2024年文章
[1] Xiaohua Luo, Wei Mao, Chen-Fei Liu, Yu-Qi Wang, Jing Nie,* Shi-Liang Shi,* Jun-An Ma*& Ming Joo Koh*. Enantioselective synthesis of multifunctional alkylboronates via N-heterocyclic carbene-nickel-catalysed carboboration of alkenes. Nature Synthesis. 2024. 3, 633-642, DOI: 10.1038/s44160-024-00492-x 
[2] Xiaodong Tang, Ming-Yue He, Ran Guo, Hao-Nan Liu, Jing Nie, Ilan Marek, Jun-An Ma and Fa-Guang Zhang*. The Smallest Monofluorodiazoethane Reagent and Its [3 + 2] Cycloaddition Reactions. CCS Chem. 2024. 6, 2825-2834. DOI: 10.31635/ccschem.024.202403849
[3] Ze-Long Mei, Cong-Cong Li, Xu Han, Yu-Chen Tian, Shuo-Han Li, Weidong Liu, Ge Qu, Manfred T. Reetz, Zhoutong Sun,* Jun-An Ma,* and Fa-Guang Zhang*. Enzymatic Stereodivergent Access to Fluorinated β‑Lactam Pharmacophores via Triple-Parameter Engineered Ketoreductases. ACS Catal. 2024, 14, 6358-6368. DOI: 10.1021/acscatal.4c00945
[4] Weimin Xuan*and Jun-An Ma*. Pinpointing Acidic Residues in Proteins. ChemMedChem. 2024, 19, e202300623. DOI: 10.1002/cmdc.202300623.
[5] Xinyi Li, Fa-Guang Zhang, Jun-An Ma,* and Yongjun Liu*. Computational insights into the binding modes, keto-enol tautomerization and stereo-electronically controlled decarboxylation of oxaloacetate in the active site of Macrophomate synthase. Phys. Chem. Chem. Phys. 2024, 26, 12331-12344. DOI: 10.1039/D4CP00716F.
[6] Haonan Liu, Jianxu Chen, Zan Yang, Liuyin Jiang, Wenya Liu, Jun-An Ma,* and Saihu Liao*. Light-Controlled Cationic RAFT Polymerization of Vinyl Ethers Using N‑Arylacridinium photocatalysts. Macromolecules, 2024. 57, 8, 3751-3756. DOI: 10.1021/acs.macromol.4c00265.
[7] Xiaodong Tang, Yang-Dong Hou, Xing-Fa Tan, Jing Nie,* Chi Wai Cheung,* and Jun-An Ma*. Synergistic Catalytic Asymmetric Decarboxylative Mannich Reaction of β‑Ketoacids with Acyclic α‑Arylenamides. ACS Catal. 2024, 14, 9701-9707. DOI: 10.1021/acscatal.4c02238
Highlighted by Benjamin List in Synfacts 2024, 20(09), 0977.
[8] Rong Wang, Jing Nie,* Xiaojuan Deng, Guosheng Ding, Fa-Guang Zhang,*and Jun-An Ma*. Regioselective Synthesis of Multisubstituted Fluoropyrazoles via Silver-Catalyzed One-Pot Cyclization Reaction of Diazo Reagents with Fluoronitroalkenes. Adv. Synth. Catal. 2024, 366, 3516-3521. DOI: 10.1002/adsc.202400385
[9] Nicolas Marie, Jun-An Ma, Vincent Tognetti, and Dominique Cahard*. Photocatalyzed Cascade Hydrogen Atom Transfers for Assembly of Multi-Substituted α-SCF3 and α-SCF2H Cyclopentanones. Angew. Chem. Int. Ed. 2024, e202407689. DOI: 10.1002/anie.202407689.
[10] Shuo-Han Li, Xue Zhang, Ze-Long Mei, Yongjun Liu,* Jun-An Ma,* and Fa-Guang Zhang*. Chemoenzymatic Synthesis of Fluorinated Mycocyclosin Enabled by the Engineered Cytochrome P450-Catalyzed Biaryl Coupling Reaction. J. Am. Chem. Soc. 2024, 146, 19962-19973. DOI: 10.1021/jacs.4c03499
[11] Hao-Yan Wu, Xiaodong Tang,* Ran Guo, Hwee Ting Ang, Jing Nie, Jie Wu, Jun-An Ma,* and Fa-Guang Zhang*. Catalytic photoactivation of a triarylamine electron donor-acceptor complex for difunctionalization of alkenes. Cell Reports Physical Science. 2024. 5, 102135. DOI: 10.1016/j.xcrp.2024.102135
[12] Haibin Li, Zhiheng Sun, Yue Liu, Yi Xing, Jing Gao, Aihong Shi, Yadong Yu, Jin Long, Dong‐Po Song, Chao Jin, Marc D. McKee*, Jun‐An Ma*, Wenge Jiang.* Chiral gypsum with high‐performance mechanical properties induced by self‐assembly of chiral amino acid on an amorphous mineral. SmartMat. 2024. e1302. DOI:10.1002/smm2.1302.
[13] Yuying Zhang, Kanghui Song, Tongtong Wang, Shuai Wu, Gang Xu, Saihu Liao, Jun-An Ma,* and Yuanming Li*. The Synthesis and Properties of Spirophenanthrene. J. Org. Chem. 2024, 89, 12044-12048. DOI: 10.1021/acs.joc.4c00782
[14] Hao Zeng, Ruize Yin, Yu Zhao, Jun-An Ma* & Jie Wu*. Modular alkene synthesis from carboxylic acids, alcohols and alkanes via integrated photocatalysis. Nature Chemistry. 2024. 16, 1822-1830. DOI: 10.1038/s41557-024-01642-6
[15] Xin-Yi Shi, Xueyuan Yan, Xiaodong Tang, Shi-Jing Zhai, Genping Huang*, Jun-An Ma* and Fa-Guang Zhang.* Nickel-catalysed enantioselective crosselectrophile coupling reaction with the retention of the β-fluorine atom. Org. Chem. Front. 2024, 11, 6459-6469. DOI: 10.1039/d4qo01555j
[16] Ting Zhou, Zhong-Wei Zhang, Jing Nie, Fuk Yee Kwong, Jun-An Ma* & Chi Wai Cheung*. Metallaphotocatalytic triple couplings for modular synthesis of elaborate N-trifluoroalkyl anilines. Nat. Commun. 2024, 15, 9926. DOI: 10.1038/s41467-024-53828-8
[17] Meng-Qi Sun, Shi-Jing Zhai, Jing Nie, Ying Cheng, Xiaojuan Deng, Guosheng Ding, Dominique Cahard, Jun-An Ma,* and Fa-Guang Zhang*. Allylation, Alkenylation and Alkynylation of Monofluoromethyl Ketyl Radical Enabled by Photoredox Halogen-Atom-Transfer. ChemCatChem. 2024, 0, e202401622. DOI: 10.1002/cctc.202401622
[18] 吴昊岩, 赫明月, 马军安, 张发光. 三芳胺在光催化反应中的研究进展. Chin. J. Org. Chem. 2024, 44. DOI: 10.6023/cjoc202408009
[19] Wiktor K. Poper, Jun-An Ma,* and Marcin Jasiński*. One-Pot Telescoping S‑Transfer and Trifluoromethylation for the Synthesis of 2‑CF3S‑Imidazoles with N‑Oxides as Convenient
Precursors. J. Org. Chem. 2024, 89, 15331-15335. DOI: 10.1021/acs.joc.4c01761
[20] Chi Liu, Yang Yang, Wenyang Hong, Jun-An Ma* and Ye Zhu*. Ion Hydration Enables Generality in Asymmetric Catalysis: Desymmetrization to P-Stereogenic Triarylphosphine Derivatives. Angew. Chem. Int. Ed. 2024, e202417827. DOI: 10.1002/anie.202417827
2023年文章
[1] Ye Yuan, Muliang Zhang, Xiaodong Tang, Jared L. Piper, Zhi-Hui Peng, Jun-An Ma,* Jie Wu,* and Fa-Guang Zhang*. Photoinduced Defluorinative Branch-Selective Olefination of Multifluoro (Hetero)arenes. Org. Lett. 2023, 25, 883-888. DOI: 10.1021/acs.orglett.3c00115
[2] Yue-Ji Chen, Jie Zheng, Jun-An Ma * , Fa-Guang Zhang *. Radical-initiated diazo-retaining nucleophilic addition reaction of trifluorodiazoethane and diazoacetate with 2H‑azirines. Journal of Fluorine Chemistry. 2023, 268, 110129. DOI: 10.1016/j.jfluchem.2023.110129
[3] Meng Li, Jun-An Ma, and Saihu Liao*. Atom-Transfer Radical Polymerization of a SuFExable Vinyl Monomer and Polymer Library Construction via SuFEx Click Reaction. Macromolecules. 2023, 56, 806-814. DOI: 10.1021/acs.macromol.2c01492.
[4] Guangrong Wang, Hui Shao, Jun-An Ma, and Saihu Liao*. Chalcogenide-Doped Anthracenes as Organophotocatalysts for Metal-Free Atom Transfer Radical Polymerization. Macromol. Chem. Phys. 2023, 224, 2200382. DOI: 10.1002/macp.202200382
[5] Jun-Hao Zhang, Hui Xu, Xiaodong Tang, Yanfeng Dang, * Fa-Guang Zhang * and Jun-An Ma*. Highly Enantio- and Diastereoselective Hydrogenation of Cyclic Tetra-Substituted β-Enamido Phosphorus Derivatives. Angew. Chem. Int. Ed. 2023, e202305315. DOI: 10.1002/anie.202305315
[6] Xuan-Yu Liu, Yi-Lin Yang, Yanfeng Dang, Ilan Marek, * Fa-Guang Zhang, * and Jun-An Ma*. Tetrazole Diversification of Amino Acids and Peptides via Silver-Catalyzed Intermolecular Cycloaddition with Aryldiazonium Salts. Angew. Chem. Int. Ed. 2023, e202304740. DOI: 10.1002/anie.202309192
[7] Nan Zhang, Hai Ma, Chi Wai Cheung, Fa-Guang Zhang, Marcin Jasiński, Jun-An Ma * and Jing Nie *. Regioselective [3 + 2] cycloaddition of di/trifluoromethylated hydrazonoyl chlorides with fluorinated nitroalkenes: a facile access to 3-di/trifluoroalkyl-5-fluoropyrazoles. Org. Biomol. Chem. 2023, 21, 5040-5045. DOI: 10.1039/d3ob00644a
[8] Xiu-Qing Cui, Meng-Meng Zheng, Xiaodong Tang, Zhi-Qi Zhang, Xiao-Song Xue, Ilan Marek, * Jun-An Ma, * and Fa-Guang Zhang*. Dirhodium(II)-catalyzed enantioselective cyclopropenation of internal alkynes with trifluoromethyl carbene. Chem. Catal. 2023, 3, 100637. DOI: 10.1016/j.checat.2023.100637
[9] Jie Zheng, Meng-Yu Rong, Fang-Fang Feng, Fa-Guang Zhang,* Chi Wai Cheung,* and Jun-An Ma*. Organocatalyst-Controlled Divergent Asymmetric Aza-Friedel-Crafts Reactions of Indol-3-ones with 1- and 2-Naphthols. Asian J. Org. Chem. 2023, e202300204. DOI: 10.1002/ajoc.202300204
[10] Tongtong Zheng, Zhe Feng, Jun-An Ma,* and Chi Wai Cheung.* Dual Nickel/Photoredox-Catalyzed Synthesis of N-formyl N,N’-Diaryl Ethylenediamines via Multiple C-N/C-C Coupling of Nitroarenes with Trimethylamine. Adv. Synth. Catal. 2023, 365, 2377-2384. DOI: 10.1002/adsc.202300431
[11] 秦沛, 马海, 张发光*, 马军安*. 含三氟甲基三氮嗪酪氨酸激酶抑制剂设计合成及生物活性研究. Acta Chim. Sinica, 2023, 81, 7, 697-702. DOI: 10.6023/A23040154
[12] Kamil Świątek, Greta Utecht-Jarzyńska, Marcin Palusiak, Jun-An Ma,* and Marcin Jasiński*. One-Pot Synthesis of 1‑Aryl-3-trifluoromethylpyrazoles Using Nitrile Imines and Mercaptoacetaldehyde As a Surrogate of Acetylene. Org. Lett. 2023, 25, 4462-4467. DOI: 10.1021/acs.orglett.3c01437
[13] Zhong-Wei Zhang, Zhe Feng, Jun-An Ma* & Chi Wai Cheung.* Metallaphotocatalytic synthesis of anilines through tandem C–N transposition and C–H alkylation of alkylamines. Nature Synthesis. 2023, 2, 1171-1183. DOI: 10.1038/s44160-023-00370-y
[14] Cheng-Feng Gao, Yue-Ji Chen, Jing Nie, Fa-Guang Zhang*, Chi Wai Cheung*, and Jun-An Ma*. Synthesis of di/trifluoromethyl cyclopropane-dicarbonitriles via [2 + 1] annulation of fluoro-based diazoethanes with (alkylidene)malononitriles. Chem. Commun. 2023, 59, 11664-11667. DOI: 10.1039/d3cc03897a
[15] Jing Gao, Haibin Li, Zhiheng Sun, Jianwei Song, Yue Liu, Chao Jin, Zhisen Zhang,* Jun-An Ma, and Wenge Jiang*. Selective Chiral Recognition between Amino Acids and Growing Gypsum Crystals. ACS Langmuir. 2023, 39, 36, 12707-12714. DOI: 10.1021/acs.langmuir.3c01429
[16] Dan Wang, Yu-Ting Tian, Jing Nie, Marcin Jasiński,* Xiaodong Tang,*and Jun-An Ma.* Traceless Directing Group Enabled One-Pot Regiospecific Synthesis of 2,3-Diaryl-4-Fluoropyrroles. Adv. Synth. Catal. 2023, 365, 1-6. DOI: 10.1002/adsc.202300625
[17] Xiaochen Yang, Lei Zhao, Ying Wang, Yanli Ji, Xun-Cheng Su, Jun-An Ma, and Weimin Xuan*. Constructing Photoactivatable Protein with Genetically Encoded Photocaged Glutamic Acid. Angew. Chem. Int. Ed. 2023, e202308472. DOI: 10.1002/anie.202308472
[18] Tao-Qian Zhao, Hui Xu, Yu-Chen Tian, Xiaodong Tang, Yanfeng Dang, Shaozhong Ge,* Jun-An Ma,* and Fa-Guang Zhang*. Copper-Catalyzed Regio- and Enantioselective Hydroboration of Difluoroalkyl-Substituted Internal Alkenes. Adv. Sci. 2023, 2304194. DOI: 10.1002/adsc.202300625
[19] Zhi-Qi Zhang, Cheng-Qiang Wang, Long-Ji Li, Jared L. Piper, Zhi-Hui Peng,* Jun-An Ma, * Fa-Guang Zhang * and Jie Wu *. Programmable synthesis of difluorinated hydrocarbons from alkenes through a photocatalytic linchpin strategy. Chem. Sci. 2023, 14, 11546. DOI: 10.1039/d3sc03951j
[20] Shuo-Han Li, Ran Guo, Ning Lv, Yu Liu,* Xiaodong Tang,* Jun-An Ma*. Regioselective [3 + 2] cycloaddition of diazo reagents and internal alkynes: Accessing regiosomers of highly substituted trifluoromethylpyrazoles. Journal of Fluorine Chemistry. 2023, 272, 110216.
DOI: 10.1016/j.jfluchem.2023.110216.
[21] Meng-Yu Rong , Jing Nie , Shen Li *, Jun-An Ma *. Enantioselective synthesis of fluorinated aromatic amino acids catalyzed by SPINOL-derived chiral quaternary ammonium salts. Molecular Catalysis, 2024, 552, 113679. DOI: 10.1016/j.mcat.2023.113679
[22] Lu-Nan Zhou, Chi Wai Cheung *, Junan Ma* . Base-promoted [3 + 2] Annulation of Carbodiimides with Diazoacetonitrile for Synthesis of 5-Amino-4-Cyano-1,2,3-triazoles. Synlett, 2024, 35, 13, 1557-1560. DOI: 10.1055/a-2216-4765.
[23] Ming-Yue He, Xiaodong Tang,* Hao-Yan Wu, Jing Nie, Jun-An Ma,* and Fa-Guang Zhang*. Electron Donor−Acceptor Complex Enabled Radical Cyclization of α‑Diazodifluoroethyl Sulfonium Salt with Unactivated Alkynes. Org. Lett. 2023, 25, 50, 9041-9046. DOI: 10.1021/acs.orglett.3c03790
2022年文章
[1] Feng-Ling Qing,* Xin-Yuan Liu,* Jun-An Ma,* Qilong Shen,* Qiuling Song,* Pingping Tang*. A Fruitful Decade of Organofluorine Chemistry: New Reagents and Reactions. CCS Chem. 2022, 4, 2518-2549. DOI: 10.31635/ccschem.022.202201935.
[2] Xuan-Yu Liu, Fa-Guang Zhang,* Jun-An Ma*. Regioselective Construction of Coumarin-1,2,4-triazines via a Cs2CO3-Catalyzed [3+3] Cycloaddition Reaction. Synlett. 2022, 3(11): 1097-1101. DOI: 10.1055/a-1828-7504
[3] Cheng-Feng Gao, Yin Zhou, Hai Ma, Yue Zhang, Jing Nie, Fa-Guang Zhang* & Jun-An Ma*. Dual Incorporation of Trifluoromethyl and Cyano Groups into Pyrazole Pharmcophores via Silver-Catalyzed Cycloaddition Reaction of Trifluorodiazoethane. CCS Chem. 2022, 4, 3693-3704. DOI: 10.31635/ccschem.022.202201923
[4] Xue-Qi Wang, Fang-Fang Feng, Jing Nie, Fa-Guang Zhang,* and Jun-An Ma*. Enantioselective Construction of Amino Carboxylic-Phosphonic Acid Derivatives Enabled by Chiral Amino Thiourea-Catalyzed Decarboxylative Mannich Reaction. Adv. Synth. Catal. 2022, 364, 1-6. DOI: 10.1002/adsc.202200306
[5] Yin Zhou, Cheng-Feng Gao, Hai Ma, Jing Nie,* Jun-An Ma,* and Fa-Guang Zhang*. Quadruple Functionalized Pyrazole Pharmacophores by One-pot Regioselective [3+2] Cycloaddition of Fluorinated Nitrile Imines and Dicyanoalkenes. Chem Asian J. 2022, e202200436. DOI: 10.1002/asia.202200436
[6] Zhe Feng, Jun-An Ma* and Chi Wai Cheung*. Ni-Catalysed intramolecular reductive aminocarbonylation of 2-haloaryl-tethered nitroarenes for the synthesis of dibenzazepine-based heterocycles. Org. Chem. Front., 2022, 9, 3869-3875. DOI: 10.1039/d2qo00699e
[7] Zhi-Qi Zhang, Yue-Qian Sang, Cheng-Qiang Wang, Peng Dai, Xiao-Song Xue, Jared L. Piper, Zhi-Hui Peng, Jun-An Ma,* Fa-Guang Zhang,* and Jie Wu*. Difluoromethylation of Unactivated Alkenes Using Freon-22 through Tertiary Amine-Borane-Triggered Halogen Atom Transfer. J. Am. Chem. Soc. 2022. 144, 14288-14296. DOI: 10.1021/jacs.2c05356
[8] Conghui Ren, Qifan Wu, Ruotong Xiao, Yanli Ji, Xiaochen Yang, Zhuo Zhang, Hongqiang Qin, Jun-An Ma, Weimin Xuan*. Expanding the Scope of Genetically Encoded Lysine PTMs with Lactylation, β-Hydroxybutyrylation and Lipoylation. ChemBioChem. 2022, e202200302. DOI: 10.1002/cbic.202200302
[9] Nicolas Marie, Jun-An Ma, and Dominique Cahard*. Amphiphilic Polyfluorinated Amino Ethers from Cyclic Sulfamidates. J. Org. Chem. 2022, 87, 24, 16665–16675. DOI：10.1021/acs.joc.2c02337
[10] Xing Peng, Meng-Meng Zheng, Pei Qin, Xiao-Song Xue,* Fa-Guang Zhang* and Jun-An Ma*. Silver-catalysed [3 + 2] annulation reaction of aryldiazonium salts with allenes enabled by boronate direction. Org. Chem. Front. 2022, 10,74–82. DOI: 10.1039/d2qo01585d
[11] Jun-Kuan Li, Ge Qu, Xu Li, Yuchen Tian, Chengsen Cui, Fa-Guang Zhang, Wuyuan Zhang, Jun-An Ma,* Manfred T. Reetz* & Zhoutong Sun*. Rational enzyme design for enabling biocatalytic Baldwin cyclization and asymmetric synthesis of chiral heterocycles. Nat. Commun. 2022, 13, 7813. DOI：10.1038/s41467-022-35468-y
2021年文章
[1] Yu-Ting Tian, Fa-Guang Zhang,* and Jun-An Ma*. Et3N-catalyzed direct cycloaddition reaction of allenoates with acceptor diazo compounds. Tetrahedron. 2021, 81, 131922. DOI: 10.1016/j.tet.2021.131922
[2] Yu-Ting Tian, Fa-Guang Zhang,* and Jun-An Ma*, Regioselective [3 + 2] Cycloaddition Reaction of 3‑Alkynoates with Seyferth−Gilbert Reagent. J. Org. Chem. 2021, 86, 3574-3582. DOI: 10.1021/acs.joc.0c02957
[3] Lu-Nan Zhou, Fang-Fang Feng, Chi Wai Cheung,* and Jun-An Ma*. Cu-Enabled [3 + 2] Annulation of In Situ Formed Nitrile Ylides with Aryldiazonium Salts: Access to 5‑Cyano-1,2,4-Triazoles. Org. Lett. 2021, 23, 739-744. DOI: 10.1021/acs.orglett.0c03960
[4] Hao-Qiang Cao, Jun-Kuan Li, Fa-Guang Zhang,* Dominique Cahard,* and Jun-An Ma*. Asymmetric Synthesis of Chiral Amino Carboxylic-Phosphonic Acid Derivatives. Adv. Synth. Catal. 2021, 363, 688-729. DOI: 10.1002/adsc.202001345
[5] Yu-Chen Tian, Jun-Kuan Li, Fa-Guang Zhang,* and Jun-An Ma*. Regioselective Decarboxylative Cycloaddition Route to Fully Substituted 3-CF3-Pyrazoles from Nitrilimines and Isoxazolidinediones. Adv. Synth. Catal. 2021, 363, 2093-2097. DOI: 10.1002/adsc.202100091
[7] Fang-Fang Feng, Xuan-Yu Liu, Chi Wai Cheung,* and Jun-An Ma*. Tungsten-Catalyzed Transamidation of Tertiary Alkyl Amides. ACS Catal. 2021, 11, 7070-7079. DOI: 10.1021/acscatal.1c01840
[8] 彭星, 张发光*, 马军安*.芳香重氮盐参与的协同环加成反应.Univ. Chem. 2021, 36 (X), 2101026 (2 of 5). DOI: 10.3866/PKU.DXHX202101026
[9] 张发光*， 曲戈*，孙周通*，马军安*. 从化学合成到生物合成—天然产物全合成新趋势. DOI: 10.12211/2096-8280.2021-039
[10] Shi-Jing Zhai, Fa-Guang Zhang*, Jun-An Ma*. Metal-free regioselective construction of 2-aryl-2H-tetrazol-5-yl diflfluoromethylene phosphonates. Chin. Chem. Lett. 2021, 32, 863-866. DOI: 10.1016/j.cclet.2021.08.007
[11] Fa-Guang Zhang,* Zhen Chen, Xiaodong Tang, and Jun-An Ma*. Triazines: Syntheses and Inverse Electron-demand Diels−Alder Reactions. Chem. Rev. 2021. 121, 14555-14593. DOI: 10.1021/acs.chemrev.1c00611
[12] Fang-Fang Feng, Jun-An Ma,* and Dominique Cahard*. Radical 1,5-Chloropentaflfluorosulfanylation of Unactivated Vinylcyclopropanes and Transformation into α‑SF5 Ketones. J. Org. Chem. 2021, 86, 19, 13808-13816. DOI: 10.1021/acs.joc.1c01886
[13] Yue-Ji Chen, Fa-Guang Zhang,* and Jun-An Ma*. Zinc-Enabled Annulation of Triflfluorodiazoethane with 2H‑Azirines to Construct Triflfluoromethyl Pyrazolines, Pyrazoles, and Pyridazines. Org. Lett. 2021, 23, 6062-6066. DOI: 10.1021/acs.orglett.1c02139
[14] 黄音君, 李金山, 李 珅*, 马军安*. 钴催化 2-芳基吲哚氧化去芳构化及与烯酰胺[3＋2]环化反应. Chin. J. Org. Chem. 2021, 41, 4028-4038. DOI: 10.6023/cjoc202104057
[15] Yi-Lin Yang, Shen Li, Fa-Guang Zhang*, Jun-An Ma.* N‑Iodosuccinimide-Promoted [3 + 2] Annulation Reaction of Aryldiazonium Salts with Guanidines To Construct Aminotetrazoles. Org. Lett. 2021, 23, 8894-8898. DOI: 10.1021/acs.orglett.1c03395
[16] Hong-Song Shi, Shuo-Han Li, Fa-Guang Zhang *, and Jun-An Ma.* Catalytic regioselective construction of phenylthio- and phenoxyldifluoroalkyl tetrazoles from difluorodiazoketones. Chem. Commun. 2021, 57, 13744-13747. DOI: 10.1039/d1cc05890h
2020年文章
[1] Shi-Jing Zhai, Xing Peng, Fa-Guang Zhang,* and Jun-An Ma*. Catalytic Direct Regioselective Synthesis of Phosphonylated Tetrazoles from Aryl Diazonium Salts and Seyferth-Gilbert Reagent. Org. Lett. 2019, 21, 9884-9888. DOI: 10.1021/acs.orglett.9b03800
[2] Xing-Fa Tan, Fa-Guang Zhang* and Jun-An Ma*. Asymmetric synthesis of CF2-functionalized aziridines by combined strong Brønsted acid catalysis. Beilstein J. Org. Chem. 2020, 16, 638-644. DOI: 10.3762/bjoc.16.60
[3] Hao-Nan Liu, Hao-Qiang Cao, Chi Wai Cheung* and Jun-An Ma*. Cu-Mediated Expeditious Annulation of Alkyl 3-Aminoacrylates with Aryldiazonium Salts: Access to Alkyl N2-Aryl 1,2,3-Triazole-carboxylates for Druglike Molecular Synthesis. Org. Lett. 2020, 22, 1396-1401. DOI: 10.1021/acs.orglett.0c00006
[4] Ming-Yang Xiao, Zhen Chen, Fa-Guang Zhang,* Jun-An Ma*. Regioselective synthesis of carboxylic and fluoromethyl tetrazoles enabled by silver-catalyzed cycloaddition of diazoacetates and aryl diazonium salts. Tetrahedron. 2020, 76, 131063. DOI: 10.1016/j.tet.2020.131063
[5] Hao-Qiang Cao, Hao-Nan Liu, Zhe-Yuan Liu, BaoKun Qiao, Fa-Guang Zhang,* Jun-An Ma*. Direct Enamido C(sp2)−H Diphosphorylation Enabled by a PCET‐Triggered Double Radical Relay: Access to gem-Bisphosphonates. Chem. Eur. J. 2020, 26, 5515-5521. DOI: 10.1002/chem.202000517
[6] Yue Zhang, Jun-Kuan Li, Fa-Guang Zhang* and Jun-An Ma*. Catalytic Asymmetric Access to Noncanonical Chiral α-Amino Acids from Cyclic Iminoglyoxylates and Enamides. J. Org. Chem. 2020, 85, 5580-5589. DOI: 10.1021/acs.joc.0c00436
[7] Junliang Zeng, Zhihonga Xu, Jun-An Ma*. Construction of 3,4-Disubstituted-3-(difluoromethyl)pyrazoles. Chin. J. Org. Chem. 2020, 40, 1105-1116. DOI: 10.6023/cjoc201912024
[8] Zelong Mei, Kun Zhang, Ge Qu, Jun-Kuan Li, Baoyan Liu, Jun-An Ma*, Ran Tu*, and Zhoutong Sun*. High-Throughput Fluorescence Assay for Ketone Detection and Its Applications in Enzyme Mining and Protein Engineering. ACS Omega. 2020. DOI: 10.1021/acsomega.0c00245
[9] Yin-Jun Huang, Jing Nie, Chi Wai Cheung,* Jun-An Ma*. Silver-Catalyzed [3+3] Annulation of Glycine Imino Esters with Seyferth–Gilbert Reagent To Access Tetrahydro-1,2,4-triazinecarboxylate Esters. Synlett. 2020, 31, 1107-1111. DOI: 10.1055/s-0039-1690894
[10] Fa-Guang Zhang*, Zhen Chen，Chi Wai Cheung* and Jun-An Ma*. Aryl Diazonium Salt-Triggered Cyclization and Cycloaddition Reactions: Past, Present, and Future. Chin.J. Chem. 2019, 37, 1132-1152. DOI: 10.1002/cjoc.202000270
[11] Fang-Fang Feng, Jun-Kuan Li, Xuan-Yu Liu, Fa-Guang Zhang,* Chi Wai Cheung,* and Jun-An Ma*. General Synthesis of Tri-Carbo-Substituted N2‑Aryl-1,2,3-triazoles via Cu-Catalyzed Annulation of Azirines with Aryldiazonium Salts. J. Org. Chem. 2020, 85, 10872-10883. DOI: 10.1021/acs.joc.0c01433
[12] Hao-Qiang Cao, Hao-Nan Liu, Zhe-Yuan Liu, Baokun Qiao, Fa-Guang Zhang,* and Jun-An Ma*. Silver-Promoted Direct Phosphorylation of Bulky C(sp2)−H Bond to Build Fully Substituted β‑Phosphonodehydroamino Acids. Org. Lett. 2020, 22, 6414-6419. DOI: 10.1021/acs.orglett.0c02229
[13] Xing Peng, Fa-Guang Zhang,* and Jun-An Ma*. Cu-Catalysed Three-Component Reaction of Aryldiazonium Salts with Fluorinated Diazo Reagents and Nitriles: Access to Difluoroand Trifluoromethylated N1-Aryl-1,2,4-triazoles. Adv. Synth. Catal. 2020, 362, 4432–4437. DOI: 10.1002/adsc.202000776
[14] Xuan-Yu Liu, Shi-Jing Zhai, Fang-Fang Feng, Fa-Guang Zhang,* and Jun-An Ma*. Silver-Catalyzed [3 + 2] Cycloaddition Approach to CoumarinDecorated Tetrazoles. ChemCatChem. 2020. 12, 5623–5626. DOI: 10.1021/acs.orglett.9b01697
[15] Fa-Guang Zhang,* Xue-Qi Wang, Yin Zhou, Hong-Song Shi, Zhe Feng, Jun-An Ma,* and Ilan Marek*. Remote Fluorination and Fluoroalkyl(thiol)ation Reactions. Chem. Eur. J. 2020. 26, 15378–15396. DOI: 10.1002/chem.202003416
[16] Jia-Pan Niu, Jing Nie, Shen Li * and Jun-An Ma*. Organocatalytic asymmetric synthesis of b,b-diaryl ketones via one-pot tandem dehydration/1,6-addition/decarboxylation transformation of b-keto acids and 4-hydroxybenzyl alcohols. Chem. Commun., 2020, 56, 8687-8690. DOI: 10.1039/d0cc02213f
[17] Ni Shen, Shi-Jing Zhai, Chi Wai Cheung * and Jun-An Ma *. Direct N-formylation of nitroarenes with CO2. Chem. Commun., 2020, 56, 9620-9623. DOI: 10.1039/d0cc03098h
[18] Wenge Jiang*, Xing Yi and Marc D. McKee*. Chiral biomineralized structures and their biomimetic synthesis. Mater. Horiz. 2019, 6, 1974-1990. DOI: 10.1039/c9mh00431a
[19] Wenge Jiang, Gabriele Griffanti , Faleh Tamimi, Marc D. McKee, Showan N. Nazhat. Multiscale structural evolution of citrate-triggered intrafibrillar and interfibrillar mineralization in dense collagen gels. Journal of Structural Biology, 2020, 212, 107592. DOI:10.1016/j.jsb.2020.107592
[20] Ming-Yang Xiao, Meng-Meng Zheng, Xing Peng, Xiao-Song Xue, Fa-Guang Zhang*, and Jun-An Ma*. Catalytic Direct Construction of Cyano-tetrazoles. Org. Lett. 2020, 22, 7762-7767. DOI: 10.1021/acs.orglett.0c03025
[21] Yu-Ting Tian, Fa-Guang Zhang, Jing Nie, Chi Wai Cheung *, and Jun-An Ma *. Metal-free Decarboxylative Annulation of 2-Aryl-2-isocyanoacetates with Aryldiazonium Salts: General Access to 1,3-Diaryl-1,2,4-triazoles. Adv. Synth. Catal. 2020, 363, 227-233. DOI: 10.1002/adsc.202001016
[22] Hongyue Wang, Ge Qu, Jun-Kuan Li, Jun-An Ma, Jinggong Guo,Yuchen Miaod and Zhoutong Sun*. Data mining of amine dehydrogenases for the synthesis of enantiopure amino alcohols. Sci. Technol., 2020,10, 5945. DOI: 10.1039/d0cy01373k
[23] Meng-Yu Rong, Jin-Shan Li, Yin Zhou, Fa-Guang Zhang*, and Jun-An Ma*. Catalytic Enantioselective Synthesis of Difluoromethylated Tetrasubstituted Stereocenters in Isoindolones Enabled by a Multiple-Fluorine System. Org. Lett. 2020, 22, 9010-9015. DOI: 10.1021/acs.orglett.0c03406
[24] Jun-Kuan Li, Biying Zhou, Yu-Chen Tian, Chunman Jia, Xiao-Song Xue, Fa-Guang Zhang*, and Jun-An Ma*. Potassium Acetate-Catalyzed Double Decarboxylative Transannulation To Access Highly Functionalized Pyrroles. Org. Lett. 2020. 22(24), 9585–9590. DOI: 10.1021/acs.orglett.0c03621
2019年文章
[1] Zhi-Qi Zhang, Meng-Meng Zheng, Xiao-Song Xue, Ilan Marek,* Fa-Guang Zhang,* and Jun-An Ma*. Catalytic Enantioselective Cyclopropenation of Internal Alkynes: Access to Difluoromethylated Three-Membered Carbocycles. Angew. Chem. Int. Ed. 2019, 58, 18191-18196. DOI: 10.1002/anie.201911701 DOI: 10.1002/anie.201913897 (Hot Paper, Back Cover)
[2] Shao-Peng Wang, Chi Wai Cheung,* and Jun-An Ma*. Direct Amidation of Carboxylic Acids with Nitroarenes. J. Org. Chem. 2019, 84, 13922-13934. DOI: 10.1021/acs.joc.9b02068
[3] Ni Shen, Chi Wai Cheung* and Jun-An Ma*. Direct amide synthesis via Ni-mediated aminocarbonylation of arylboronic acids with CO and nitroarenes. Chem. Commun. 2019, 55, 13709-13712. DOI: 10.1039/c9cc06638a
[4] Jun-Liang Zeng, Yue Zhang, Meng-Meng Zheng, Zhi-Qi Zhang, Xiao-Song Xue, Fa-Guang Zhang*, and Jun-An Ma*. Chemodivergent and Stereoselective Construction of gemDifluoroallylic Amines from Masked Difluorodiazo Reagents. Org. Lett. 2019, 21, 20, 8244-8249. DOI: 10.1021/acs.orglett.9b02989
[5] Zhen Chen, Wakana Mori, Jun-An Ma, Ming-Rong Zhang*, and Steven H. Liang*. Design, Synthesis, and Evaluation of 18F‑Labeled Monoacylglycerol Lipase Inhibitors as Novel Positron Emission Tomography Probes. J. Med. Chem. 2019, 62, 19, 8866-8872. DOI: 10.1021/acs.jmedchem.9b00936
[6] Fang-Fang Feng, Shen Li, Chi Wai Cheung*, and Jun-An Ma*. Chiral β‑Keto Propargylamine Synthesis via Enantioselective Mannich Reaction of Enamides with C‑Alkynyl N‑Boc N,O‑Acetals. Org. Lett. 2019, 21, 20, 8419-8423. DOI: 10.1021/acs.orglett.9b03181
[7] Fang-Fang Feng, Jin-Shan Li, Shen Li* and Jun-An Ma*. Enantioselective Addition of Enamides to Cyclic Ketimines: Access to Chiral 3,3-Disubstituted Isoindolin-1-ones. Advanced Synthesis & Catalysis, 2019, 361, 18, 4222-4226. DOI: 10.1002/adsc.201900710
[8] Zhen Chen, Meng-Yu Rong, Jing Nie, Xue-Feng Zhu*, Bing-Feng Shi * and Jun-An Ma *. Catalytic alkylation of unactivated C(sp3)–H bonds for C(sp3)–C(sp3) bond formation. Chem. Soc. Rev. 2019, 48, 4921. DOI: 10.1039/c9cs00086k
[9] Yu-Ting Tian, Yu-Wei Zong, Jing Nie, Fa-Guang Zhang*, and Jun-An Ma*. Construction of pyrrole- and indole-fused CF3-piperazine derivatives. Journal of Fluorine Chemistry. 2019, 226, 226, 109361. DOI: 10.1016/j.jfluchem.2019.109361
[10] Xing Peng, Ming-Yang Xiao, Jun-Liang Zeng, Fa-Guang Zhang*, and Jun-An Ma*. Construction of Difluoromethylated Tetrazoles via Silver-Catalyzed Regioselective [3 + 2] Cycloadditions of Aryl Diazonium Salts. Org. Lett. 2019, 21, 4808-4811. DOI: 10.1021/acs.orglett.9b01697
[11] Wenge Jiang, Dimitra Athanasiadou, Jun-An Ma,* Julian D. Gale* & Marc D. McKee*. Homochirality in biomineral suprastructures induced by assembly of single-enantiomer amino acids from a nonracemic mixture. Nat. Commun. 2019, 10, 2318. DOI: 10.1038/s41467-019-10383-x
[12] Meng-Yu Rong, Lijun Yang, Jing Nie, Fa-Guang Zhang*, and Jun-An Ma*. Construction of Chiral β‑Trifluoromethyl Alcohols Enabled by Catalytic Enantioselective Aldol-Type Reaction of CF3CHN2. Org. Lett. 2019, 21, 11, 4280-4283. DOI: 10.1021/acs.orglett.9b01468
[13] Yue Zhang, Zhen Chen, Jing Nie, Fa-Guang Zhang*, and Jun-An Ma*. Development of Cyanopyrazoles as Building Blocks to Fungicide Fluxapyroxad and Analogues. J. Org. Chem. 2019, 84, 7148-7158. DOI: 10.1021/acs.joc.9b00819
[14] Zhen Chen, Nan Ren, Xiaoxiao Ma, Jing Nie, Fa-Guang Zhang*, and Jun-An Ma*. Silver-Catalyzed [3 + 3] Dipolar Cycloaddition of Trifluorodiazoethane and Glycine Imines: Access to Highly Functionalized Trifluoromethyl-Substituted Triazines and Pyridines. ACS Catal. 2019, 9, 4600-4608. DOI: 10.1021/acscatal.9b00846
[15] Zhen Chen, Wakana Mori,Xiaoyun Deng, Ran Cheng, Jun-An Ma, Ming-Rong Zhang* and Steven H. Liang*. Design, Synthesis, and Evaluation of Reversible and Irreversible Monoacylglycerol Lipase Positron Emission Tomography (PET) Tracers Using a “Tail Switching” Strategy on a Piperazinyl Azetidine Skeleton. J. Med. Chem. 2019, 62, 3336-3353. DOI: 10.1021/acs.jmedchem.8b01778
[16] Beibei Liu, Ge Qu, Jun-Kuan Li, Wenchao Fan, Jun-An Ma, Yan Xu, YaoNie*, and Zhoutong Sun*.Conformational Dynamics-Guided Loop Engineering of an Alcohol Dehydrogenase: Capture, Turnover and Enantioselective Transformation of Difficult-to-Reduce Ketones. Adv. Synth. Catal. 2019, 361, 3182-3190. DOI: 10.1002/adsc.201900249
[17] Ge Qu, Mingxing Fu, Lili Zhao, Beibei Liu, Pi Liu, Wenchao Fan, Jun-An Ma,* and Zhoutong Sun*. Computational Insights into the Catalytic Mechanism of Bacterial Carboxylic Acid Reductase. J. Chem. Inf. Model. 2019, 59, 832-841. DOI: 10.1021/acs.jcim.8b00763
[18] Ning Lva, Yi-Qiang Tiana, Fa-Guang Zhang*, Jun-An Ma*. One-Pot Sequential Multistep Transformation of α,β-Unsaturated Trifluoromethyl Ketones: Facile Synthesis of Trifluoromethylated 2-Pyridones. Synlett. 2019, 30, 5, 605-609. DOI: 10.1055/s-0037-1612077
[19] Chi Wai Cheung*, Ni Shen, Shao-Peng Wang, Asim Ullah, Xile Hu, and Jun-An Ma *. Manganese-mediated reductive amidation of esters with nitroarenes. Org. Chem. Front. 2019, 6, 756. DOI: 10.1039/c8qo01405a
[20]Yue Zhang, Yi Wei, Shen Li* and Jun-An Ma*. Stereoselective One-Pot Synthesis of cis-1,2-Dicyanoalkenes from 1,1-Bis(benzenesulfonyl)alkenes and KCN. Eur. J. Org. Chem. 2019, 199-203. DOI: 10.1002/ejoc.201801504
2018年文章
[1] Jin-Shan Li, Yong-Jie Liu, Shen Li and Jun-An Ma*. Chiral phosphoric acid-catalyzed direct asymmetric mannich reaction of cyclic C-acylimines with simple ketones: facile access to C2-quaternary indolin-3-ones. Chem. Commun., 2018, 54, 9151. DOI: 10.1039/c8cc05125a
[2] Ran Guo, Ning Lv, Fa-Guang Zhang,* and Jun-An Ma*. Zinc-Mediated Mannich-Type Reaction of 2,2,2-Trifluorodiazoethane with Imines: Access to β‑CF3‑Amines. Org. Lett. 2018, 20, 22, 6994-6997. DOI: 10.1021/acs.orglett.8b02816
[3] Zhang Fa-Guang*, Peng Xing, Ma Jun-An*. Recent Advances in the Synthesis of CF3-Substituted Triazoles and Tetrazoles. Chin. J. Org. Chem. 2018, 38. DOI: 10.6023/cjoc201808007
[4] Ren Zhiwen, Ren Nan, Zhang Faguang*, Ma Junan*. Facile Synthesis of Fluorinated Isoxazoles via Consecutive Double C-F Bond Cleavage. Acta Chim. Sinica. 2018, 76. DOI: 10.6023/A18070279
[5] Jun-Liang Zeng, Zhen Chen, Fa-Guang Zhang,* and Jun-An Ma*. Direct Regioselective [3 + 2] Cycloaddition Reactions of Masked Difluorodiazoethane with Electron-Deficient Alkynes and Alkenes: Synthesis of Difluoromethyl-Substituted Pyrazoles. Org. Lett. 2018, 20, 15, 4562-4565. DOI: 10.1021/acs.orglett.8b01854
[6] Huan Zhou, Botao Wu, Jun-An Ma and Yanfeng Dang* . Mechanistic understanding of [Rh(NHC)]-catalyzed intramolecular [5 + 2] cycloadditions of vinyloxiranes and vinylcyclopropanes with alkynes. Org. Biomol. Chem. 2018, 16, 4295. DOI: 10.1039/c8ob01117frsc.li/obc
[7] Baokun Qiao, Hao-Qiang Cao, Fa-Guang Zhang,* Jun-An Ma*. Pd(II)-Catalyzed Phosphorylation of Enamido C(sp2)‒H Bonds: A General Route to β-Amido-Vinylphosphonates. Chin. J. Chem. 2018, 36, 9, 809-814. DOI: 10.1002/cjoc.201800262
[8] Fa‐Guang Zhang,* Ning Lv, Yan Zheng, and Jun‐An Ma* . Phosphine‐Relayed Aldehyde‐Olefination and Aza‐Wittig Reaction with 2,2,2‐Trifluorodiazoethane. Chin. J. Chem. 2018, 36, 8, 723-730. DOI: 10.1002/cjoc.201800158
[9] Yong-Jie Liu, Jin-Shan Li, Jing Nie,* and Jun-An Ma *. Organocatalytic Asymmetric Decarboxylative Mannich Reaction of β Keto Acids with Cyclic α Ketiminophosphonates: Access to Quaternary α Aminophosphonates. Org. Lett. 2018, 20, 12, 3643-3646. DOI: 10.1021/acs.orglett.8b01422
[10] Yue Zhang, Jing Nie, Fa-Guang Zhang*, Jun-An Ma*. Zinc-mediated enantioselective addition of terminal 3-en-1-ynes to cycli trifluoromethyl ketimines. Journal of Fluorine Chemistry, 2018, 208, 1-9. DOI: 10.1016/j.jfluchem.2018.01.008
[11] Chi Wai Cheung， Jun-An Ma* and Xile Hu*. Manganese-Mediated Reductive Transamidation of Tertiary Amides with Nitroarenes. J. Am. Chem. Soc. 2018, 140, 6789-6792. DOI: 10.1021/jacs.8b03739
[12] Fa-Guang Zhang, Jun-Liang Zeng, Jun-An Ma*. Telescoping Reactions of Trifluorodiazoethane‐derived Aza‐Wittig Reagents with Allenyl esters. Chem. Eur. J. 2018, 24, 30, 7749-7754. DOI: 10.1002/chem.201801171
[13] Zhen Chen, Yue Zhang, Jing Nie, and Jun-An Ma*. Transition-Metal-Free [3 + 2] Cycloaddition of Nitroolefins and Diazoacetonitrile: A Facile Access to Multisubstituted Cyanopyrazoles. Org. Lett. 2018, 20, 7, 2120-2124. DOI: 10.1021/acs.orglett.8b00729
[14] Yin-Jun Huang, Baokun Qiao, Fa-Guang Zhang*, Jun-An Ma*. Facile construction of trifluoromethyl-azirines via one-pot metal-free Neber reaction. Tetrahedron. 2018, 1-6. DOI: 10.1016/j.tet.2018.05.033
[15] Ya-Jing Fan, Lei Zhou and Shen Li *. Catalytic asymmetric 1,6-conjugate addition of in situ generated para-quinone methides with tritylthiol. Org. Chem. Front. 2018, 5, 1820-1824. DOI: 10.1039/c8qo00211h
2017年文章
[1] Zhen Chen, Yan Zheng, Jun-An Ma*. Use of a Traceless Activating and Directing Group for the Construction of Trifluoromethylpyrazoles: One‐Pot Transformation of Nitroolefins and Trifluorodiazoethane. Angew. Chem. Int. Ed. 2017. 56, 4569–4574. DOI: 10.1002/anie.201700955
[2] Shuang Qin, Yan Zheng, Fa-Guang Zhang*, Jun-An Ma*. One-Pot Cascade Transformations of Zinc Trifluorodiazoethylide and α, β-Unsaturated Enones: Access to Trifluoromethylated Polycyclic Pyrazolines. Org. Lett. 2017, 19, 13, 3406-3409. DOI: 10.1021/acs.orglett.7b01362
[3] Jin-Shan Li, Han-Feng Cui, Ke-Feng Zhang, Jing Nie, Jun-An Ma*. Phase‐Transfer‐Catalyzed Asymmetric Michael Addition of (Iminomethyl) phosphonates to α,β‐Unsaturated Ketones: Access to α‐Aminophosphonic Acid Derivatives. Eur. J. Org. Chem. 2017, 17, 2545-2552. DOI: 10.1002/ejoc.201700249
[4] Jun-Liang Zeng, Helene Chachignon, Jun-An Ma*, Dominique Cahard*. Nucleophilic Trifluoromethylthiolation of Cyclic Sulfamidates: Access to Chiral β-and γ-SCF3 Amines and α-Amino Esters. Org. Lett. 2017, 19, 8, 1974-1977. DOI: 10.1021/acs.orglett.7b00501
[5] Yi Wei, Heng-Xia Zhang, Jun-Liang Zeng, Jing Nie, Jun-An Ma*. Organocatalytic Asymmetric Decarboxylative Amination of β-Keto Acids: Access to Optically Active α-Amino Ketones and 1,2-Amino Alcohols. Org. Lett. 2017, 19, 8, 2162-2165. DOI: 10.1021/acs.orglett.7b00797
[6] Shen Li, Wen-Jie Cao, Jun-An Ma*. Stereoselective Cycloaddition of 2,2,2-Trifluorodiazoethane with α-Methylene-β-lactams: Facile Synthesis of Trifluoromethyl-Substituted Spirocyclic β-Lactams. Synlett. 2017, 28, 6, 673-678. DOI: 10.1055/s-0036-1588363
[7] Jin-Shan Li, Yong-Jie Liu, Guang-Wu Zhang, and Jun-An Ma*. Catalytic Asymmetric Mukaiyama–Mannich Reaction of Cyclic C-Acylimines with Difluoroenoxysilanes: Access to Difluoroalkylated Indolin-3-ones. Org. Lett. 2017, 19, 23, 6364-6367. DOI: 10.1021/acs.orglett.7b03213
2016年文章
[1] Zhen-Yan Yang, Jun-Liang Zeng, Nan Ren, Wei Meng, Jing Nie, Jun-An Ma*. C2-Symmetric Chiral Bisoxazolines as Hydrogen-Bond-Acceptor Catalysts in Enantioselective Aldol Reaction of β-Carbonyl Acids with Trifluoroacetaldehyde Hemiacetals. Org. Lett. 2016, 18, 24, 6364-6367. DOI: 10.1021/acs.orglett.6b03256
[2] Chun-Man Jia, Heng-Xia Zhang, Jing Nie, Jun-An Ma*. Catalytic Asymmetric Decarboxylative Mannich Reaction of Malonic Acid Half Esters with Cyclic Aldimines: Access to Chiral β-Amino Esters and Chroman-4-amines. J. Org. Chem. 2016, 81, 18, 8561-8569. DOI: 10.1021/acs.joc.6b01750
[3] Ran Guo, Yan Zheng, Jun-An Ma*. Electrophilic Reaction of 2,2,2-Trifluorodiazoethane with the in Situ Generated N-Heterocyclic Carbenes: Access to N-Aminoguanidines. Org. Lett. 2016, 18, 17, 4170-4173. DOI: 10.1021/acs.orglett.6b01191
[4] Yi Wei, Ran Guo, Yanfeng Dang, Jing Nie, Jun-An Ma*. Organocatalytic Enantioselective Decarboxylative Michael Addition of β‐Keto Acids to Dicyanoolefins and Disulfonylolefins. Advanced Synthesis & Catalysis. 2016, 358, 17, 2721-2726. DOI: 10.1002/adsc.201600485
[5] Yan Zheng, Hai Ma, Jun-An Ma*. Catalytic Enantioselective 1,2‐Addition of Terminal 1,3‐Diynes to Trifluoromethyl Ketones. Chinese Journal of Chemistry, 2016, 34, 5, 511-518. DOI: 10.1002/cjoc.201500901
[6] Bo-Nan Lai, Jian-Feng Qiu, Heng-Xia Zhang, Jing Nie, Jun-An Ma*. Stereoselective Synthesis of Fused Aziridines via One-Pot Sequential Decarboxylative Mannich Reaction and Oxidative C–H Amination of Cyclic Imines with β-Ketoacids. Org. Lett. 2016, 18, 3, 520-523. DOI: 10.1021/acs.orglett.5b03551
[7] Nan Ren, Jing Nie, Jun-An Ma*. Base-and metal-free decarboxylative aldol reaction of β-ketoacids with glyoxylate hydrates and glyoxal monohydrates in water. Green Chemistry. 2016, 18, 24, 6609-6617. DOI: 10.1039/c6gc02705a
[8] Chuan-Le Zhu, Jun-An Ma*, Dominique Cahard*. Trifluorodiazoethane (CF3CHN2) in the Uncatalyzed Cyclopropanation of 3‐Arylmethylenebenzofuran‐2(3H)‐ones. Asian Journal of Organic Chemistry. 2016, 5, 1, 66-69. DOI: 10.1002/ajoc.201500409
2015年文章
[1] Baokun Qiao, Yin-Jun Huang, Jing Nie, Jun-An Ma*. Highly regio-, diastereo-, and enantioselective Mannich reaction of allylic ketones and cyclic ketimines: Access to chiral benzosultam. Org. Lett. 2015, 17, 18, 4608-4611. DOI: 10.1021/acs.orglett.5b02351
[2] Yu-Ping Yi, Yan Zheng, Jing Nie, Jun-An Ma*. Oxone-promoted hydration of electron-deficient allenic esters and ketones into 1,3-dicarbonyl compounds. Tetrahedron Letters. 2015, 56(30): 4523-4526. DOI: 10.1016/j.tetlet.2015.05.120。
[3] Chuan-Le Zhu, Li-Jun Yang, Shen Li, Yan Zheng, Jun-An Ma*. Brine-Stabilized 2,2,2-Trifluorodiazoethane and Its Application in the Synthesis of CF3–Substituted Cyclopropane α-Amino Acids. Org. Lett. 2015, 17, 14, 3442-3445. DOI: 10.1021/acs.orglett.5b01450
[4] Jun-Liang Zeng, Jian Wang, Jun-An Ma*. New strategies for rapid 18F-radiolabeling of biomolecules for radionuclide-based in vivo imaging. Bioconjugate Chemistry. 2015, 26, 6, 1000-1003. DOI: 10.1021/acs.bioconjchem.5b00180
[5] Zhen-Yan Yang, Tian-Lin Liu, Yan Zheng, Shen Li, Jun-An Ma*. Asymmetric Enynylation of N‐Sulfonyl Aldimines Catalyzed by Zn‐BINOL Complexes. European Journal of Organic Chemistry, 2015. DOI: 10.1002/ejoc.201500400
[6] Long Sun, Jing Nie, Yan Zheng, Jun-An Ma*. [3+2] Cycloaddition of arynes with CF3CHN2: Access to 3-trifluoromethyl-1H-indazoles. Journal of Fluorine Chemistry. 2015, 174, 88-94. DOI: 10.1016/j.jfluchem.2014.06.002
[7] Ai-Jia Wei, Jing Nie, Yan Zheng, Jun-An Ma*. Ni-Catalyzed Highly Chemo-, Regio-, and Enantioselective Decarboxylative Aldol Reaction of β, γ-Unsaturated α-Ketoesters with β-Ketoacids. J. Org. Chem. 2015, 80, 8, 3766-3776. DOI: 10.1021/jo502741z
[8] Xiao-Dong Tang, Shen Li, Ran Guo, Jun-An Ma*. Chiral Phosphoric Acid Catalyzed Enantioselective Decarboxylative Alkylation of β-Keto Acids with 3-Hydroxy-3-indolyloxindoles. Org. Lett. 2015, 17, 6, 1389-1392. DOI: 10.1021/acs.orglett.5b00159
[9] Jian Wang, Guan-Bo Huang, Li-Jun Yang, Feng Li, Jing Nie, Jun-An Ma*. Tandem stereoselective synthesis of new trifluoromethylated pyranopyrazoles. Journal of Fluorine Chemistry, 2015, 171, 27-35. DOI: 10.1016/j.jfluchem.2014.10.008
[10] Zhen Chen, Shuang-Qing Fan, Yan Zheng , Jun-An Ma*. Silver-catalyzed regioselective [3+2] cycloaddition of arene-diazonium salts with 2,2,2-trifluorodiazoethane (CF3CHN2): a facile access to 2-aryl-5-trifluoromethyltetrazoles. Chem. Commun. 2015, 51, 92, 16545-16548. DOI: 10.1039/c5cc07324c
[11] Shuai Wang, Li-Jun Yang, Jun-Liang Zeng, Yan Zheng, Jun-An Ma*. Silver-catalyzed [3+2] cycloaddition of isocyanides with diazo compounds: new regioselective access to 1,4-disubstituted-1,2,3-triazoles. Organic Chemistry Frontiers. 2015, 2, 11, 1468-1474. DOI: 10.1039/c5qo00219b
[12] Shen Li, Jun-An Ma*. Core-structure-inspired asymmetric addition reactions: enantioselective synthesis of dihydrobenzoxazinone-and dihydroquinazolinone-based anti-HIV agents. Chem. Soc. Rev. 2015, 44, 21, 7439-7448. DOI: 10.1039/c5cs00342c
[13] Ai-Jie Cai, Yan Zheng, Jun-An Ma*. Copper-triggered majunan-component reaction of CF3CHN2, nitriles, and aldehydes: highly diastereoselective synthesis of CF 3-substituted oxazolines and vicinal amino alcohols. Chem. Commun. 2015, 51, 43, 8946-8949. DOI: 10.1039/c5cc02749g
2015年以前文章
[1] Manfred T. Reetz,* Jun-An Ma, and Richard Goddard. Binol-Derived Monodentate Phosphites and Phosphoramidites with Phosphorus Stereogenic Centers: Novel Ligands for Transition-Metal Catalysis. Angew. Chem. Int. Ed. 2005, 44, 412-415. DOI: 10.1002/anie.200461624
[2] Hong-Chao Guo and Jun-An Ma*. Catalytic Asymmetric Tandem Transformations Triggered by Conjugate Additions. Angew. Chem. Int. Ed. 2006, 45, 354-366. DOI: 10.1002/anie.200500195
[3] Jun-An Ma*. Catalytic asymmetric synthesis of a- and b-amino phosphonic acid derivatives. Chem. Soc. Rev. 2006, 35, 630-636. DOI: 10.1002/adsc.202001345
[4] Jun-An Ma and Dominique Cahard*. Asymmetric Fluorination, Trifluoromethylation, and Perfluoroalkylation Reactions. Chem. Rev. 2008, 108, PR1-PR43. DOI: 10.1021/cr030143e
[5] Ming-Qing Hua, Han-Feng Cui, Lian Wang, Jing Nie, and Jun-An Ma*. Reversal of Enantioselectivity by Tuning the Conformational Flexibility of Phase-Transfer Catalysts. Angew. Chem. Int. Ed. 2010, 49, 2772-2776. DOI: 10.1002/ange.200906814
[6] Jing Nie, Hong-Chao Guo, Dominique Cahard, and Jun-An Ma*. Asymmetric Construction of Stereogenic Carbon Centers Featuring a Trifluoromethyl Group from Prochiral Trifluoromethylated Substrates. Chem. Rev. 2011, 111, 455-529. DOI: 10.1021/cr100166a
[7] Chuan-Le Zhu, Fa-Guang Zhang, Wei Meng, Jing Nie, Dominique Cahard, and Jun-An Ma*. Enantioselective Base-Free Electrophilic Amination of Benzofuran- 2(3H)-ones: Catalysis by Binol-Derived P-Spiro Quaternary Phosphonium Salts. Angew. Chem. Int. Ed. 2011, 50, 5869-5872. DOI: 10.1002/ange.201100283
[8] Guang-Wu Zhang, Wei Meng, Hai Ma, Jing Nie, Wen-Qin Zhang, and Jun-An Ma*. Catalytic Enantioselective Alkynylation of Trifluoromethyl Ketones: Pronounced Metal Fluoride Effects and Implications of Zinc-to-Titanium Transmetallation. Angew. Chem. Int. Ed. 2011, 50, 3538-3542. DOI: 10.1002/ange.201007341
[9] Lian Wang, Wei Meng, Chuan-Le Zhu, Yan Zheng, Jing Nie, and Jun-An Ma*. The Long-Arm Effect: Influence of Axially Chiral Phosphoramidite Ligands on the Diastereo- and Enantioselectivity of the Tandem 1,4-Addition/Fluorination. Angew. Chem. Int. Ed. 2011, 50, 9442-9446. DOI: 10.1002/ange.201104565
[10] Wei Meng, Hai-Tao Zhao,a Jing Nie, Yan Zheng, Aiping Fu and Jun-An Ma*. Allenoate-derived 1,5-, 1,7-, and 1,9-zwitterions as highly versatile couplingpartners for phosphine-triggered cycloaddition reactions. Chem. Sci. 2012, 3, 3053. DOI: 10.1039/c2sc20805a
[11] Teng Wang, Wang Zhou, Hang Yin, Jun-An Ma, and Ning Jiao*. Iron-Facilitated Oxidative Dehydrogenative C=O Bond Formation by Propargylic Csp3-H Functionalization. Angew. Chem. Int. Ed. 2012, 51, 10823-10826. DOI: 10.1002/anie.201205779
[12] Cui-Bo Liu, Wei Meng, Feng Li, Shuai Wang, Jing Nie, and Jun-An Ma*. A Facile Parallel Synthesis of Trifluoroethyl-Substituted Alkynes. Angew. Chem. Int. Ed. 2012, 51, 6227-6230. DOI: 10.1002/ange.201202372
[13] Feng Li, Jing Nie, Long Sun, Yan Zheng, and Jun-An Ma*. Silver-Mediated Cycloaddition of Alkynes with CF3CHN2 : Highly Regioselective Synthesis of 3-Trifluoromethylpyrazoles. Angew. Chem. Int. Ed. 2013, 52, 6255-6258. DOI: 10.1002/ange.201301870
[14] Hai-Na Yuan, Shuai Wang, Jing Nie, Wei Meng, Qingwei Yao, and Jun-An Ma*. Hydrogen-Bond-Directed Enantioselective Decarboxylative Mannich Reaction of b-Ketoacids with Ketimines: Application to the Synthesis of Anti-HIV Drug DPC 083. Angew. Chem. Int. Ed. 2013, 52, 3869-3873. DOI: 10.1002/ange.201210361
[15] Shen Li and Jun-An Ma*. Core-structure-inspired asymmetric addition reactions: enantioselective synthesis of dihydrobenzoxazinone- and dihydroquinazolinonebased anti-HIV agents. Chem. Soc. Rev. 2015, 44. 7439. DOI: 10.1039/c5cs00342c
