Katzenellenbogen, John A. - University of Illinois at Urbana-Champaign

个人简介

Professor John A. Katzenellenbogen attended Harvard University for his undergraduate and graduate work. He received his B.A. in 1966 and his Ph.D. in 1969, at which time he joined the faculty at Illinois.

研究领域

organic and inorganic chemistry, biochemistry, molecular biology, and radiochemistry

近期论文

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M. Jeyakumar and J.A. Katzenellenbogen. A Dual-Acceptor Time-Resolved Foster Resonance Energy Transfer Assay for Simultaneous Determination of Thyroid Hormone Regulation of Corepressor and Coactivator Binding to the Thyroid Hormone Receptor: Mimicking the Cellular Context of Thyroid Hormone Action, Anal. Biochem., 2009, 386, 73-78. PMID: 19111515 J.R. Gunther, Y. Du, E. Rhoden, I. Lewis, B. Revennaugh, T.W. Moore, S.H. Kim, R. Dingledine, H. Fu, and J.A. Katzenellenbogen. A Set of Time-Resolved Fluorescence Resonance Energy Transfer Assays or the Discovery of Inhibitors of Estrogen Receptor-Coactivator Binding, J. Biomol. Screening, 2009, 14, 181-93. Pub Med Abstract PMC2731238 J.R. Gunther, A.A. Parent, J. A. Katzenellenbogen. Alternative Inhibition of Androgen Receptor Signaling: Peptidomimetic Pyrimidines as Direct Androgen Receptor/Coactivator Disruptors. ACS Chem. Biol. , 2009, 4, 435-440. Pub Med Abstract PMID: 19441848 A.L. LaFrate, K.E. Carlson, J. A. Katzenellenbogen. Steriodal Bivalent Ligands for the Estrogen Receptor: Design, Synthesis, Characterization and Binding Affinities. Bioorg. Med. Chem., 2009, 17, 3528-3535. Pub Med Abstract PMID: 19394231 H. B. Zhou, K. W. Nettles, J. B. Bruning, Y. Kime, A. Joachimiak, S. Sharma, K. E. Carlson, F. Stossi, G. L. Greene, and J. A. Katzenellenbogen. Elemental Isomerism: A Boron-Nitrogen Surrogate for a Carbon-Carbon Double Bond Increases the Chemical Diversity of Estrogen Receptor Ligands. Chem. Biol. 2007, 14, 659-669. E. E. Parent, K. E. Carlson, J. A. Katzenellenbogen. Synthesis of 7alpha-(fluoromethyl)dihydrotestosterone and 7alpha-(fluoromethyl)nortestosterone, structurally paired androgens designed to probe the role of sex hormone binding globulin in imaging androgen receptors in prostate tumors by positron emission tomography. J. Org. Chem. 2007, 72, 5546-5554. K. W. Nettles, J. B. Bruning, G. Gil, J. Nowak, S. K. Sharma, J. B. Hahm, K. Kulp, R. B. Hochberg, H. Zhou, J. A. Katzenellenbogen, B. S. Katzenellenbogen, Y. Kim, A. Joachmiak, G. L. Greene. NFkB Selectivity of Estrogen Receptor Ligands Revealed by Comparative Crystallographic Analyses, Nature Chem. Bio. 2008, 4, 241-247. J. R. Gunther, T.W. Moore, M.L. Collins, J.A. Katzenellenbogen. Amphipathic Benzenes are Designed Inhibitors of the Estrogen Receptor Alpha/Steroid Receptor Coactivator Interaction, ACS Chem Bio, 2008, 5, 282-286. E. E. Parent, C. S. Dence, Terry L. Sharp, M. J. Welch, J. A. Katzenellenbogen. 7α-[18F]Fluoromethyl-dihydrotestosterone and 7α-[18F]Fluoromethyl-nortestosterone: Ligands to Determine the Role of Sex Hormone Binding Globulin for Steroidal Radiopharmaceuticals, J. Nucl. Med., 2008 49, 987-994. A. A. Parent, J. R. Gunther, and J. A. Katzenellenbogen. Blocking Estrogen Signaling After the Hormone: Pyrimidine-Core Inhibitors of Estrogen Receptor-Binding, J. Med. Chem., 2008, 51, 6512-6530. S. H. Kim, P. Ge, and J. A. Katzenellenbogen. A New Quinoline Sensitizer-Centered Lanthanide Chelate and Its Use for Protein Labling on Ni-NTA Beads for TR LRET Assays. Chem. Commun., 2009, 2, 183-185.