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Rhodium(III)-Catalyzed Synthesis of Quinazolin-4(3H)-ones with N-Methoxyamides as Synthesis Reagents
Synthesis ( IF 2.2 ) Pub Date : 2022-03-09 , DOI: 10.1055/a-1792-9930 Guanyu Zhou 1 , Zhibin Huang 2 , Xu Xu 1 , Zhang Fang 1 , Pengcheng Huang 1 , Zefeng Deng 1 , Bao Li 3 , Yingsheng Zhao 4
中文翻译:
以N-甲氧基酰胺为合成试剂铑(III)-催化合成喹唑啉-4(3H)-ones
更新日期:2022-03-09
Synthesis ( IF 2.2 ) Pub Date : 2022-03-09 , DOI: 10.1055/a-1792-9930 Guanyu Zhou 1 , Zhibin Huang 2 , Xu Xu 1 , Zhang Fang 1 , Pengcheng Huang 1 , Zefeng Deng 1 , Bao Li 3 , Yingsheng Zhao 4
Affiliation
A practical method to synthesize quinoxalinones via intra/intermolecular amination using rhodium as the catalyst was developed. A wide variety of quinoxalinones were prepared from N-methoxybenzamides in moderate to excellent yields. Gram-scale reactions were also achieved, highlighting the synthetic importance of this new transformation.
中文翻译:
以N-甲氧基酰胺为合成试剂铑(III)-催化合成喹唑啉-4(3H)-ones
开发了一种以铑为催化剂通过分子内/分子间胺化合成喹喔啉酮的实用方法。由N-甲氧基苯甲酰胺以中等至优异的产率制备了多种喹喔啉酮。还实现了克级反应,突出了这种新转化的综合重要性。