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个人简介

2014/01——至今 中山大学药学院,教授,博士生导师 2010/11——2013/12 中山大学药学院,副教授,博士生导师 2008/06——2010/06 澳大利亚Eskitis研究所,博士后研究员 2008/06——2010/10 中国科学院上海药物研究所,助理研究员 2003/09——2008/07 中国科学院上海药物研究所,药物化学,博士 1999/09——2003/07 复旦大学,化学系,学士

研究领域

研究领域为以活性筛选为导向从天然产物中发现抗炎、抗肿瘤、抗肥胖症活性小分子化合物,并进行结构修饰和相关的药理活性研究。

近期论文

查看导师最新文章 (温馨提示:请注意重名现象,建议点开原文通过作者单位确认)

Jun Sang, Lu Gan, Ming-Feng Zou, Zi-Jun Lin, Run-Zhu Fan, Jia-Luo Huang, Wei Li, Gui-Hua Tang, Sheng Yin*, Jolkinolide B sensitizes bladder cancer to mTOR inhibitors via dual inhibition of Akt signaling and autophagy, Cancer Letters, 2022, 526: 352-362. Fang-Yu Yuan, Yue-Hua Pan, Ai-Ping Yin, Wei Li, Dong Huang, Xue-Long Yan, Shu-Qi Wu, Gui-Hua Tang, Rong Pu, Sheng Yin*, Euphorstranoids A and B, two highly rearranged ingenane diterpenoids from Euphorbia stracheyi: structural elucidation, chemical transformation, and lipid-lowering activity, Organic Chemistry Frontiers, 2022, 9: 775-780. Wei Li, Gui-Hua Tang and Sheng Yin, Selaginellins from the genus Selaginella: isolation, structure, biological activity, and synthesis, Natural Product Reports, 2021, 38: 822-842 Dong Huang, Yue-Hua Pan, Fang-Yu Yuan, Wei Li, Xue-Long Yan, Ming-Feng Zou, Gui-Hua Tang, Sheng Yin*, Euphohyrisnoids A and B, two highly rearranged lathyrane diterpenoids from Euphorbia lathyris, Organic Letters, 2021, 23: 9602-9605. Fang-Yu Yuan#, Fan Xu#, Run-Zhu Fan, Wei Li, Dong Huang, Gui-Hua Tang, Tao Yuan, Li-She Gan*, Sheng Yin*, Structural elucidation of three 9,11-seco tetracyclic triterpenoids enables the structural revision of euphorol J, Journal of Organic Chemistry, 2021, 86: 7588-7593 Run-Zhu Fan#, Lin Chen#, Tong Su, Wei Li, Jia-Luo Huang, Jun Sang, Gui-Hua Tang, Sheng Yin*, Discovery of 8,9-seco-ent-kaurane diterpenoids as potential leads for the treatment of triple-negative breast cancer, Journal of Medicinal Chemistry, 2021, 64: 9926-9942. Dong Huang#, Rui-Min Wang#, Wei Li, Ying-Yuan Zhao, Fang-Yu Yuan, Xue-Long Yan, Ye Chen, Gui-Hua Tang, Hui-Chang Bi*, Sheng Yin*, Lathyrane diterpenoids as novel hPXR agonists: isolation, structural modification, and structure−activity relationships, ACS Medicinal Chemistry Letters, 2021, 12: 1159-1165 Dong Huang#, Ying-Yuan Zhao#, Rui-Min Wang, Wei Li, Fang-Yu Yuan, Xue-Long Yan, Xiao Yang, Gui-Hua Tang, Sheng Yin*, Hui-Chang Bi*, Natural product-based screening led to the discovery of a novel PXR agonist with anti-cholestasis activity, Acta Pharmacologica Sinica, 2021, https://doi.org/10.1038/s41401-021-00793-3. Jun Sang, Wei Li, Hong-Juan Diao, Run-Zhu Fan, Jia-Luo Huang, Lu Gan, Ming-Feng Zou, Gui-Hua Tang, Sheng Yin*, Jolkinolide B targets thioredoxin and glutathione systems to induce ROS-mediated paraptosis and apoptosis in bladder cancer cells, Cancer Letters, 2021, 509, 13-25. Wei Li, Gui-Hua Tang and Sheng Yin* Selaginellins from the genus Selaginella: isolation,structure, biological activity, and synthesis,Natural Product Reports, 2020, DOI: 10.1039/d0np00065e. Xue-Long Yan, Jun Sang, Shi-Xin Chen, Wei Li, Gui-Hua Tang, Li-She Gan, and Sheng Yin* , Euphorkanlide A, a Highly Modified Ingenane Diterpenoid with a C 24 Appendage from Euphorbia kansuensis, Organic Letters, 2019, 21, 4128−4131. Lan-Lan Lou#, Fu-Qiang Ni#, Lin Chen, Sharpkate Shaker, Wei Li, Rong Wang, Gui-Hua Tang, and Sheng Yin*, Germacrane Sesquiterpenoids as a New Type of Anticardiac Fibrosis Agent Targeting Transforming Growth Factor β Type I Receptor, Journal of Medicinal Chemistry, 2019, 62 , 7961-7975. Qin-Qin Song, # Yong Rao, # Gui-Hua Tang, # Zhang-Hua Sun, Jun-Sheng Zhang, Zhi-Shu Huang,* and Sheng Yin*. Tigliane Diterpenoids as a New Type of Antiadipogenic Agents Inhibit GRa-Dexras1 Axis in Adipocytes, Journal of Medicinal Chemistry, 2019, 62, 2060-2075. Yanqing Pang, Baijiao An, Lanlan Lou, Junsheng Zhang, Jun Yan, Ling Huang, Xingshu Li*, and Sheng Yin*;Design, Synthesis, and Biological Evaluation of Novel Selenium-Containing Isocombretastatins and Phenstatins as Antitumor Agents,Journal of Medicinal Chemistry,2017,60, 7300-7314. Zhu Jianyong, Wang Ruimin, Lou Lanlan, Li Wei, Tang Guihua, Bu Xianzhang,* and Sheng Yin*;Jatrophane Diterpenoids as Modulators of P-Glycoprotein-Dependent Multidrug Resistance (MDR): Advances of Structure-Activity Relationships and Discovery of Promising MDR Reversal Agents,Journal of Medicinal Chemistry,2016, 13, 6353–6369. Xin Liu, Hai-Bin Luo, Yi-You Huang, Jing-Mei Bao, Gui-Hua Tang, Yun-Yun Chen, Jun Wang, and Sheng Yin*; Selaginpulvilins A−D, New Phosphodiesterase‑4 Inhibitors with an Unprecedented Skeleton from Selaginella pulvinata; Organic Letters, 2014, 16, 282-285. Jun-Sheng Zhang, Xin Liu, Jiang Weng, Yan-Qiong Guo, Qing-Jiang Li, Abrar Ahmed, Gui-Hua Tang and Sheng Yin*;Natural diarylfluorene derivatives: isolation, total synthesis, and phosphodiesterase-4 inhibition,Organic Chemistry Frontiers, 2017, 4, 170. Gui-Hua Tang ,Zi-Wei Chen ,Ting-Ting Lin,,Min Tan,Xiao-Yun Gao,Jing-Mei Bao,Zhong-Bin Cheng,Zhang-Hua Sun,Gang Huang,Sheng Yin*; Neolignans from Aristolochia fordiana Prevent Oxidative Stress-Induced Neuronal Death through Maintaining the Nrf2/HO-1 Pathway in HT22 Cells,Journal of Natural Products,2015, 78, 1894-1903.

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