Malkinson, John - University College London

个人简介

BPharm (Hons), First Class, The School of Pharmacy, University of London, 1996 PhD in Pharmaceutical Chemistry, The School of Pharmacy, University of London, 2000 Certificate in Teaching and Learning in Higher and Professional Education, Institute of Education, University of London, 2006

研究领域

Solid-phase synthesis of complex non-ribosomal peptides Natural product peptide conjugates including depsipeptides, lipopeptides and glycopeptides Peptides with anti-infective and anti-cancer activity

近期论文

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Synthesis and antibacterial evaluation of 3-Farnesyl-2-hydroxybenzoic acid from Piper multiplinervium. Journal article ; 2014 ; Fitoterapia ; Netherlands links: IRIS ; UCL Discovery ; doi ; author's authors [click to collapse] : Malami I,Gibbons S,Malkinson JP 2-Hydroxy-substituted cinnamic acids and acetanilides are selective growth inhibitors of Mycobacterium tuberculosis Journal article ; 2014 ; MedChemComm links: IRIS ; UCL Discovery ; doi authors [click to collapse] : Guzman JD,Mortazavi PN,Munshi T,Evangelopoulos D,McHugh TD,Gibbons S,Malkinson J,Bhakta S A new plant-derived antibacterial is an inhibitor of efflux pumps in Staphylococcus aureus Journal article ; 2013 ; International Journal of Antimicrobial Agents links: IRIS ; UCL Discovery ; doi authors [click to collapse] : Shiu WKP,Malkinson JP,Rahman MM,Curry J,Stapleton P,Gunaratnam M,Neidle S,Mushtaq S,Warner M,Livermore DM,Evangelopoulos D,Basavannacharya C,Bhakta S,Schindler BD,Seo SM,Coleman D,Kaatz GW,Gibbons S A new plant-derived antibacterial is an inhibitor of efflux pumps in Staphylococcus aureus. Journal article ; 2013 ; International Journal of Antimicrobial Agents links: IRIS ; UCL Discovery authors [click to collapse] : Shiu WKP,Malkinson JP,Rahman MM,Curry J,Stapleton P,Gunaratnam M,Neidle S,Mushtaq S,Warner M,Livermore DM,Evangelopoulos D,Basavannacharya C,Bhakta S,Schindler BS,Seo SM,Gruber S,Kaatz GW,Gibbons S Antitubercular specific activity of ibuprofen and the other 2-arylpropanoic acids using the HT-SPOTi whole-cell phenotypic assay. Journal article ; 2013 ; BMJ Open ; England links: IRIS ; UCL Discovery ; doi ; author's authors [click to collapse] : Guzman JD,Evangelopoulos D,Gupta A,Birchall K,Mwaigwisya S,Saxty B,McHugh TD,Gibbons S,Malkinson J,Bhakta S Towards the total synthesis of chlorofusin: Solid phase synthesis of the cyclic peptide Conference ; 2003 ; ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY links: IRIS ; UCL Discovery ; author's authors [click to collapse] : Searcey M,Malkinson JP,Kadom M Solid-phase synthesis of the mixirins: Cyclic lipopeptides with anti-tumour activity. Conference ; 2005 ; ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY links: IRIS ; UCL Discovery ; author's authors : Malkinson JP beta-AMINO ACID SYNTHESIS AND THE TOTAL SOLID-PHASE SYNTHESIS OF MIXIRINS A AND B Journal article ; 2009 ; BIOPOLYMERS links: IRIS ; UCL Discovery ; author's authors : Kemp G,Malkinson JP TOWARDS THE TOTAL SOLID-PHASE SYNTHESIS OF THE CYCLIC LIPODEPSIPEPTIDE DAPTOMYCIN Journal article ; 2009 ; BIOPOLYMERS links: IRIS ; UCL Discovery ; author's authors : Ezeigwe E,Malkinson JP Novel lipoamino acid and liposaccharide based peptide delivery system for tumor selective somatostatin analogs Conference ; 2000 ; PEPTIDES FOR THE NEW MILLENNIUM links: IRIS ; UCL Discovery ; author's authors [click to collapse] : Malkinson JP,Keri G,Artursson P,Toth I Solid-phase synthesis of des-N-tetramethyl triostin A (TANDEM) Conference ; 2004 ; Peptide Revolution: Genomics, Proteomics & Therapeutics links: IRIS ; UCL Discovery ; author's authors : Malkinson JP,Searcey M ORGN 223-Solid phase-supported synthesis of a water-soluble TANDEM analog Journal article ; 2006 ; ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY links: IRIS ; UCL Discovery ; author's authors [click to collapse] : Paumier D,Malkinson JP,Hampshire AJ,Fox KR,Searcey M Solid-phase synthesis of des-N-tetramethyltriostin a (TANDEM) Conference ; 2003 ; BIOPOLYMERS links: IRIS ; UCL Discovery ; author's authors : Malkinson JP,Searcey M Solid-phase synthesis of C-terminal thio-linked glycopeptides Conference ; 2003 ; BIOPOLYMERS links: IRIS ; UCL Discovery ; author's authors : Malkinson JP,Falconer RA Solid-phase synthesis of C-terminal thio-linked glycopeptides Conference ; 2004 ; Peptide Revolution: Genomics, Proteomics & Therapeutics links: IRIS ; UCL Discovery ; author's authors : Malkinson JP,Falconer RA Novel Lipoamino Acid- and Liposaccharide-Based System for Peptide Delivery:� Application for Oral Administration of Tumor-Selective Somatostatin Analogues Journal article ; 1999 ; Journal of Medicinal Chemistry links: IRIS ; UCL Discovery ; doi ; publisher authors [click to collapse] : Toth I,Malkinson JP,Flinn NS,Drouillat B,Horvath A,Erchegyi J,Idei M,Venetianer A,Artursson P,Lazorova L,Szende B,Keri G Lipoamino acid and liposaccharide based peptide delivery system for tumour selective somatostatin analogues Journal article ; 1999 ; Journal of Pharmacy and Pharmacology links: IRIS ; UCL Discovery authors [click to collapse] : Malkinson JP,Keri G,Artursson P,Toth I Synthesis ofC-Terminal Glycopeptides from Resin-Bound Glycosyl Azides via a Modified Staudinger Reaction Journal article ; 2000 ; Journal of Organic Chemistry links: IRIS ; UCL Discovery ; doi ; publisher authors [click to collapse] : Malkinson JP,Falconer RA,Toth I Solid-phase synthesis of C-terminal thio-linked glycopeptides Journal article ; 2002 ; Tetrahedron Letters links: IRIS ; UCL Discovery ; doi ; publisher authors : Malkinson JP,Falconer RA A new principle for tight junction modulation based on occludin peptides. Journal article ; 2003 ; Molecular pharmacology links: IRIS ; UCL Discovery ; doi ; publisher authors [click to collapse] : Tavelin S,Hashimoto K,Malkinson JP,Lazorova L,Toth I,Artursson P Pharmacists are scientists and clinicians Journal article ; 2004 ; Pharmaceutical Journal links: IRIS ; UCL Discovery authors : Malkinson JP Solid-Phase Synthesis of Chlorofusin Analogues Journal article ; 2007 ; Journal of Organic Chemistry links: IRIS ; UCL Discovery ; doi ; publisher authors [click to collapse] : Woon ECY,Arcieri M,Wilderspin AF,Malkinson JP,Searcey M Bioactive pyridine-N-oxide disulphides from Allium stipitatum. Journal article ; 2009 ; Journal of Natural Products links: IRIS ; UCL Discovery ; doi ; publisher authors [click to collapse] : Gibbons S,O'Donnell G,Poeschl R,Zimhony O,Gunaratnam M,Moreira JB,Neidle S,Evangelopoulos D,Bhakta S,Malkinson JP,Boshoff H,Lenaerts A A prodrug nanoparticle approach for the oral delivery of a hydrophilic peptide, leucine(5)-enkephalin, to the brain. Journal article ; 2012 ; Mol Pharm ; United States links: IRIS ; UCL Discovery ; doi ; author's authors [click to collapse] : Lalatsa A,Lee V,Malkinson JP,Zloh M,Schätzlein AG,Uchegbu IF Antibacterial acylphloroglucinols from Hypericum olympicum. Journal article ; 2012 ; J Nat Prod ; United States links: IRIS ; UCL Discovery ; doi ; author's authors [click to collapse] : Shiu WK,Rahman MM,Curry J,Stapleton P,Zloh M,Malkinson JP,Gibbons S