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个人简介

教育经历 2005.9-2009.6 四川大学 | 药物化学 | 博士研究生毕业 | 理学博士学位 2002.9-2005.6 四川大学 | 药物化学 | 硕士研究生毕业 | 理学硕士学位 1998.9-2002.7 四川大学 | 药学 | 大学本科毕业 | 理学学士学位 工作经历 生命科学与工程学院 | 西南交通大学 四川农业大学

研究领域

[1]天然抗癌药物的发现及其结构修饰 [2]AI指导的小分子药物的发现、合成及作用机制 [3]金属催化的小分子药物Late-stage修饰及活性筛选

近期论文

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Bo Yin, Yu-Feng Du, Yan-Zuo Chen, Xiaohuan Li, Dong-Mei Fang, Feng Gao*, Palladium-catalyzed direct deprotonative arylation of 2-pyridylacetonitriles: Facile synthesis of alpha-aryl-2-pyridylacetonitrile, Tetrahedron Lett., 2020, 61, 152534. Lin-Xi Wan, Ji-Fa Zhang, Yong-Qi Zhen, Lan Zhang, Xiaohuan Li, Feng Gao*, and Xian-Li Zhou*, Isolation, Structure Elucidation, Semi-Synthesis, and Structural Modification of C19-Diterpenoid Alkaloids from Aconitum apetalum and Their Neuroprotective Activities, J. Nat. Prod., 2021, 84, 1067−1077. Lin-Xi Wan, Yong-Qi Zhe, Zhen-Xiang He, Yang Zhang, Lan Zhang, Xiaohuan Li, Feng Gao*, and Xian-Li Zhou, Late-stage modification of medicine: Pb-catalyzed direct synthesis and biological evaluation of N-aryltacrine derivatives, ACS Omega, 2021, 6, 9960−9972. Jing Lu, Jin-Pu Xu, Xiao-Huan Li, Chun-Gu Zhang, Feng Gao*, Three new C19-diterpenoid alkaloids from Aconitum novoluridum, Chem. Pharm. Bull., 2021, 69, 811–816. Lin-Xi Wan, Shi-Xing Miao, Zhen-Xiang He, Xiaohuan Li, Xian-Li Zhou, Feng Gao*, Pd-Catalyzed Direct Modification of an Anti-Alzheimers Disease Drug: Synthesis and Biological Evaluation of Aryl Donepezil Analogues, ACS Omega, 2021, 6, 36, 23347–23354 Shi-Xing Miao, Lin-Xi Wan, Zhen-Xiang He, Xian-Li Zhou, Xiaohuan Li, and Feng Gao*, Pd-Catalyzed Direct Diversification of Natural Anti-Alzheimer’s Disease Drug: Synthesis and Biological Evaluation of N‑Aryl Huperzine A Analogues, J. Nat. Prod., 2021, 84, 2374−2379. Yao Xiao, Neng Wang, Lin-Xi Wan, Xiao-Huan Li, Xian-Li Zhou, Feng Gao*, Iron-Catalyzed Skeletal Conversion of Lathyrane to Premyrsinane Euphorbia Diterpenes and Their Cytotoxic Activities, J. Nat. Prod., 2021, 84, 1838−1842 Ji-Fa Zhang, Lin Chen, Shuai Huang, Lian-Hai Shan, Feng Gao,* and Xian-Li Zhou*, Diterpenoid Alkaloids from Two Aconitum Species with Antifeedant Activity against Spodoptera exigua, J. Nat. Prod., 2017, 80, 3136–3142. Pei-Geng Xiao*, Feng-Peng Wang, Feng Gao, Lu-Ping Yan, Dong-Lin Chen, Yong Liu, A pharmacophylogenetic study of Aconitum L. (Ranunculaceae) from China, Acta Phytotaxonomic Sinica, 2006, 44, 1-46. (第五届中国科协期刊优秀学术论文奖) Yan-Nan Cao, Xin-Chuan Tian, Xing-Xiu Chen, Yun-Xin Yao, Feng Gao*, Xian-Li Zhou*, Rapid Ligand-Free Base-Accelerated Copper-Catalyzed Homo-coupling Reaction of Arylboronic Acids, Synlett, 2017, 28, 601-606. Nan-Nan Jia, Xin-Chuan Tian, Xiao-Xia Qu, Xing-Xiu Chen, Ya-Nan Cao, Yun-Xin Yao, Feng Gao*, Xian-Li Zhou, Copper-catalyzed Direct 2-Arylation of Benzoxazoles and Benzoimidazoles with Aryl Bromides and Cytotoxicity of Products, Scientific Reports, 2017, 7, 43758. Tianyi Liu, Annemarie L. Exarhos, Ethan C. Alguire, Feng Gao, Elmira Salami-Ranjbaran, Kevin Cheng, Tiezheng Jia, Joseph E. Subotnik, Patrick J. Walsh, James M. Kikkawa, and Zahra Fakhraai, Phys. Rev. Lett., 2017, 119, 095502. Jiadi Zhang, Sheng-Chun Sha, Ana Bellomo, Nisalak, Trongsiriwat, Feng Gao, Neil Tomson*, Patrick J. Walsh*, Positional Selectivity in C–H Functionalizations of 2-Benzyl Furans with Bimetallic Catalysts, J. Am. Chem. Soc., 2016, 138, 4260-4266 Guan Wen, Xiao-Xia Qu, Dan Wang, Xing-Xiu Chen, Xing Chuan Tian, Feng Gao*, Xian-Li Zhou*, Recent advances in design, synthesis and bioactivity of paclitaxel-mimics, Fitoterapia, 2016, 110, 26-37. Zhong-Sheng Wang, Wei Chen, Hai-Yue Jiang, Feng Gao∗, Xian Li Zhou∗, Semi-synthesis and structural elucidation of brevicanines A–D, four new C19-diterpenoid alkaloids with rotameric phenomenon from Aconitum brevicalcaratum, Fitoterapia, 2019, 134, 404-410. Jia-Xi Wang, Ling-Li Zheng, Feng Gao∗, Xian Li Zhou∗, Lewis acid-mediated skeleton transformation of Euphorbia diterpenes: From lathyrane to euphoractane and myrsinane, Fitoterapia, 2019, 133, 212-218. Tianyi Liu, Kevin Cheng, Elmira Salami-Ranjbaran, Feng Gao, Chen Li, Xiao Tong, Yi-Chih Lin, Yue Zhang, William Zhang, Lindsey Klinge, Patrick J. Walsh*, and Zahra Fakhraai*, The effect of chemical structure on the stability of physical vapor deposited glasses of 1,3,5-triarylbenzene, J. Chem. Phys., 2015, 143, 084506. Ling Li Zheng, Dan Wang, Yuan Yuan Li, Hong Yan Peng, Ming Yong Yuan, Feng Gao*, Ultrasound assisted extraction of total flavonoids from Aconitum gymnandrum, Pharmacog., Mag., 2014, 10, S141-146.

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