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Jingjing Zhang,Xia Wu,Qinghe Gao, Xiao Geng, Peng Zhao, Yan-Dong Wu,*and Anxin Wu* Diamination/Oxidative Cross-Coupling/Bicyclization of Anilines and Methyl Ketones: Direct I2‑Promoted Synthesis of 1,2-Fused Oxindoles. Org. Lett. 2017, 19, 408−411.
Zhi-Wen Zhou, Feng-Cheng Jia, Cheng Xu, Shi-Fen Jiang, Yan-Dong Wu* and An-Xin Wu* Concise construction of 12H-benzo[4,5]thiazolo[2,3-b]quinazolin-12-ones via an unusual TBHP/Na2CO3 promoted cascade oxidative cyclization and interrupted Dimroth rearrangement, Chem. Commun. 2017, 53, 1056-1059.
Cai, Q.; Li, D. K.; Zhou, R. R.; Shu, W. M.; Wu, Y. D.*; Wu, A. X.* Acid-Catalyzed Multicomponent Tandem Cyclizations: Access to Polyfunctional Dihydroindolizino[8,7‑b]indoles. Org. Lett. 2016, 18, 1342−1345.
Cai, Q.; Li, D. K.; Zhou, R. R.; Zhuang, S. Y.; Ma, J. T.; Wu, Y. D.*; Wu, A. X.* Acid-Catalyzed Multicomponent Tandem Double Cyclization: A Onepot, Metal-free Route to Synthesize Polyfunctional 4,9-Dihydropyrrolo[2,1.b]quinazolines. J. Org. Chem. 2016, 81, 8104-8111.
Jia, F. C.; Zhou, Z. W.; Xu, C.; Wu, Y. D.*; Wu, A. X.* Divergent Synthesis of Quinazolin-4(3H)‑ones and Tryptanthrins Enabled by a tert-Butyl Hydroperoxide/K3PO4‑Promoted Oxidative Cyclization of Isatins at Room Temperature. Org. Lett. 2016, 18, 2942–2945.
Jia, F. C.; Xu, C.; Zhou, Z. W.; Cai, Q.; Wu, Y. D.*; Wu, A. X.* Substrates as Electron-Donor Precursors: Synthesis of Naphtho-Fused Oxindoles via Benzannulation of 2-Halobenzaldehydes and Indolin-2-ones. Org. Lett. 2016, 18, 5232–5235.
Shu, W. M.; Ma, J. R.; Zheng, K. L.; Wu, A. X.* Multicomponent Coupling Cyclization Access to Cinnolines via in Situ Generated Diazene with Arynes, and α‑Bromo Ketones. Org. Lett. 2016, 18, 196–199.
Shu, W. M.; Zheng, K. L.; Ma, J. R.; Wu, A. X.* Transition-Metal-Free Coupling Annulation of Arynes with Ketones and Alkynoates: Assembly of Functionalized Naphthalenes. Org. Lett. 2016, 18, 3762–3765.
Wang, M.; Xiang, J. C.; Cheng, Y.; Wu, Y. D.*; Wu, A. X.* Synthesis of 2,4,5-Trisubstituted Furans via a Triple C(sp3)−H Functionalization Reaction Using Rongalite as the C1 Unit. Org. Lett. 2016, 18, 524–527.
Wu, X.; Zhang, J. J.; Liu, S.; Gao, Q. H.; Wu, A. X.* An Efficient Synthesis of Polysubstituted Pyridines via Csp3–H Oxidation and C-S Cleavage of Dimethyl Sulfoxide. Adv. Synth. Catal. 2016, 358, 218–225.
Wu, X.; Gao, Q. H.; Geng, X.; Zhang, J. J.; Wu, Y. D.*; Wu, A. X.* Iodine-Promoted Oxidative Cross-Coupling of Unprotected Anilines with Methyl Ketones: A Site-Selective Direct C−H Bond Functionalization to C4-Dicarbonylation of Anilines. Org. Lett. 2016, 18, 2507–2510.
Xiang, J. C.; Cheng, Y.; Wang, M.; Wu, Y. D.*; Wu, A. X.* Direct Construction of 4-Hydroxybenzils via Para-Selective C–C Bond Coupling of Phenols and Aryl Methyl Ketones. Org. Lett. 2016, 18, 4360–4363.
Xiang, J. C.; Wang, M.; Cheng, Y.; Wu, Y. D.*; Wu, A. X.* Molecular Iodine-Mediated Chemoselective Synthesis of Multisubstituted Pyridines through Catabolism and Reconstruction Behavior of Natural Amino Acids. Org. Lett. 2016, 18, 24–27
Zhang, J. J.; Gao, Q. H.; Wu, X.; Geng, X.; Wu, Y. D.*; Wu, A. X.* Dual Roles of Methyl Ketones in Radziszewski-Type Reaction: Formal [2 + 1 + 1 + 1] Synthesis of 1,2,5-Trisubstituted Imidazoles. Org. Lett. 2016, 18, 1686–1689.
Zheng, K. L.; Shu, W. M.; Ma, J. R.; Wu, Y. D.*; Wu, A. X.* Acid-Mediated N−H/α,β-C(sp3)−H Trifunctionalization of Pyrrolidine: Intermolecular [3 + 2] Cycloaddition for the Construction of 2,3- Dihydro‑1H‑Pyrrolizine Derivatives. Org. Lett. 2016, 18, 3526–3529.
Xu, C.; Jia, F. C.; Zhou, Z. W.; Zheng, S. J.; Li, H.; Wu, A. X.* Copper-Catalyzed Multicomponent Domino Reaction of 2‑Bromoaldehydes, Benzylamines, and Sodium Azide for the Assembly of Quinazoline Derivatives. J. Org. Chem. 2016, 81, 3000–3006.
Gao, Q.; Liu, S.; Wu, X.; Zhang, J.; Wu, A., Direct Annulation of Hydrazides to 1,3,4-Oxadiazoles via Oxidative C(CO)-C(Methyl) Bond Cleavage of Methyl Ketones. Org. Lett. 2015, 17, 2960-2963.
Gao, Q.; Zhang, J.; Wu, X.; Liu, S.; Wu, A., Direct regioselective oxidative cross-coupling of indoles with methyl ketones: a novel route to C3-dicarbonylation of indoles. Org. Lett. 2015, 17, 134-137.
Jia, F. C.; Xu, C.; Zhou, Z. W.; Cai, Q.; Li, D. K.; Wu, A. X., Consecutive Cycloaddition/S(N)Ar/Reduction/Cyclization/Oxidation Sequences: A Copper-Catalyzed Multicomponent Synthesis of Fused N-Heterocycles. Org. Lett. 2015, 17, 2820-2823
Jia, F. C.; Zhou, Z. W.; Xu, C.; Cai, Q.; Li, D. K.; Wu, A. X., Expeditious Synthesis of 2-Phenylquinazolin-4-amines via a Fe/Cu Relay-Catalyzed Domino Strategy. Org. Lett. 2015, 17, 4236-4239.
Shu, W. M.; Zheng, K. L.; Ma, J. R.; Sun, H. Y.; Wang, M.; Wu, A. X., Convenient access to polyfunctional pyrazoles via a highly efficient and regioselective multicomponent reaction. Org. Lett. 2015, 17, 1914-1917.
Shu, W.-M.; Zheng, K.-L.; Ma, J.-R.; Wu, A.-X., Transition-Metal-Free Multicomponent Benzannulation Reactions for the Construction of Polysubstituted Benzene Derivatives. Org. Lett. 2015, 17, 5216-5219.
Xu, C.; Jia, F.-C.; Cai, Q.; Li, D.-K.; Zhou, Z.-W.; Wu, A.-X., Intramolecular decarboxylative coupling as the key step in copper-catalyzed domino reaction: facile access to 2-(1,3,4-oxadiazol-2-yl)aniline derivatives. Chem. Commun. 2015, 51, 6629-6632.
Gao, Q.; Liu, S.; Wu, X.; Zhang, J.; Wu, A., Coproduct Promoted Povarov Reaction: Synthesis of Substituted Quinolines from Methyl Ketones, Arylamines, and α-Ketoesters. J. Org. Chem. 2015, 80, 5984-5991.
Gao, Qinghe; Wu, Xia; Liu, Shan; Wu, Anxin*, I2-Promoted Selective Oxidative Cross-Coupling/Annulation of 2-Naphthols with Methyl Ketones: A Strategy To Build Naphtho[2,1-b]furan-1(2H)-ones with a Quaternary Center. Org. Lett. 2014, 16, 1732-1735.
Shu, Wen-Ming; Ma, Jun-Rui; Yang, Yan; Wu, An-Xin*, An Efficient Synthesis of Novel Fused Cycloheptatrienes through Mn(II)-Mediated Formal Intermolecular [2 + 2 + 2 + 1] Cycloaddition. Org. Lett. 2014, 16, 1286-1289.
Wu, Xia; Gao, Qinghe; Liu, Shan; Wu, Anxin*, I2-Catalyzed Oxidative Cross-Coupling of Methyl Ketones and Benzamidines Hydrochloride: A Facile Access to α-Ketoimides. Org. Lett. 2014, 16, 2888-2891.
Gao, Qinghe; Liu, Shan; Wu, Xia; Wu, Anxin*, Povarov-Type Reaction Using Methyl as New Input: Direct Synthesis of Substituted Quinolines by I2-Mediated Formal [3 + 2 + 1] Cycloaddition. Org. Lett. 2014, 16, 4582-4585.
Gao, Qinghe; Wu, Xia; Li, Yuhong; Liu, Shan; Meng, Xianggao; Wu, Anxin*, Iodine-Promoted Sequential C(sp3)H Functionalization Reactions: An Annulation Strategy for the Construction of 3-Methylthio-4-arylmaleimides. Adv. Synth. Catal. 2014, 356, 2924-2930.
Jia, Feng-Cheng; Xu, Cheng; Cai, Qun; Wu, An-Xin*, An integration of condensation/Ullmann-type coupling/bicyclization sequences: copper-catalyzed three-component direct synthesis of [1,2,4]triazolo[1,5-b]isoquinolin-5(1H)-ones. Chem. Commun. 2014, 50, 9914-9916.
Yang, Yan; Ni, Fan; Shu, Wen-Ming; Wu, An-Xin*, Copper-Catalyzed Domino Synthesis of 2-Imino-1H-imidazol-5(2H)-ones and Quinoxalines Involving CC Bond Cleavage with a 1,3-Dicarbonyl Unit as a Leaving Group. Chem. Eur. J. 2014, 20, 11776-11782.
Xue, Wei-Jian; Guo, Ya-Qiong; Gao, Fang-Fang; Li, Hong-Zheng; Wu, An-Xin*, A Novel Self-Sequence Reaction Network Involving a Set of Six Reactions in One Pot: The Synthesis of Substituted Benzothiazoles from Aromatic Ketones and Anilines. Org. Lett. 2013, 15, 890-893.
Gao, Qinghe; Wu, Xia; Jia, Fengcheng; Liu, Meicai; Zhu, Yanping; Cai, Qun; Wu, Anxin*, Design and Synthesis of 2-Acylbenzothiazoles via In Situ Cross-Trapping Strategy from Benzothiazoles with Aryl Ketones. J. Org. Chem. 2013, 78, 2792-2797.
Zhu, Yan-ping; Fei, Zhuan; Liu, Mei-Cai; Jia, Feng-Cheng; Wu, An-Xin*, Direct One-Pot Synthesis of Luotonin F and Analogues via Rational Logical Design. Org. Lett. 2013, 15, 378-381.
Zhu, Yan-Ping; Liu, Mei-Cai; Cai, Qun; Jia, Feng-Cheng; Wu, An-Xin*, A Cascade Coupling Strategy for One-Pot Total Synthesis of β-Carboline and Isoquinoline-Containing Natural Products and Derivatives. Chem. Eur. J. 2013, 10132-10137.
Shu, Wen-Ming; Yang, Yan; Zhang, Dong-Xue; Wu, Liu-Ming; Zhu, Yan-Ping; Yin, Guo-Dong; Wu, An-Xin*, Highly Efficient Synthesis of 3a,6a-Dihydrofuro[2,3-b]furans via a Novel Bicyclization. Org. Lett. 2013, 15, 456-459.
Yang, Yan; Shu, Wen-Ming; Yu, Shang-Bo; Ni, Fan; Gao, Meng; Wu, An-Xin*, Auto-tandem catalysis: synthesis of 4H-pyrido[1,2-a]pyrimidin-4-ones via copper-catalyzed aza-Michael addition-aerobic dehydrogenation-intramolecular amidation. Chem. Commun. 2013, 49, 1729-1731.
Yang, Yan; Ni, Fan; Shu, Wen-Ming; Yu, Shang-Bo; Gao, Meng; Wu, An-Xin*, Synthesis of Tetrasubstituted Unsymmetrical 1,4-Enediones via Copper-Promoted Autotandem Catalysis and Air As the Oxidant. J. Org. Chem. 2013, 78, 5418-5426.
Pang, Tao; Sun, Yu; Xue, Wei-Jian; Zhu, Yan-Ping; Yu, Guang-Ao; Wu, An-Xin*, Selective Synthesis of Six-Membered and Five-Membered Spiro Compounds by Controlling the Molar Ratio of Ternary Gallium/Indium/Copper (Ga/In/Cu) Catalysts. Adv. Synth. Catal. 2013, 355, 2208-2216.
Yin, Guodong; Ren, Tianbing; Rao, Yin; Zhou, Yifan; Li, Zhexian; Shu, Wenming; Wu, Anxin*, Stereoselective Synthesis of 2,8-Dioxabicyclo[3.3.1]nonane Derivatives via a Sequential Michael Addition/Bicyclization Reaction. J. Org. Chem. 2013, 78, 3132-3141.
Wang, Jun-Gang; Xiang, Jia-Chen; Wu, An-Xin *; Meng, Xiang-Gao*, Robust R-2(2)(8) hydrogen bonded dimer for crystal engineering of glycoluril derivatives. Crystengcomm 2013, 15, 10079-10085.
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