Starting from 2-aminobenzoic acid and correspondingly substituted 2-chloronitrobenzenes, 5-substituted-aminoacyl-5,10-dihydro-11H-dibenzo[b,e][1,4]diazepin -11- one derivatives with a differently high activity on ulcers were prepared. 8-Chloro-5,10-dihydro-5-[bis(2-hydroxyethyl)a-minoacetyl]-11H- dibenzo[b,e][1,4]diazepin-11-one hydrochloride (AWD 26-06) was selected for further clinical evaluation.

中文翻译：

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[具有抗胆碱活性的5,10-二氢-11H-二苯并[b，e] [1,4]二氮杂-11-酮的新衍生物]。

从2-氨基苯甲酸和相应取代的2-氯硝基苯开始，5-取代-氨基酰基-5,10-二氢-11H-二苯并[b，e] [1,4]二氮杂pin-11-具有一种高活性的衍生物准备好溃疡。8-氯-5,10-二氢-5- [双（2-羟乙基）α-氨基乙酰基] -11H-二苯并[b，e] [1,4]二氮杂-11-一盐酸盐（AWD 26-06）为选择进行进一步的临床评估。