A synthesis of five 1-methoxy-1H-indole derivatives with imidazole, pyrazole, 1H-1,2,3-triazole, and 1H-1,2,4-triazole moieties was achieved by focusing on the formation mechanism of plant constituents. The objective 1-methoxy-1H-indole derivatives were obtained in situ (in one step) through the reaction of an unstable 3-(isothiocyanatomethyl)-1-methoxy-1H-indole, which was derived from neoglucobrassicin and plant enzyme myrosinase, and a heterocyclic compound. We have great hopes that this method would be useful for the development of medicinal seeds.

中文翻译：

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1-甲氧基-1的合成

通过关注咪唑，吡唑，1 H -1,2,3-三唑和1 H -1,2,4-三唑部分的合成，合成了5种1-甲氧基-1 H-吲哚衍生物。植物成分。通过不稳定的3-（异硫氰酸根合甲基）-1-甲氧基-1H-吲哚的反应原位（一步一步）制得目标1-甲氧基-1H-吲哚衍生物，该衍生物衍生自新葡糖溴素和植物酶黑芥子酶。和杂环化合物。我们非常希望该方法对药用种子的开发有用。