Hejian; Li, Gaoquan; Tan, Jian; Ma, Hong; Chen, Deben; Xie, Maonong; “Studies on the Laser Degradation of Polysilane Solutions,” European Polymer Journal, Volume 34, Number 2, pages 287-290, 1998. Fu, Hejian; Li, Gaoquan; Chen, Deben; Ma, Hong; Xie, Maonong; Chen, Shudong; “Studies on the Laser Degradation of the CHCl3 Solution of Polysilane,” Journal of Applied Polymer Science, Volume 66, Number 8, pages 1515-1519, 1997. Li, Gaoquan; Chen, Deben; Mo, Yiming; Bai, Fenglian; “Studies on the Fluorescence Quenching of Anthracenes by Polysilane Copolymers,” Journal of Applied Polymer Science, Volume 59, Number 9, pages 1463-1466, 1996. Chen, Deben; Li, Gaoquan; Mo, Yiming; Bai, Fenglian; “Studies on the Room-Temperature Solution Fluorescence Quenching of Polusilane Copolymers by Bromohydrocarbons,” European Polymer Journal, Volume 32, Number 5, pages 665-667, 1996. Li, Gaoquan; Chen, Deben; Bai, Fenglian; Mo, Yiming; “Studies on the Fluorescence Quenching of Polysilane Copolymers by Chlorohydrocarbons,” Journal of Polymer Science, Part B: Polymer Physics, Volume 34, pages 1583-1589, 1996.

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