当前位置: X-MOL 学术Synthesis › 论文详情
Our official English website, www.x-mol.net, welcomes your feedback! (Note: you will need to create a separate account there.)
Synthesis of Borylated Hydrazino Acid Derivatives
Synthesis ( IF 2.2 ) Pub Date : 2021-05-31 , DOI: 10.1055/s-0040-1706046
Andrei K. Yudin , Chieh-Hung Tien , Alina Trofimova , Wenjie Shao

α-Boryl-α-hydrazinoacetic acid is a highly functionalized boron-containing building block that can be easily accessed from readily available α-borylacetaldehyde. The hydrazine motif can be converted into a variety of α-borylated azoles and diazines in a straightforward protocol. Furthermore, the carboxy group can be derivatized to afford novel organoboron compounds that should find applications in various cross-coupling transformations.



中文翻译:

硼酰肼酸衍生物的合成

α-硼酸-α-肼基乙酸是一种高度官能化的含硼结构单元,可以从现成的 α-硼基乙醛中轻松获取。肼基序可以通过简单的方案转化为各种 α-硼化唑和二嗪。此外,可以将羧基衍生化以提供新型有机硼化合物,这些化合物应该在各种交叉偶联转化中得到应用。

更新日期:2021-06-01
down
wechat
bug