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成果及论文

1. Xintong Wang+Haoran Xiao+Jing Wang+Zongze Huang,Geng Peng, Wenjun Xie, Xiling Bian, Huijie Liu, Cheng Shi, Taoyi Yang, Xin Li, Jian Gao, Ying Meng, Qianchen Jiang, Wei Chen,Fang Hu, Ningning Wei, Xiaowei Wang, Liangren Zhang, KeWei Wangand Qi SunSynthesis and biological evaluation of novel triazine derivatives as positive allosteric modulators of α7 nicotinic acetylcholine receptors. J. Med. Chem. 202164 (16)12379-12396;

2. 王佳杰王新童李远恒焦文宣肖浩然孙崎*王克威*用于改善认知障碍的靶向α7型尼古丁乙酰胆碱受体正向变构调节剂的研发现状,《药学进展》(药咖论坛),202044(8), 573-587;

3. Yuanheng Li+, Lilan Sun+, Taoyi Yang+, Wenxuan Jiao, Jingshu Tang, Xiaomin Huang, Zongze Huang, Ying Meng, Laichun Luo, Xintong Wang, Xiling Bian, Fang Zhang, KeWei Wang* and Qi Sun*The design and synthesis of novel positive allosteric modulators of α7 nicotinic acetylcholine receptors with the ability to rescue auditory gating deficit in mice. J. Med. Chem. 201962, 159-173;

4. Xin Li+, Wenjun Xie+, Xintong Wang, Zongze Huang, Xiling Bian, KeWei Wang* and Qi Sun* Chemical conversion of nicotinamide into type I positive allosteric modulator of α7 nAChRsBioorg. Med. Chem. Lett. 201929, 1928-1933;

5. Jiao Gong, Yuanheng Li, Chanjuan Zhang, Jian Huang* and Qi Sun* A thiazolo[4,5-b]pyridine-based fluorescent probe for detection of zinc ions and application for in vitro and in vivo bioimaging. Talanta 2018185, 396-404;

6. Wenxing Zou, Zongze Huang, Kang Jiang, You Wu, Yuqing Xue, Franck Suzenet*, Qi Sun*, Gerald Guillaumet Chelation-assisted C-S activation/cascade heteroannulation of pyridine-2-thione derivatives in Pd-catalyzed cross-coupling reaction with alkynes. Tetrahedron 201773, 5485-5492;

7. Songwen Lin+, Yingbo Li+, Yufen Zheng, Laichun Luo, Qi Sun*, Zemei Ge, Tieming Cheng and Runtao Li* Design, synthesis and biological evaluation of quinazoline–phosphoramidate mustard conjugates as anticancer drugs. Eur. J. Med. Chem. 2017127, 442-458;

8.  Dan Wan, Ding Wang, Qi Sun, Yan Song, Yimin Jiang, Runtao Li, Jia YeAntinociception of spirocyclopiperazinium salt compound LXM-10-M targeting α7 nicotinic receptor and M4 muscarinic receptor and inhibiting CaMKIIα/CREB/CGRP signaling pathway in mice. Eur. J. Pharmacol. 2016770, 92-98;

9. Yufen Zheng, Wenxing Zou, Laichun Luo, Jiabei Chen, Songwen Lin and Qi Sun*Ligand-free Cu-catalyzed O-arylation of aliphatic diols. RSC Adv. 20155, 66104-66108;

10. You Wu, Yongning Xing, Jie Wang, Qi Sun*, Weiqi Kong, and Franck Suzenet Palladium-catalyzed desulfurative Sonogashira cross-coupling reaction of 3-cyano assisted thioamide-type quinolone derivatives with alkynes. RSC Adv. 20155, 48558-48562;

11. Dongmei Xiao, Liqiang Han, Qi Sun*, Qianxi Chen, Ningbo Gong, Yang Lv, Franck Suzenet, Gérald Guillaumet, Tieming Cheng and Runtao Li* Copper-mediated synthesis of N-fused heterocycles via Csp-S coupling reaction and 5-endo-dig cyclization sequence. RSC Adv. 20122, 5054-5057;

12. Qi Sun, Franck Suzenet* and Gérald Guillaumet Optimized Liebeskind-Srogl coupling reaction between dihydropyrimidines and tributyltin compounds. Tetrahedron Lett. 201253, 2694-2698;

13. Qi Sun, Franck Suzenet* and Gérald Guillaumet Desulfitative cross-coupling of protecting group-free 2-thiouracil derivatives with organostannanes. J. Org. Chem. 201075, 3473-3476.