Click chemistry for disulfide formation (Huang, 2024)

Hydrophobic Amplification Enabled High-Turnover Phosphazene Superbase Catalysis (Han, 2024)

Synthesis of Aliphatic Sulfonyl Fluorides in Developing Radical Methods (Han, 2024)

Horner–Wadsworth–Emmons olefination of proteins and glycoproteins (Huang, 2024)

Syntheses of 2-Thiazolines (Lu, 2024)

Chemoenzymatic Synthesis of 2-Aryl Thiazolines (Wu, 2024)

Cationic, Aromatic Acyl Donors for Directing Protein Acylation Using non-Covalent Interactions (Lu, 2024)

Ethenesulfonyl Fluoride (Han, 2024)

Synthesis of Highly Reactive Sulfone Iminium Fluorides (Wu, 2024)

N‐Vinyl Acrylamides: Versatile Heterobifunctional Electrophiles for Thiol−Thiol Bioconjugations （Ding, 2024)

Genetically enabling phosphorus fluoride exchange click chemistry in proteins (Lu, 2024)

Application of Perfluorobenzene as A Linker in Peptide Binding (Ding, 2024)

Non-symmetric Stapling of Native Peptides (Han, 2024)

A General Strategy to Install Amidine Functional Groups (Huang, 2024)

Peptide/Protein Stapling and Unstapling (Han, 2024)

Native Peptide Cyclization, Sequential Chemoselective Amidation in Water (Lu, 2023)

Comparative a-Helicity of Cyclic Pentapeptides in Water （Ding, 2023)

C−H Arylation of Tryptophans by [ArN2]X Promoted by Tosic Acid (Lu, 2023)

Cyclic Peptides for Drug Development (Ding, 2023)

Rapid Arene Triazene Chemistry for Macrocyclization (Lu, 2023)

Cascade Synthesis of Fluorinated Spiroheterocyclic Scaffolding for Peptidic Macrobicycles (Wu, 2023)

Synthesis of Aldehyde by Alcohol Oxidation (Gu, 2023)

Cys–Cys and Cys–Lys Stapling of Unprotected Peptides (Lu, 2023)

Non-Canonical Amino Acids in Peptide Drug Discovery (Gu, 2023)

Tyrosinase-Catalyzed Peptide Macrocyclization for mRNA Display (Huang, 2023)

Warheads for Targeted Covalent Inhibitors (Lu, Ding, Wu, 2023)

Tyrosinase—Catalyzed Peptide Macrocyclization for mRNA Display (Gu, 2023)

Cyclic peptide therapeutics (Huang, 2023)

Methionine Bioconjugation (Lu, 2023)

Prebiotic Synthesis of Cysteine Peptides (Ding, 2023)

Posttranslational Mutagenesis (Wu, 2023)

A Cysteine-Directed Proximity-Driven Crosslinking Method for Native Peptide Bicyclization (Gu, 2023)

Cooperative Stapling of Native Peptides (Huang, 2023)

Synthesis of Glycosyl Chlorooxime (Gu, 2023)

Disulfide Bond Formation (Huang, 2023)

Saccharides (Gu, 2023)

Trends in Peptide Drug Discovery (Huang, 2023)

Protecting-Group-Free S-Glycosylation (Gu, 2023)

Chlorooxime-Cysteine Bioconjugation (Huang, 2023)