A novel and flexible sequentially cascade iodocyclization for the synthesis of highly substituted 1,3-diiodinated naphthalene derivatives in up to 99% yield under mild conditions is reported. The dihalogenated moiety can be readily introduced into the naphthalenes in a position that is usually not easily functionalized.

中文翻译：

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通过顺序级联碘环化反应的1,3-二碘萘衍生物的高度区域选择性合成

报道了在温和条件下以高达99％的收率合成高度取代的1,3-二碘代萘衍生物的新颖灵活的级联碘环化反应。二卤代部分可以容易地在通常不容易官能化的位置引入萘中。