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1) Da-Li Zhang, Li-Yan Zhou, Jun-Min Quan, Wei Zhang, Lian-Quan Gu, Zhi-Shu Huang, Lin-Kun An*. Oxygen-Insertion of o-Quinone under Catalytic Hydrogenation Conditions. Org. Lett. 2013, 15 (6), 1162–1165. 2) Lin-Kun An*, Run-Lin Li, Ying-Lin Zuo, Lian-Quan Gu. Solvent-Free Thermocyclization of the Unactivated Linear Gramicidin S Precursor and Analogues. Org. Lett. 2011, 13 (1), 34-37. 3) Xi Cheng, Da-Li Zhang, Xiao-Bing Li, Jian-Tao Ye, Lei Shi, Zhi-Shu Huang, Lian-Quan Gu, Lin-Kun An*. Syntheses of diacyltanshinol derivatives and their suppressive effects on macrophage foam cell formation by reducing oxidized LDL uptake. Bioorg. Chem. 2014, 52, 24–30. 4) Wei Zhang, Qiu-Mao Chen, Xi Cheng, Ning Wu, Guo-Bin Yi, Ding Li, Jia-Heng Tan, Zhi-Shu Huang, Lian-Quan Gu, Lin-Kun An*. Syntheses, spectroscopic characterization and application to DNA determination of novel fluorescent pyridophenazine derivatives. Dyes Pigments 2013, 99, 82-89. 5) Zu-Ping Wu, Xi-Wei Wu, Ting Shen, Yan-Ping Li, Xi Cheng, Lian-Quan Gu, Zhi-Shu Huang, Lin-Kun An*. Synthesis, acetylcholinesterase and butyrylcholinesterase inhibitory activities of 7-alkoxyl substituted indolizinoquinoline-5,12-dione derivatives. Arch. Pharm. Chem. Life Sci. 2012, 345(3), 175-184. 6) Xi-Wei Wu, Zu-Ping Wu, Lu-Xia Wang, Hong-Bin Zhang, Jian-Wen Chen, Wei Zhang, Lian-Quan Gu, Zhi-Shu Huang, Lin-Kun An*. Synthesis, antimicrobial activity and possible mechanism of action of 9-bromo-substituted indolizinoquinoline-5,12-dione derivatives. Eur. J. Med. Chem. 2011, 46 (9), 4625-4633. 7) Ning Wu, Xi-Wei Wu, Keli Agama, Yves Pommier, Jun Du, Ding Li, Lian-Quan Gu*, Zhi-Shu Huang, Lin-Kun An*. A Novel DNA Topoisomerase I Inhibitor with Different Mechanism from Camptothecin Induces G2/M Phase Cell Cycle Arrest to K562 Cells. Biochemistry 2010, 49, 10131–10136. 8) De-Qing Shen, Zu-Ping Wu, Xi-Wei Wu, Zeng-Yun An, Xiang-Zhang Bu, Lian-Quan Gu, Zhi-Shu Huang, Lin-Kun An*. Synthesis and Antiproliferative Activity of Indolizinophthalazine-5,12-dione Derivatives, DNA Topoisomerase IB Inhibitors. Eur. J. Med. Chem. 2010, 45, 3938-3942. 9) De-Qing Shen, Ning Wu, Yan-Ping Li, Zu-Ping Wu, Hong-Bin Zhang, Zhi-Shu Huang, Lian-Quan Gu, Lin-Kun An*. Design, synthesis, and cytotoxicity of indolizinoquinoxaline-5,12-dione derivatives, novel DNA topoisomerase IB inhibitors. Aust. J. Chem. 2010, 63, 1116-1121. 10) Yu Cheng, Lin-Kun An*, Ning Wu, Xiao-Dong Wang, Xian-Zhang Bu, Zhi-Shu Huang and Lian-Quan Gu*. Synthesis, cytotoxic activities and structure–activity relationships of topoisomerase I inhibitors: indolizinoquinoline-5,12-dione derivatives. Bioorg. Med. Chem. 2008, 16, 4617–4625.

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