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药物合成工艺

近期论文

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1. One-Pot Addition–Intramolecular N-Cyclization of Carbamates Mediated by Alkali Metallic Reagents as an Approach to 4-(Fluoroalkyl)oxazolidin-2-ones, SYNTHESIS, 2011,3627-3634 2. Sodium Dithionite Initiated Reaction of Pent-4-en-1-amines with Fluoroalkyl Iodides for the Synthesis of 2-Fluoroalkyl Pyrrolidine Derivatives,Tetrahedron,2011,(6)761251-1257 3. Syntheisis of bromodifluoromethyl substituted pyrazoles and isoxazoles Journal of Fluorine Chemistry,2010,131, 426-432. 4. Stereoselective cycloaddition– lactonization reaction of 2-allyl-4- pentenoic acids with polyfluoroalkyl iodides. An efficient synthesis of polyfluoroalkyl-containing bicyclolactone derivatives,Tetrahedron,2010, 66, 7288-7294

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