2024
120. Shi-Jiang He, Boming Shen, Lian-Zheng Zuo, Shao-Hua Xiang*, Huan-Huan Liu, Peiyuan Yu*, and Bin Tan*. Enantioselective Construction of Anthracenylidene-Based Axial Chirality by Asymmetric Heck Reaction. J. Am. Chem. Soc. 2024.
DOI: 10.1021/jacs.4c04024. Publication Date: Jul. 2, 2024.
119. Shao-Hua Xiang, Wei-Yi Ding*, Yong-Bin Wang, Bin Tan*. Catalytic atroposelective synthesis. Nat. Catal. 2024, 7, 483-498 (Invited Review Article).
DOI: 10.1038/s41929-024-01138-z. Publication Date: Apr. 30, 2024.
118. Quan-Hao Wu, Meng Duan, Yu Chen, Peiyuan Yu, Yong-Bin Wang*, Jun Kee Cheng, Shao-Hua Xiang, Kendall N. Houk*, Bin Tan*. Organocatalytic olefin C–H functionalization for enantioselective synthesis of atropisomeric 1,3-dienes. Nat. Catal. 2024, 7, 185-194.
DOI: 10.1038/s41929-023-01097-x. Publication Date: Jan. 17, 2024.
117. Ye-Hui Chen, Meng Duan, Si-Li Lin, Yu-Wei Liu, Jun Kee Cheng, Shao-Hua Xiang, Peiyuan Yu, Kendall N. Houk*, and Bin Tan*. Organocatalytic aromatization-promoted umpolung reaction of imines. Nat. Chem. 2024. 16, 408-416.
DOI: 10.1038/s41557-023-01384-x. Publication Date: Dec. 7, 2023.
116. Wen Bao, Ye-Hui Chen*, Yu-Wei Liu, Shao-Hua Xiang, and Bin Tan*. Atroposelective synthesis of 2-arylindoles via chiral phosphoric acid-catalyzed direct amination of indoles. Chin. J. Chem. 2024, 42, 731-735.
DOI: 10.1002/cjoc.202300589. Publication Date: Nov. 29, 2023.
2023
115. Si-Li Lin, Ye-Hui Chen*, Huan-Huan Liu, Shao-Hua Xiang, and Bin Tan*. Enantioselective Synthesis of Chiral Cyclobutenes Enabled by Brønsted Acid-Catalyzed Isomerization of BCBs. J. Am. Chem. Soc. 2023, 145, 21152-21158.
DOI: 10.1021/jacs.3c06525. Publication Date: Sep. 21, 2023.
114. Ming Wu, Yi-Wei Chen, Qian Lu, Yong-Bin Wang*, Jun Kee Cheng, Peiyuan Yu*, Bin Tan*. Organocatalytic Si-CAryl bond functionalization enabled atroposelective synthesis of axially chiral biaryl siloxanes. J. Am. Chem. Soc. 2023, 145, 20646-20654.
DOI: 10.1021/jacs.3c07839. Publication Date: Sep. 12, 2023.
113. Peng-Ying Jiang, San Wu, Guan-Jun Wang, Shao-Hua Xiang,* Bin Tan*. Synthesis of axially chiral QUINAP derivatives by ketone-catalyzed enantioselective oxidation. Angew. Chem. Int. Ed. 2023, 62, e202309272.
DOI: 10.1002/anie.202309272. Publication Date: Aug. 16, 2023.
112. Jun Kee Cheng, Bin Tan*. Chiral phosphoric acid-catalyzed enantioselective synthesis of axially chiral compounds involving indole derivatives. Chem. Rec. 2023, e202300147 (Invited Review Article).
DOI: 10.1002/tcr.202300147. Publication Date: Jun. 26, 2023.
111. Bing-Chao Da, Yong-Bin Wang, Jun Kee Cheng, Shao-Hua Xiang, Bin Tan*. Organocatalytic atroposelective cross-coupling of 1-azonaphthalenes and 2-naphthols. Angew. Chem. Int. Ed. 2023, 62, e202303128.
DOI: 10.1002/anie.202303128. Publication Date: Apr. 25, 2023.
110. Jun Wei, Jian Zhang, Jun Kee Cheng, Shao-Hua Xiang,* Bin Tan*. Modular enantioselective access to β-amino amides by Brønsted acid-catalysed multicomponent reaction. Nat. Chem. 2023, 15, 647-657.
DOI: 10.1038/s41557-023-01179-0. Publication Date: Apr. 13, 2023.
109. Xu-Jie Wang, Huan-Huan Liu, Jun Kee Cheng, Shao-Hua Xiang,* Bin Tan*. Catalytic enantioselective synthesis of chiral sulfonium ylides with S-stereogenic center. Chem 2023, 9, 1495-1504.
DOI: 10.1016/j.chempr.2023.02.017. Publication Date: Mar. 21, 2023.
108. Yu-Wei Liu, Ye-Hui Chen, Jun Kee Cheng, Shao-Hua Xiang, Bin Tan*. Enantioselective synthesis of 3-arylindole atropisomers via organocatalytic indolization of iminoquinones. Chem. Synth. 2023; 3: 11.
DOI: 10.20517/cs.2022.46. Publication Date: Feb. 26, 2023.
107. Pengquan Chen, Mei-Jun Lv, Jun Kee Cheng, Shao-Hua Xiang, Xiang-Zhong Ren, Junmin Zhang*, Bin Tan*. Enantioselective construction of triaryl-substituted all-carbon quaternary stereocenters via organocatalytic arylation of oxindoles with azonaphthalenes. Chem. Sci. 2023, 14, 2330-2335.
DOI: 10.1039/d2sc07103g. Publication Date: Feb. 6, 2023.
106. Jun Kee Cheng, Bin Tan*. Atroposelectivity with two catalysts. Nat. Synth. 2023, 2, 83-85 (Invited News & Views).
DOI: 10.1038/s44160-022-00209-y. Publication Date: Jan. 5, 2023.
105. Baohua Cai, Yuan Cui, Jian Zhou, Yong-Bin Wang, Limin Yang*, Bin Tan*, Jun Wang*. Asymmetric hydrophosphinylation of alkynes: facile access to axially chiral styrene-phosphines. Angew. Chem. Int. Ed. 2023, 62, e202215820.
DOI: 10.1002/anie.202215820. Publication Date: Nov. 24, 2022.
104. Jun Kee Cheng, Shao-Hua Xiang, Bin Tan*. Imidodiphosphorimidates (IDPis): catalyst motifs with unprecedented reactivity and selectivity. Chin. J. Chem. 2023, 41, 685-694 (Invited Review Article).
DOI: 10.1002/cjoc.202200618. Publication Date: Nov. 12, 2022.
103. Shi-Jiang He, Shuai Zhu, Sheng-Qi Qiu, Wei-Yi Ding*, Jun Kee Cheng, Shao-Hua Xiang*, Bin Tan*. Phosphoric Acid-Catalyzed enantioselective synthesis of axially chiral anthrone-based compounds. Angew. Chem. Int. Ed. 2023. 62, e202213914.
DOI: 10.1002/anie.202213914. Publication Date: Nov. 8, 2022.
2022
102. Jun Kee Cheng, Shao-Hua Xiang, Bin Tan*. IDPi-catalyzed highly enantioselective Pictet-Spengler reaction. Chem. Catal. 2022, 2, 2802–2839 (Invited Preview).
DOI: 10.1016/j.checat.2022.10.025. Publication Date: Nov. 17, 2022.
101. Shao-Hua Xiang, Jun Kee Cheng, Bin Tan*. The application of 2-naphthols in asymmetric synthesis of atropisomers. Synlett 2022, 33, 1991-2003 (Invited Review Article).
DOI: 10.1055/a-1965-2928. Publication Date: Oct. 20, 2022.
100. Jun Kee Cheng, Shao-Hua Xiang, Bin Tan*. Organocatalytic enantioselective synthesis of axially chiral molecules: development of strategies and skeletons. Acc. Chem. Res. 2022, 55, 2920-2937 (Invited Personal Account).
DOI: 10.1021/acs.accounts.2c00509. Publication Date: Sep. 29, 2022.
99. Sheng-Qi Qiu, Yu Chen, Xiang-Jun Peng, Shi-Jiang He, Jun Kee Cheng, Yong-Bin Wang, Shao-Hua Xiang, Jun Song, Peiyuan Yu*, Junmin Zhang*, Bin Tan*. Asymmetric construction of aryl-alkene axis by palladium-catalyzed Suzuki–Miyaura coupling reaction. Angew. Chem. Int. Ed. 2022, 61, e202211211.
DOI: 10.1002/anie.202211211. Publication Date: Sep. 16, 2022.
98. Shuai Zhu, Jian-Hui Mao, Jun Kee Cheng, Shao-Hua Xiang*, Bin Tan*. Discovery and organocatalytic enantioselective construction of axially chiral cyclohexadienylidene skeletons. Chem. 2022, 8, 2529-2541.
DOI: 10.1016/j.chempr.2022.06.014. Publication Date: Jul. 20, 2022. Highlighted by Synfacts 2022, 18, 1136.
97. Heng-Hui Li, Jia-Yan Zhang, Shaoyu Li, Yong-Bin Wang, Jun Kee Cheng, Shao-Hua Xiang, Bin Tan*. Asymmetric synthesis of binaphthyls through photocatalytic cross-coupling and organocatalytic kinetic resolution. Sci. Chin. Chem. 2022, 65, 1142-1148.
DOI: 10.1007/s11426-022-1246-8. Publication Date: May. 18, 2022.
96. San Wu, Shao-Hua Xiang, Jun Kee Cheng *, Bin Tan *. Axially chiral alkenes: Atroposelective synthesis and applications. Tetrahedron Chem 2022, 1, 100009.
DOI: 10.1016/j.tchem.2022.100009. Publication Date: Mar. 17, 2022.
95. Heng-Hui Li, Shaoyu Li, Jun Kee Cheng*, Shao-Hua Xiang, Bin Tan*. Direct arylation of N-heterocycles enabled by photoredox catalysis. Chem. Commun. 2022, 58, 4392-4395.
DOI: 10.1039/D2CC01212J. Publication Date: Mar. 10, 2022.
94. Wang Xia, Zi-An Zhou, Jie Lv, Shao-Hua Xiang*, Yong-Bin Wang, Bin Tan*. Facile synthesis of N-aryl phenothiazines and phenoxazines via Brønsted acid catalyzed C–H amination of arenes. Chem. Commun. 2022,58, 1613-1616.
DOI: 10.1039/d1cc06730c. Publication Date: Dec. 28, 2021.
2021
93. Qian-Jin An, Wang Xia, Wei-Yi Ding, Huan-Huan Liu, Shao-Hua Xiang, Yong-Bin Wang, Guofu Zhong*, Bin Tan*. Nitrosobenzene-enabled chiral phosphoric acid catalyzed enantioselective construction of atropisomeric N-arylbenzimidazoles. Angew. Chem. Int. Ed. 2021, 60, 24888-24893.
DOI: 10.1002/anie.202111251. Publication Date: Sep. 23, 2021.
92. Junxian Yang, Ji-Wei Zhang, Wen Bao, Sheng-Qi Qiu, Shaoyu Li, Shao-Hua Xiang*, Jun Song, Junmin Zhang*, Bin Tan*. Chiral phosphoric acid-catalyzed remote control of axial chirality at boron–carbon bond. J. Am. Chem. Soc. 2021, 143, 12924-12929.
DOI: 10.1021/jacs.1c05079. Publication Date: Aug. 12, 2021.
91. San Wu, Shao-Hua Xiang, Shaoyu Li, Wei-Yi Ding, Lei Zhang, Peng-Ying Jiang, Zi-An Zhou, Bin Tan*. Urea group-directed organocatalytic asymmetric versatile dihalogenation of alkenes and alkynes. Nat. Catal. 2021, 4, 692-702.
DOI: 10.1038/s41929-021-00660-8. Publication Date: Aug. 9, 2021.
90. Jian-Hui Mao, Yong-Bin Wang, Limin Yang, Shao-Hua Xiang, Quan-Hao Wu, Yuan Cui, Qian Lu, Jie Lv, Shaoyu Li, Bin Tan*. Organocatalyst-controlled site-selective arene C–H functionalization. Nat. Chem. 2021, 13, 982-991.
DOI: 10.1038/s41557-021-00750-x. Publication Date: Aug. 9, 2021.
89. Song Chen, Ya-Nan Li, Shao-Hua Xiang,* Shaoyu Li* and Bin Tan*. Electrochemical phenothiazination of naphthylamines and its application in photocatalysis. Chem. Comm. 2021, 57, 8512-8515.
DOI: 10.1039/d1cc03276c. Publication Date: Jul. 29, 2021.
88. Ji-Wei Zhang, Fei Jiang, Ye-Hui Chen, Shao-Hua Xiang, Bin Tan*. Synthesis of structurally diversified BINOLs and NOBINs via palladium-catalyzed C-H arylation with diazoquinones. Sci. China Chem. 2021, 64, 1515-1521.
DOI: 10.1007/s11426-021-1003-9. Publication Date: Jun. 23, 2021.
87. Ji-Wei Zhang, Shao-Hua Xiang*, Shaoyu Li, Bin Tan*. Copper-catalyzed synthesis of axially chiral biaryls with diaryliodonium salts as arylation reagents. Molecules 2021, 26, 3223 (Invited Article).
DOI: 10.3390/molecules26113223. Publication Date: May 27, 2021.
86. Jian Zhang, Jun Wei, Wei-Yi Ding, Shaoyu Li, Shao-Hua Xiang, Bin Tan*. Asymmetric pnictogen-bonding catalysis: transfer hydrogenation by a chiral antimony(V) cation/anion Pair. J. Am. Chem. Soc. 2021, 143, 6382-6387.
DOI: 10.1021/jacs.1c02808. Publication Date: Apr, 27, 2021.
85. Peng-Ying Jiang, Kai-Fang Fan, Shaoyu Li*, Shao-Hua Xiang, Bin Tan*. Metal-free oxidative cross-coupling enabled practical synthesis of atropisomeric QUINOL and its derivatives. Nat. Commun. 2021, 12, 2384.
DOI: 10.1038/s41467-021-22621-2. Publication Date: Apr, 22, 2021.
84. Jun Kee Cheng, Shao-Hua Xiang, Shaoyu Li, Liu Ye, Bin Tan*. Recent advances in catalytic asymmetric construction of atropisomers. Chem. Rev. 2021, 121, 4805-4902 (Invited Review Article).
DOI: 10.1021/acs.chemrev.0c01306. Publication Date: Mar. 27, 2021.
83. Bing-Chao Da, Shao-Hua Xiang, Shaoyu Li, Bin Tan*. Chiral phosphoric acid catalyzed asymmetric synthesis of axially chiral compounds. Chin. J. Chem. 2021, 39, 1787-1796 (Invited Personal Account).
DOI: 10.1002/cjoc.202000751. Publication Date: Jan. 22, 2021.
2020
82. Lei Zhang*, Jiahua Shen, San Wu, Guofu Zhong*, Yong-Bin Wang, Bin Tan*. Design and atroposelective construction of IAN analogues by organocatalytic asymmetric heteroannulation of alkynes. Angew. Chem. Int. Ed. 2020, 59, 23077-23082.
DOI: 10.1002/anie.202010598. Publication Date: Sep. 4, 2020.
81. Shao-Hua Xiang, Bin Tan. Advances in asymmetric organocatalysis over the last 10 years. Nat. Commun. 2020, 11, 3786 (Invited Comment).
DOI: 10.1038/s41467-020-17580-z. Publication Date: Jul. 29, 2020.
80. Ji-Wei Zhang, Liang-Wen Qi, Shaoyu Li*, Shao-Hua Xiang, Bin Tan*. Direct construction of NOBINs via domino arylation and sigmatropic rearrangement reactions. Chin. J. Chem. 2020, 38, 1503-1514.
DOI: 10.1002/cjoc.202000358. Publication Date: Jul. 13, 2020.
79. Wei-Yi Ding, Peiyuan Yu, Qian-Jin An, Katherine L. Bay, Shao-Hua Xiang, Shaoyu Li, Ying Chen, K.N. Houk*, Bin Tan*. DFT-guided phosphoric-acid-catalyzed atroposelective arene functionalization of nitrosonaphthalene. Chem 2020, 6, 2046-2059.
DOI: 10.1016/j.chempr.2020.06.001. Publication Date: Jun. 23, 2020.
78. Ye-Hui Chen, Heng-Hui Li, Xiao Zhang, Shao-Hua Xiang*, Shaoyu Li, Bin Tan*. Organocatalytic enantioselective synthesis of atropisomeric aryl-p-quinones: Platform molecules for diversity-oriented synthesis of biaryldiols. Angew. Chem. Int. Ed. 2020, 59, 11374-11378.
DOI: 10.1002/anie.202004671. Publication Date: Apr. 10, 2020.
77. Shengyi Yan, Wang Xia, Shaoyu Li, Qiuling Song*, Shao-Hua Xiang, Bin Tan*. Michael reaction inspired atroposelective construction of axially chiral biaryls. J. Am. Chem. Soc. 2020, 142, 7322-7327.
DOI: 10.1021/jacs.0c01963. Publication Date: Apr. 8, 2020.
76. Wang Xia, Qian-Jin An, Shao-Hua Xiang, Shaoyu Li, Yong-Bin Wang, Bin Tan*. Chiral phosphoric acid catalyzed atroposelective C-H amination of arenes. Angew. Chem. Int. Ed. 2020, 59, 6775-6779.
DOI: 10.1002/anie.202000585. Publication Date: Feb. 4, 2020.
75. Shaoyu Li, Shao-Hua Xiang*, Bin Tan*. Chiral phosphoric acid creates promising opportunities for enantioselective photoredox catalysis. Chin. J. Chem. 2020, 38, 213-214 (Invited Emerging Topic).
DOI: 10.1002/cjoc.201900472. Publication Date: Dec. 23, 2019.
74. Jian Zhang, Yi-Yan Wang, He Sun, Shao-Yu Li, Shao-Hua Xiang, Bin Tan*. Enantioselective three-component Ugi reaction catalyzed by chiral phosphoric acid. Sci. China Chem. 2020, 63, 47-54.
DOI: 10.1007/s11426-019-9606-2. Publication Date: Oct. 22, 2019.
2019
73. Shuai Zhu, Ye-Hui Chen, Yong-Bin Wang, Peiyuan Yu, Shao-Yu Li, Shao-Hua Xiang, Jun-Qi Wang, Jian Xiao, Bin Tan*. Organocatalytic atroposelective construction of axially chiral arylquinones. Nat. Commun. 2019, 10, 4268.
DOI: 10.1038/s41467-019-12269-4. Publication Date: Sep. 19, 2019.
72. Yong-Bin Wang, Quan-Hao Wu, Zhi-Peng Zhou, Shao-Hua Xiang, Yuan Cui, Peiyuan Yu, Bin Tan*. Asymmetric construction of axially chiral 2-arylpyrroles by chirality transfer of atropisomeric alkenes. Angew. Chem. Int. Ed. 2019, 58, 13443-13447.
DOI: 10.1002/anie.201907470. Publication Date: Jul. 23, 2019.
71. Dong-Liang Lu, Ye-Hui Chen, Shao-Hua Xiang, Peiyuan Yu, Bin Tan, Shaoyu Li*. Atroposelective construction of arylindoles by chiral phosphoric acid-catalyzed cross-coupling of indoles and quinones. Org. Lett. 2019, 21, 6000-6004.
DOI: 10.1021/acs.orglett.9b02143. Publication Date: Jul. 23, 2019.
70. Yong-Bin Wang, Peiyuan Yu, Zhi-Peng Zhou, Jian Zhang, Jun (Joelle) Wang, Shi-Hui Luo, Qiang-Shuai Gu, K. N. Houk*, Bin Tan*. Rational design, enantioselective synthesis and catalytic applications of axially chiral EBINOLs. Nat. Catal. 2019, 2, 504-513.
DOI: 10.1038/s41929-019-0278-7. Publication Date: Jun. 3, 2019.
69. Liang-Wen Qi, Shaoyu Li, Shao-Hua Xiang, Jun (Joelle) Wang*, Bin Tan*. Asymmetric construction of atropisomeric biaryls via a redox neutral cross-coupling strategy. Nat. Catal. 2019, 2, 314-323.
DOI: 10.1038/s41929-019-0247-1. Publication Date: Mar. 25, 2019.
68. Lei Zhang, Shao-Hua Xiang, Jun (Joelle) Wang*, Jian Xiao, Jun-Qi Wang, Bin Tan*. Phosphoric acid-catalyzed atroposelective construction of axially chiral arylpyrroles. Nat. Commun. 2019, 10, 566.
DOI: 10.1038/s41467-019-08447-z. Publication Date: Feb. 4, 2019.
67. Lin-Lin Zhang, Bing-Chao Da, Shao-Hua Xiang*, Shuai Zhu, Zi-Yun Yuan, Zhen Guo*, Bin Tan*. Organocatalytic double arylation of 3-isothiocyanato oxindoles: Stereocontrolled synthesis of complex spirooxindoles. Tetrahedron 2019, 75, 1689-1696.
DOI: 10.1016/j.tet.2018.11.016. Publication Date: Nov. 16, 2018.
2018
66. Lin-Lin Zhang, Ji-Wei Zhang, Shao-Hua Xiang*, Zhen Guo*, Bin Tan*. Stereoselective construction of complex spirooxindoles via bisthiourea catalyzed three-component reactions. Chin. J. Chem. 2018, 36, 1182-1186.
DOI: 10.1002/cjoc.201800368. Publication Date: Dec. 18, 2018.
65. Lin-Lin Zhang, Ji-Wei Zhang, Shao-Hua Xiang*, Zhen Guo*, Bin Tan*. Remote control of axial chirality: synthesis of spirooxindole–urazoles via desymmetrization of ATAD. Org. Lett. 2018, 20, 6022-6025.
DOI: 10.1021/acs.orglett.8b02361. Publication Date: Sep. 17, 2018.
64. Jian Zhang, Peiyuan Yu, Shao-Yu Li, He Sun, Shao-Hua Xiang, Jun Wang, Kendall N. Houk*, Bin Tan*. Asymmetric phosphoric acid–catalyzed four-component Ugi reaction. Science 2018, 361, eaas8707.
DOI: 10.1126/science.aas8707. Publication Date: Sep. 14, 2018.
63. Yong-Bin Wang, Bin Tan*. Construction of axially chiral compounds via asymmetric organocatalysis. Acc. Chem. Res. 2018, 51, 534-547 (Invited Personal Account).
DOI: 10.1021/acs.accounts.7b00602. Publication Date: Feb. 8, 2018.
62. Xiao Zhang, Ye-Hui Chen, Bin Tan*. Organocatalytic enantioselective transformations involving quinone derivatives as reaction partners. Tetrahedron Lett. 2018, 59, 473-486 (Invited Review).
DOI: 10.1016/j.tetlet.2017.12.055. Publication Date: Dec. 18, 2017.
61. Liang-Wen Qi, Jian-Hui Mao, Jian Zhang, Bin Tan*. Organocatalytic asymmetric arylation of indoles enabled by azo groups. Nat. Chem. 2018, 10, 58-64.
DOI: 10.1038/NCHEM.2866. Publication Date: Oct. 2, 2017.
2017
60. Ye-Hui Chen, Liang-Wen Qi, Fang Fang, Bin Tan*. Organocatalytic atroposelective arylation of 2-naphthylamines as a practical approach to axially chiral biaryl amino alcohols. Angew. Chem. Int. Ed. 2017, 56, 16308-16311.
DOI: 10.1002/anie.201710537. Publication Date: Nov. 5, 2017.
59. Yong-Bin Wang, Sheng-Cai Zheng, Yu-Mei Hu, Bin Tan*. Brønsted Acid-Catalysed Enantio-selective Construction of Axially Chiral Arylquinazolinones. Nat. Commun. 2017, 8, 15489.
DOI: 10.1038/ncomms15489. Publication Date: Mar. 19, 2017.
58. Sheng-Cai Zheng, San Wu, Yun-Hao Zhang, Qinghai Zhou, Lung Wa Chung, Liu Ye, Bin Tan*. Organocatalytic atroposelective synthesis of axially chiral styrenes. Nat. Commun. 2017, 8, 15238.
DOI: 10.1038/ncomms15238. Publication Date: Mar. 3, 2017.
57. Lei Zhang, Jian Zhang, Ji Ma, Dao-Juan Cheng, Bin Tan*. Highly atroposelective synthesis of arylpyrroles by catalytic asymmetric Paal-Knorr reaction. J. Am. Chem. Soc. 2017, 139, 1714-1717.
DOI: 10.1021/jacs.6b09634. Publication Date: Jan. 20, 2017.
2016
56. Lei Li, Zhong-Liang Li, Fu-Li Wang, Zhen Guo, Yong-Feng Cheng, Na Wang, Chao Fang, Jingjiang Liu, Chunhui Hou, Bin Tan, Xin-Yuan Liu*. Radical aryl migration enables diversity-oriented synthesis of structurally diverse medium/macro- or bridged-rings. Nat. Commun. 2016, 7, 13852.
DOI: 10.1038/ncomms13852. Publication Date: Dec. 22, 2016.
55. Shao-Yu Li, Ji-Wei Zhang, Xian-Lin Li, Dao-Juan Cheng, Bin Tan*. Phosphoric acid-catalyzed asymmetric synthesis of SPINOL derivatives. J. Am. Chem. Soc. 2016, 138, 16561-16566.
DOI: 10.1021/jacs.6b11435. Publication Date: Dec. 2, 2016.
54. Jin-Hui Xu, Sheng-Cai Zheng, Ji-Wei Zhang, Xin-Yuan Liu, Bin Tan*. Construction of tropane derivatives by organocatalytic asymmetric dearomatization of isoquinolines. Angew. Chem. Int. Ed. 2016, 55, 11834-11839.
DOI: 10.1002/anie.201605736. Publication Date: Sep. 7, 2016.
53. Xiao-Long Yu, Liping Kuang, Su Chen, Xiao-Long Zhu, Zhong-Liang Li, Bin Tan, Xin-Yuan Liu*. Counteranion-controlled unprecedented diastereo- and enantioselective tandem Povarov reaction for construction of bioactive octahydro-dipyrroloquinolines. ACS Catal. 2016, 6, 6182-6190.
DOI: 10.1021/acscatal.6b01492. Publication Date: Aug. 8, 2016.
52. Jin-Shun Lin, Xiao-Yang Dong, Tao-Tao Li, Na-Chuan Jiang, Bin Tan, Xin-Yuan Liu*. A dual-catalytic strategy to direct asymmetric radical aminotrifluoromethylation of alkenes. J. Am. Chem. Soc. 2016, 138, 9357-9360.
DOI: 10.1021/jacs.6b04077. Publication Date: Jul. 14, 2016.
51. Ji-Wei Zhang, Jin-Hui Xu, Dao-Juan Cheng, Chuan Shi, Xin-Yuan Liu*, Bin Tan*. Discovery and enantiocontrol of axially chiral urazoles via organocatalytic tyrosine click reaction. Nat. Commun. 2016, 7, 10677.
DOI: 10.1038/ncomms10677. Publication Date: Feb. 11, 2016.
50. Ning-Yuan Yang, Zhong-Liang Li, Liu Ye, Bin Tan, Xin-Yuan Liu*. Organic base-catalysed solvent-tuned chemoselective carbotrifluoromethylation and oxytrifluoromethylation of unactivated alkenes. Chem. Commun. 2016, 52, 9052-9055.
DOI: 10.1039/C6CC00364H. Publication Date: Feb. 1, 2016.
49. Can-Liang Ma, Xiao-Hua Li, Xiao-Long Yu, Xiao-Long Zhu, Yong-Zhou Hu, Xiao-Wu Dong*, Bin Tan*, Xin-Yuan Liu*. Gold-catalyzed tandem synthesis of bioactive spiro-dipyrroloquinolines and its application in the one-step synthesis of incargranine B aglycone and seneciobipyrrolidine (I). Org. Chem. Front. 2016, 3, 324-329.
DOI: 10.1039/C5QO003. Publication Date: Jan. 6, 2016.
2015
48. Ye-Hui Chen, Dao-Juan Cheng, Jian Zhang, Yong Wang, Xin-Yuan Liu*, Bin Tan*. Atroposelective synthesis of axially chiral biaryldiols via organocatalytic arylation of 2‑naphthols. J. Am. Chem. Soc. 2015, 137, 15062-15065.
DOI: 10.1021/jacs.5b10152. Publication Date: Nov. 11, 2015.
47. Jian Zhang, Shao-Xia Lin, Dao-Juan Cheng, Xin-Yuan Liu*, Bin Tan*. Phosphoric acid-catalyzed asymmetric classic Passerini reaction. J. Am. Chem. Soc. 2015, 137, 14039-14042.
DOI: 10.1021/jacs.5b09117. Publication Date: Oct. 21, 2015.
46. Zhi-Jia Fang, Sheng-Cai Zheng, Zhen Guo, Jing-Yao Guo, Bin Tan*, Xin-Yuan Liu*. Asymmetric synthesis of axially chiral isoquinolones: nickel-catalyzed denitrogenative transannulation. Angew. Chem. Int. Ed. 2015, 54, 9528-9532.
DOI: 10.1002/anie.201503207. Publication Date: Jun. 26, 2015.
45. Ming-Yue Wu, Wei-Wei He, Xin-Yuan Liu*, Bin Tan*. Asymmetric construction of spirooxindoles by organocatalytic multicomponent reactions using diazooxindoles. Angew. Chem. Int. Ed. 2015, 54, 9409-9413.
DOI: 10.1002/anie.201504640. Publication Date: Jun. 19, 2015.
44. Jin-Shun Lin, Peng Yu, Lin Huang, Pan Zhang, Bin Tan*, Xin-Yuan Liu*. Brønsted acid-catalyzed asymmetric hydroamination of alkenes: synthesis of pyrrolidines bearing a tetrasubstituted carbon stereocenter. Angew. Chem. Int. Ed. 2015, 54, 7847-7851.
DOI: 10.1002/anie.201501762. Publication Date: May 26, 2015.
43. Lin Huang, Jin-Shun Lin, Bin Tan*, Xin-Yuan Liu*. Alkene trifluoromethylation-initiated remote α-azidation of carbonyl compounds toward trifluoromethyl γ-lactam and spirobenzofuranone-lactam. ACS Catal. 2015, 5, 2826-2831.
DOI: 10.1021/acscatal.5b00311. Publication Date: Mar. 20, 2015.
42. Lin Huang, Sheng-Cai Zheng, Bin Tan*, Xin-Yuan Liu*. Metal-free direct 1,6- and 1,2-difunctionalization triggered by radical trifluoromethylation of alkenes. Org. Lett. 2015, 17, 1589-1592.
DOI: 10.1021/acs.orglett.5b00479. Publication Date: Mar. 12, 2015.
41. Lin Huang, Sheng-Cai Zheng, Bin Tan*, Xin-Yuan Liu*. Trifluoromethylation-initiated remote cross-coupling of carbonyl compounds to form carbon–heteroatom/carbon bonds. Chem. Eur. J. 2015, 21, 6718-6722.
DOI: 10.1002/chem.201500629. Publication Date: Mar. 12, 2015.
40. Peng Yu, Sheng-Cai Zheng, Ning-Yuan Yang, Bin Tan*, Xin-Yuan Liu*. Phosphine-catalyzed remote β-C-H functionalization of amine triggered by trifluoromethylation of alkene: one-pot synthesis of bistrifluoromethylated enamides and oxazoles. Angew. Chem. Int. Ed. 2015, 54, 4041-4045.
DOI: 10.1002/anie.201412310. Publication Date: Feb. 18, 2015.
39. Can-Liang Ma, Xiao-Long Yu, Xiao-Long Zhu, Yong-Zhou Hu, Xiao-Wu Dong, Bin Tan*, Xin-Yuan Liu*. Platinum-catalyzed tandem cyclization reaction to multiply substituted indolines under microwave-assisted conditions. Adv. Synth. Catal. 2015, 357, 569-575.
DOI: 10.1002/adsc.201400933. Publication Date: Jan. 29, 2015.
2014
38. Lei Li, Jing-Yao Guo, Xing-Guo Liu, Su Chen, Yong Wang, Bin Tan*, Xin-Yuan Liu*. Amide groups switch selectivity: C–H trifluoromethylation of α,β-unsaturated amides and subsequent asymmetric transformation. Org. Lett. 2014, 16, 6032-6035.
DOI: 10.1021/ol503067g. Publication Date: Nov. 10, 2014.
37. Peng Yu, Jin-Shun Lin, Lei Li, Sheng-Cai Zheng, Ya-Ping Xiong, Li-Jiao Zhao, Bin Tan*, Xin-Yuan Liu*. Enantioselective C–H bond functionalization triggered by radical trifluoromethylation of unactivated alkene. Angew. Chem. Int. Ed. 2014, 53, 11890-11894.
DOI: 10.1002/anie.201405401. Publication Date: Sep. 8, 2014.
36. Jin-Shun Lin, Xiang-Geng Liu, Xiao-Long Zhu, Bin Tan*, Xin-Yuan Liu*. Copper-catalyzed aminotrifluoromethylation of unactivated alkenes with TMSCF3: construction of trifluoromethylated azaheterocycles. J. Org. Chem. 2014, 79, 7084-7092.
DOI: 10.1021/jo5012619. Publication Date: Jul. 8, 2014.
35. Xing-Li Zhu, Jin-Hui Xu, Dao-Juan Cheng, Li-Jiao Zhao, Xin-Yuan Liu*, Bin Tan*. In situ generation of electrophilic trifluoromethylthio reagents for enantioselective trifluoromethylthiolation of oxindoles. Org. Lett. 2014, 16, 2192-2195.
DOI: 10.1021/ol5006888. Publication Date: Apr. 3, 2014.
34. Dao-Juan Cheng, Liang Yan, Shi-Kai Tian*, Ming-Yue Wu, Lu-Xin Wang, Zi-Li Fan, Sheng-Cai Zheng, Xin-Yuan Liu*, Bin Tan*. Highly enantioselective kinetic resolution of axially chiral BINAM derivatives catalyzed by a Brønsted acid. Angew. Chem. Int. Ed. 2014, 53, 3684-3687.
DOI: 10.1002/anie.201310562. Publication Date: Mar. 3, 2014.
33. Ya-Ping Xiong, Ming-Yue Wu, Xiang-Yu Zhang, Can-Liang Ma, Lin Huang, Li-Jiao Zhao, Bin Tan*, Xin-Yuan Liu*. Direct access to α-CF3-enones via efficient copper-catalyzed trifluoromethylation of Meyer-Schuster rearrangement. Org. Lett. 2014, 16, 1000-1003.
DOI: 10.1021/ol403741m. Publication Date: Jan. 27, 2014.
32. Daojuan Cheng, Yoshihiro Ishihara, Bin Tan*, Carlos F. BarbasIII*. Organocatalytic asymmetric assembly reactions: synthesis of spirooxindoles via organocascade Strategies. ACS Catal. 2014, 4, 743-762 (Invited Review Article).
DOI: 10.1021/cs401172r. Publication Date: Jan. 20, 2014.
31. Jin-Shun Lin, Ya-Ping Xiong, Can-Liang Ma, Li-Jiao Zhao, Bin Tan*, Xin-Yuan Liu*. Efficient copper-catalyzed direct intramolecular aminotrifluoromethylation of unactivated alkenes with diverse nitrogen-based nucleophiles. Chem. Eur. J. 2014, 20, 1332-1340.
DOI: 10.1002/chem.201303387. Publication Date: Dec. 20, 2013.
30. Lei Li, Min Deng, Sheng-Cai Zheng, Ya-Ping Xiong, Bin Tan*, Xin-Yuan Liu*. Metal-free direct intramolecular carbotrifluoromethylation of alkenes to functionalized trifluoromethyl azaheterocycles. Org. Lett. 2014, 16, 504-507.
DOI: 10.1021/ol403391v. Publication Date: Dec. 18, 2013.
Before SUSTech
29. Bin Tan, Xuan Zhang, Guofu Zhong*. Protecting-group directed stereospecific organocatalytic [3+2] cycloadditions: a facile access to chiral spirocyclic oxindoles. Source: Arkivoc Pages: 124-142 Published: 2014.
28. Klaus Albertshofer, Bin Tan, Carlos F. Barbas III*. Asymmetric Construction of Spirocyclopentenebenzofuranone Core Structures via Highly Selective Phosphine-Catalyzed [3+2] Cycloaddition Reactions. Org. Lett. 2013, 15, 2958.
27. Xianxing Jiang, Bin Tan, Carlos F. Barbas III*. Core-Structure-Motivated Design of Iminium-Enolate Organocascade Reactions: Enantioselective Syntheses of 5,6-Dihydroindolizines. Angew. Chem. Int. Ed. 2013, 52, 9261.
26. Klaus Albertshofer, Bin Tan, Carlos F. Barbas III*. Assembly of Spirooxindole Derivatives Containing Four Consecutive Stereocenters via Organocatalytic Michael-Henry Cascade Reactions. Org. Lett. 2012, 14, 1834.
25. Bin Tan, Xiaofei Zeng, Wendy Wen Yi Leong, Zugui Shi, Carlos F. Barbas III*, Guofu Zhong*. Core Structure-Based Design of Organocatalytic [3+2]-Cycloaddition Reactions: Highly Efficient and Stereocontrolled Syntheses of 3,3'-Pyrrolidonyl Spirooxindoles. Chem. Eur. J. 2012, 18, 63.
24. Gloria Hernández-Torres, Bin Tan, Carlos F. BarbasIII*. Organocatalysis as a Safe Practical Method for the Stereospecific Dibromination of Unsaturated Compounds. Org. Lett. 2012, 14, 1858.
23. Bin Tan, Narihiro Toda, Carlos F. Barbas III*. Organocatalytic Amidation and Esterification of Aldehydes with Activating Reagents by a Cross-Coupling Strategy. Angew. Chem. Int. Ed. 2012, 51, 12538.
22. Bin Tan, Gloria Hernández-Torres, Carlos F. Barbas III*. Rationally Designed Amide Donors for Organocatalytic Asymmetric Michael Reactions. Angew. Chem. Int. Ed. 2012, 51, 5381.
21. Bin Tan, Nuno R. Candeias, Carlos F. Barbas III. Construction of bispirooxindoles containing three quaternary stereocentres in a cascade using a single multifunctional organocatalyst. Nature Chem. 2011, 3, 473.
20. Bin Tan, Nuno R. Candeias, Carlos F. BarbasIII*. Core-Structure-Motivated Design of a Phosphine-Catalyzed [3+2] Cycloaddition Reaction: Enantioselective Syntheses of Spirocyclopenteneoxindoles. J. Am. Chem. Soc. 2011, 133, 4672.
19. Bin Tan, Gloria Hernández-Torres, Carlos F. BarbasIII*. Highly Efficient Hydrogen-Bonding Catalysis of the Diels-Alder Reaction of 3-Vinylindoles and Methyleneindolinones Provides Carbazolespirooxindole Skeletons. J. Am. Chem. Soc. 2011, 133, 12354.
18. Zugui Shi, Bin Tan, Wendy Wen Yi Leong, Xiaofei Zeng, Min Lu, Guofu Zhong*. Catalytic Asymmetric Formal [4+1] Annulation Leading to Optically Active cis-Isoxazoline N-Oxides. Org. Lett. 2010, 12, 5402.
17. Xiaofei Zeng, Kehan Ye, Min Lu, Pei Juan Chua, Bin Tan, Guofu Zhong*. Chiral Bronsted Acid Catalyzed Enantioselective Addition of alpha-Isocyanoacetamides to Aldehydes. Org. Lett. 2010, 12, 2414.
16. Zhen-Jiang Xu, Di Zhu, Xiaofei Zeng, Fei Wang, Bin Tan, Yuxuan Hou, Yunbo Lva, Guofu Zhong*. Diastereoselective HOTf-catalyzed three-component one-pot 1,3-dipolar cycloaddition of alpha-diazo ester, nitrosobenzene and electron-deficient alkene. Chem. Commun. 2010, 46, 2504.
15. Bin Tan, Yunpeng Lu, Xiaofei Zeng, Pei Juan Chua, Guofu Zhong*. Facile Domino Access to Chiral Bicyclo[3.2.1]octanes and Discovery of a New Catalytic Activation Mode. Org. Lett. 2010, 12, 2682.
14. Pei Juan Chua, Bin Tan, Limin Yang, Xiaofei Zeng, Di Zhua, Guofu Zhong*. Highly stereoselective synthesis of indanes with four stereogenic centers via sequential Michael reaction and [3+2] cycloaddition. Chem. Commun. 2010, 46, 7611.
13. Bin Tan, Di Zhu, Lihong Zhang, Pei Juan Chua, Xiaofei Zeng, Guofu Zhong*. Water-More Than Just a Green Solvent: A Stereoselective One-Pot Access to All-Chiral Tetrahydronaphthalenes in Aqueous Media. Chem. Eur. J. 2010, 16, 3842.
12. Pei Juan Chua, Bin Tan, Guofu Zhong*. Highly enantioselective L-thiaproline catalyzed α-aminoxylation of aldehydes in aqueous media. Green Chem. 2009, 11, 543.
11. Limin Yang, Bin Tan, Fei Wang, Guofu Zhong*. An Unexpected N-Heterocyclic Carbene-Catalyzed Annulation of Enals and Nitroso Compounds. Org. Chem. 2009, 74, 1744.
10. Min Lu, Di Zhu, Yunpeng Lu, Xiaofei Zeng, Bin Tan, Zhenjiang Xu, Guofu Zhong*. Chiral Bronsted Acid-Catalyzed Enantioselective alpha-Hydroxylation of beta-Dicarbonyl Compounds. J. Am. Chem. Soc. 2009, 131, 4562.
9. Pei Juan Chua, Bin Tan, Xiaofei Zeng, Guofu Zhong*. L-Prolinol as a highly enantioselective catalyst for Michael addition of cyclohexanone to nitroolefins. Bioorg. Med. Chem. Lett. 2009, 19, 3915.
8. Bin Tan, Xiaofei Zeng, Yunpeng Lu, Pei Juan Chua, Guofu Zhong*. Rational Design of Organocatalyst: Highly Stereoselective Michael Addition of Cyclic Ketones to Nitroolefins. Org. Lett. 2009, 11, 1927.
7. Bin Tan, Xuan Zhang, Pei Juan Chua, Guofu Zhong*. Recyclable organocatalysis: highly enantioselective Michael addition of 1,3-diaryl-1,3-propanedione to nitroolefins. Chem. Commun. 2009, 12, 779.
6. Bin Tan, Zugui Shi, Pei Juan Chua, Yongxin Li, Guofu Zhong*.Unusual Domino Michael/Aldol Condensation Reactions Employing Oximes as N-Selective Nucleophiles Synthesis of N-Hydroxypyrroles. Angew. Chem. Int. Ed. 2009, 48, 758.
5. Bin Tan, Pei Juan Chua, Xiaofei Zeng, Min Lu, Guofu Zhong*. A highly diastereo- and enantioselective synthesis of multisubstituted cyclopentanes with four chiral carbons by the organocatalytic domino Michael-Henry reaction. Org. Lett. 2008, 10, 3489.
4. Di Zhu, Min Lu, Pei Juan Chua, Bin Tan, Fei Wang, Xinhao Yang, Guofu Zhong*. A Highly Stereoselective Organocatalytic Tandem Aminoxylation/Aza-Michael Reaction for the Synthesis of Tetrahydro-1,2-Oxazines. Org. Lett. 2008, 10, 4585.
3. Bin Tan, Zugui Shi, Pei Juan Chua, Guofu Zhong*. Control of four stereocenters in an organocatalytic domino double Michael reaction: Efficient synthesis of multisubstituted cyclopentanes. Org. Lett. 2008, 10, 3425.
2. Min Lu, Di Zhu, Yunpeng Lu, Yuxuan Hou, Bin Tan, Guofu Zhong*. Organocatalytic Asymmetric alpha-Aminoxylation/Aza-Michael Reactions for the Synthesis of Functionalized Tetrahydro-1,2-oxazines. Angew. Chem. Int. Ed. 2008, 47, 10187.
1. Bin Tan, Pei Juan Chua, Yongxin Li, Guofu Zhong. Organocatalytic asymmetric tandem Michael-Henry reactions: A highly stereoselective synthesis of multifunctionalized cyclohexanes with two quaternary stereocenters. Org. Lett. 2008, 10, 2437.