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成果及论文

一、期刊论文

  1. Gao, Y. Q.; Hu, Y. G.; Ye, J. H.; Ma, Z. Q.; Feng, J. T.; Liu, X. L.; Lei, P.*; Szostak, M.* Pd–NHC (NHC = N-Heterocyclic Carbene)-Catalyzed B-Alkyl Suzuki Cross-Coupling of 2-Pyridyl Ammonium Salts by N–C Activation: Application to the Discovery of Agrochemical Molecular Hybrids. Org. Lett. 2024, 26(11), 2309–2314. DOI: 10.1021/acs.orglett.4c00549.

  2. Liu, H. R.; Cai, C. L.; Zhang, X. J.; Li, W. K.; Ma, Z. Q.; Feng, J. T.; Liu, X. L.; Lei, P.* Discovery of Novel Cinnamic Acid Derivatives as Fungicide Candidates. J. Agric. Food Chem. 2024, 72(5), 2492–2500. DOI: 10.1021/acs.jafc.3c05655.

  3. Zhang, J.#; Zhao, Y. C.#; Zhu, Y. Y.#; Lei, P.#; Liu, H. R.; Wang, C. S.; Xing, S. Y.; Liu, Y.; Ni, S. F.*; Castanheiro, T.*; Xu, L. W.; Shao. X. X.* Base-induced azofluoroalkylation of unactivated alkenes via halogen atom transfer. Org. Chem. Front. 2024, DOI: 10.1039/D3QO02114A.

  4. 刘函如, 王宇佳, 李来福, 周一万*, 马志卿*, 雷鹏*. 生物农药防治花椒窄吉丁虫和流胶病的使用技术筛选与评价. 中国生物防治学报. 2023, 39(6), 1482–1487. DOI: 10.16409/j.cnki.2095-039x.2023.01.043.

  5. Hu, Y. G.; Gao, Y. Q.; Ye, J. H.; Ma, Z. Q.; Feng, J. T.; Liu, X. L.; Szostak, R.; Lei, P.*; Szostak, M.* Suzuki–Miyaura Cross-Coupling of 2-Pyridyl Trimethylammonium Salts by N–C Activation Catalyzed by Air- and Moisture-Stable Pd–NHC Precatalysts: Application to the Discovery of Agrochemicals. Org. Lett. 2023, 25(17), 2975–2980. DOI: 10.1021/acs.orglett.3c00741.

  6. Zhang, C. X.; Yuan, H. X.; Hu, Y. G.; Li, X. H.; Gao, Y. Q.; Ma, Z. Q.*; Lei, P.* Structural Diversity Design, Synthesis, and Insecticidal Activity Analysis of Ester-Containing Isoxazoline Derivatives Acting on GABA Receptor. J. Agric. Food Chem. 2023, 71(7), 3184–3191. DOI: 10.1021/acs.jafc.2c07910.

  7. Pan, T. M.#; Ye, J. H.#; Li, J. N.; Gui, K.; Li, J.; Feng, J. T.; Ma, Z. Q.; Lei, P.*; Gao, Y. Q.* Discovery of Terpene-derived Quaternary Ring Compounds Containing an Oxime Moiety as Potential Fungicides. J. Agric. Food Chem. 2023, 71(7), 3164–3172. DOI: 10.1021/acs.jafc.2c07387.

  8. 张文广#, 刘函如#, 魏志敏, 袁含笑, 王瑞龙, 张洪艳, 张璟, 李秀环*, 雷鹏*. 5-甲基异噁唑-4-甲酸肟酯衍生物的合成及抑菌活性. 农药学学报, 2023, 25(2), 468–473. DOI: 10.16801/j.issn.1008-7303.2022.0105.

  9. Lei, P.*; Wang, Y. B.; Zhang, C. X.; Hu, Y. G.; Feng, J. T.; Ma, Z. Q.*; Liu, X. L.*; Szostak, R.; Szostak, M.* Sonogashira Cross-Coupling of Aryl Ammonium Salts by Selective C–N Activation Catalyzed by Air- and Moisture-Stable, Highly Ac-tive [Pd(NHC)(3-CF3-An)Cl2] (An = Aniline) Precatalysts. Org. Lett. 2022, 24(34), 6310–6315.  DOI: 10.1021/acs.orglett.2c02534.

  10. 袁含笑, 张文广, 刘函如, 张云天, 张彩霞, 郭孜怡, 高艳清, 雷  鹏*, 刘西莉*. 香豆素肟酯衍生物的合成及抑菌活性. 农药学学报, 2022, 24(5), 1189–1195. DOI: 10.16801/j.issn.1008-7303.2022.0078.

  11. Hu, Y. G.#; Gao, Y. Q.#; Wang, Y. J.; Zhang, W. G.; Liu, H. R.; Zhang, X. J.; Ma, Z. Q.; Liu, X. L.; Lei, P.* Non-food bioactive products: Diversified invention of 1,2,4-oxadiazole-containing amide derivatives for novel fungicidal candidate discovery. Ind. Crops Prod. 2022, 184, 115087. DOI: 10.1016/j.indcrop.2022.115087.

  12. Wang, Y. J.; Mu, Y. L.; Hu, X. T.; Zhang, C. X.; Gao, Y. Q.; Ma, Z. Q.; Feng, J. T.; Liu, X. L.; Lei, P.* Indole/Tetrahydroquinoline as Renewable Natural Resource-Inspired Scaffolds in the Devising and Preparation of Potential Fungicide Candidates. J. Agric. Food. Chem. 2022, 70(15), 4582–4590. DOI: 10.1021/acs.jafc.1c07879.

  13. 王宇佳, 耿媛霄, 高艳清, 王建花, 冯俊涛, 周一万, 雷 鹏*, 马志卿. 8种植物源农药对花椒蚜虫的田间防效. 西北农林科技大学学报(自然科学版), 2022, 50(8), 88–93. DOI: 10.13207/j.cnki.jnwafu.2022.08.010.

  14. 张兴甲, 魏志敏, 王宇佳, 杨龙港, 袁含笑, 冯俊涛, 高艳清*, 雷 鹏*, 马志卿. 3-二氟甲基-1-甲基吡唑-4-羧酸肟酯衍生物的合成及抑菌活性. 农药学学报, 2022, 24(1), 59–65. DOI: 10.16801/j.issn.1008-7303.2021.0140

  15. Lei, P.*,#; Wang, Y. B.#; Mu, Y. L.; Wang, Y. J.; Ma, Z. Q.; Feng, J. T.; Liu, X. L.; Szostak, M.* Green Solvent Selection for Acyl Buchwald-Hartwig Cross-Coupling of Amides (Transamidation). ACS Sustain. Chem. Eng. 2021, 9(44), 14937–14945. DOI: 10.1021/acssuschemeng.1c05307.

  16. Lei, P.*#; Mu, Y.L.#; Wang, Y.B.#; Wang, Y.J.; Ma, Z.Q.; Feng, J.T.; Liu, X.L.; Szostak, M.* Green Solvent Selection for Suzuki−Miyaura Coupling of Amides. ACS Sustain. Chem. Eng. 2021, 9(1), 552−559. DOI: 10.1021/acssuschemeng.0c08044.

  17. Lei, P.* #; Li, G. C. #; Ling, Y.; An, J.; Nolan S. P.; Szostak, M.* Protocol for Palladium/N-Heterocyclic Carbene-Catalyzed Suzuki–Miyaura Cross-Coupling of Amides by N-C(O) Activation. Synthesis 2021, 53(04), 682−687. DOI: 10.1055/s-0040-1705956. (Practical Synthetic Procedure; Selected as Front Cover)

  18. 沈安泽#, 胡恩畅#, 刘函如, 王宇佳, 王  勇, 马志卿, 冯俊涛, 雷鹏*. 含肟酯的吡唑衍生物的合成及其抑菌活性. 农药学学报, 2021, 23(1), 69−75. DOI: 10.16801/j.issn.1009-7303.2021.0005.

  19. Lei, P.*; Ling, Y.; An, J.; Nolan S. P.; Szostak, M.* 2-Methyltetrahydrofuran (2-MeTHF): A Green Solvent for Pd–NHC-Catalyzed Amide and Ester Suzuki–Miyaura Cross-Coupling by N-C/O-C Cleavage. Adv. Synth. Catal. 2019, 361(24), 5654−5660. 

  20. 穆雅利, 胡夏桐, 马志卿, 雷鹏*. 异噁唑啉类化合物生物活性研究进展. 农药, 2019, 58(12), 864−869.

  21. 雷鹏#, 丁新吉#, 吴远勇, 马志卿*. 含肟醚的松油烯-4-醇衍生物的合成及杀虫活性. 有机化学, 2019, 39, 2070−2074.

  22. Lei, P.#; Ding, Y.X.#; Zhang, X.H.; Adijiang, A.; Li, H.Z.; Ling, Y.; An, J.* A practical and chemoselective ammonia-free Birch reduction. Org. Lett. 2018, 20, 3439−3442.  (Highlighted on c&en) 

  23. Lei, P.#; Meng, G. R.#; Szostak, M.* A general method for the Suzuki-Miyaura cross-coupling of amides using commercially available, air- and moisture-stable palladium/NHC (NHC = N-heterocyclic carbene) complexes. ACS Catal. 2017, 7, 1960–1965. (Highly Cited & Hot Paper) 

  24. Lei, P.; Meng, G. R.; Shi, S. C.; Ling, Y.; An, J.; Szostak, R.; Szostak, M.* Suzuki–Miyaura cross-coupling of amides and esters at room temperature: correlation with barriers to rotation around C–N and C–O bonds. Chem. Sci. 2017, 8, 6525–6530. (Highlighted in Synfacts, 2017, 13, 1189) (Hot Paper) 

  25. Lei, P.; Meng, G. R.; Ling, Y.; An, J.; Nolan S. P.; Szostak, M.* General method for the Suzuki-Miyaura Cross-Coupling of primary amides enabled by [Pd(NHC)(cin)Cl] at room temperature. Org. Lett. 2017, 19, 6510–6513.

  26. Lei, P.; Meng, G. R.; Ling, Y.; An, J.; Szostak, M.* Pd-PEPPSI: Pd-NHC precatalyst for Suzuki−Miyaura cross-coupling reactions of amides. J. Org. Chem. 2017, 82, 6638−6646. (Highlighted on Organic Chemistry Portal)

  27. Shi, S. C.#; Lei, P.#; Szostak, M.* Pd-PEPPSI: A general Pd-NHC precatalyst for Suzuki–Miyaura cross-coupling of esters by C–O cleavage. Organometallics 2017, 36, 3784–3789.

  28. Lei, P.; Xu, Y.; Du, J.; Yang, X. L.; Yuan, H. Z.; Xu, G. F.; Ling, Y.* Design, synthesis and fungicidal activity of N-substituted benzoyl-1,2,3,4-tetrahydroquinolyl-1-carboxamide. Bioorg. Med. Chem. Lett. 2016, 26, 2544–2546. 

  29. Lei, P.; Zhang, X. B.; Xu, Y.; Xu, G. F.; Liu, X. L.; Yang, X. L.; Zhang, X. H.; Ling, Y.* Synthesis and fungicidal activity of pyrazole derivatives containing 1,2,3,4-tetrahydro-quinoline. Chem. Cent. J. 2016, 10, 40. 


  1. Zhou, R.; Liu, X.; Hui, T. P.; Ye, J. H.; Chen, G. Y.; Lei, P.; Li, J.; Feng, J. T.; Gao, Y. Q. Discovery of Novel Cyclobutyl Oxime Ester Derivatives Containing an α,β-Unsaturated Carbonyl Moiety as Potential Mitochondrial Toxins. J. Agric. Food Chem. 2024, 72(40), 22054–22062. DOI: 10.1021/acs.jafc.4c05066.

  2. Li, L. W.; Chen, G. Y.; Gu, H. P.; Lei, P.; Gao, Y. Q.; Ma, Z. Q.; Feng, J. T. Natural α-Methylene-γ-Butyrolactone Analogues: Synthesis and Evaluation of Isoaurone Derivatives as Antifungal Agents. Chem. Biodiversity 2024, e202401955. DOI: 10.1002/cbdv.202401955.

  3. Chen, G. Y.; Bai, J.; Wu, X. Y.; Huo, X. Y.; Li, Y. Q.; Lei, P.; Ma, Z. Q. Amphiphilic amidines as potential plasmic membrane-targeting antifungal agents: synthesis, bio-activities and QSAR. Pest Manag. Sci. 2024, 80(10), 5266–5276. DOI: 10.1002/ps.8253.

  4. 桂阔, 周瑞, 惠托平, 刘夷宁, 张欣茹, 李文奎, 雷鹏, 高艳清*, 马志卿. 中空介孔二氧化硅负载戊唑醇纳米缓释颗粒的制备及生物活性. 农药学学报 2024, 26(3), 559–569. DOI: 10.16801/j.issn.1008-7303.2024.0036.

  5. 叶久辉, 桂阔, 殷妮, 刘新, 李璇, 雷鹏, 冯俊涛, 马志卿, 高艳清*. 桧木醇酯类衍生物的设计合成及抑菌活性. 农药学学报 2024, 26(3), 462–471. DOI: 10.16801/j.issn.1008-7303.2024.0039.

  6. Li, L. W.; Hui, T. P.; Li, Y. Y.; Wang, Y. Q.; Gu, H. P.; Chen, G. Y.; Lei, P.; Gao, Y. Q.; Feng, J. T. Design, synthesis and antifungal activity of novel α-methylene-γ-butyrolactone derivatives containing benzothiophene moiety. Pest Manag. Sci. 2024, 80(8), 3776–3785. DOI: 10.1002/ps.8080.

  7. Li, L. W.; Yang, D. Y.; Li, H.; Chen, G. Y.; Lei. P.; Gao, Y. Q.; Feng, J. T. Heterocycle-Substituted α-Methylene-γ-Butyrolactones Derivatives Synthesis, Antifungal Activity, and 3D-QSAR. J. Agric. Food Chem. 2023, 71(29), 11008–11015. DOI: 10.1021/acs.jafc.3c02117.

  8. Li, J. N.; Ye, J. H.; Zhou, R.; Gui, K.; Li, J.; Feng, J. T.; Ma, Z. Q.; Lei, P.; Gao, Y. Q. Systematic Study on Turpentine-Derived Amides from Natural Plant Monoterpenes as Potential Antifungal Candidates. J. Agric. Food Chem. 2023, 71(14), 5507–5515. DOI: 10.1021/acs.jafc.3c00314.

  9. 张旭欢, 王阿玲, 李文奎, 吴华, 雷鹏, 冯俊涛, 王勇, 马志卿. 桧木醇对西瓜枯萎病菌抑菌作用研究. 农药学学报 2023, 25(3), 630–637. DOI: 10.16801/j.issn.1008-7303.2023.0010.

  10. 桂阔, 叶久辉, 李璇, 周海玉, 李婕宁, 冯俊涛, 雷鹏, 高艳清*, 马志卿. 桧木醇衍生物的合成及抑菌活性. 农药学学报, 2023, 25(1), 73–80. DOI: 10.16801/j.issn.1008-7303.2022.0106.

  11. Pan, T.M.; Geng, Y.X.; Hao, J.; He, X.H.; Li, J.*; Gao, Y.Q.*; Shang, S.B.; Song, Z.Q. Taking Advantage of the Renewable Forest Bioresource Turpentine to Prepare α,β-Unsaturated Compounds as Highly Efficient Fungicidal Candidates. J. Agric. Food Chem. 2021, 69(44), 12985–12993. DOI: 10.1021/acs.jafc.1c05364.

  12. Geng, Y. X.; Gui, K.; Pan, T. M.; Ye, J. H.; Li, J.; Feng, J. T.; Ma, Z. Q.; Lei, P.; Gao, Y. Q. Preparation of terpene-derived fungicidal candidates with a 1,3,4-thiadiazole moiety for natural product-inspired agrochemical discovery. Ind. Crops Prod. 2022, 189, 115889. DOI: 10.1016/j.indcrop.2022.115889.

  13. 张学博, 马航宇, 孙腾达, 雷鹏, 杨新玲, 张晓鸣, 凌云. 新型哌啶基肉桂醛缩氨基硫脲衍生物的设计、合成及抑菌活性研究. 有机化学 2019, 39, 2965–2972. 

  14. 张晓鸣, 雷鹏, 李欣潞, 杨新玲, 张学博, 孙腾达, 凌云. 新型含硫羰基结构的Aspernigerin衍生物的合成及抑菌活性研究. 有机化学 2019, 39, 3197–3203.

  15. Li, G. C.; Lei, P.; Szostak, M. Transition-Metal-Free Esterification of Amides via Selective N−C Cleavage under Mild Conditions. Org. Lett. 2018, 20, 5622−5625.

  16. Li, G. C.; Lei, P.; Szostak, M.; Casals-Cruañas, E.; Poater, A.; Cavallo, L.; Nolan, S. P. Mechanistic Study of Suzuki-Miyaura Cross-Coupling Reactions of Amides Mediated by [Pd(NHC)(allyl)Cl] Precatalysts. ChemCatChem 2018, 10, 3096–3106.

  17. Li, G. C.; Shi, S. C.; Lei, P.; Szostak, M. Pd-PEPPSI: Water-Assisted Suzuki–Miyaura Cross-Coupling of Aryl Esters at Room Temperature using a Practical Pd-NHC Precatalyst. Adv. Synth. Catal. 2018, 360, 1538–1543.

  18. Meng, G. R.; Lei, P.; Szostak, M. Pd-PEPPSI: A general method for two-step transamidation of secondary amides using commercially available, air- and moisture-stable palladium/NHC (N-heterocyclic carbene) complexes. Org. Lett. 2017, 19, 2158−2161. (Highly Cited Paper)

  19. Zhang, X. B.; Lei, P.; Sun, T. D.; Jin, X. Y.; Yang, X. L.; Ling, Y. Design, synthesis and fungicidal activity of novel benzaldehyde thiosemicarbazide derivatives containing piperidine fragments. Molecules 2017, 22, 2085. 

  20. Han, M.; Ma, X.; Yao, S.; Ding, Y.; Yan, Z.; ADiJiang, A.; Wu, Y.; Li, H.; Zhang, Y.; Lei, P.; Ling, Y.; An, J. Development of a modified Bouveault-Blanc reduction for the selective synthesis of alpha,alpha-dideuterio alcohols. J. Org. Chem. 2017, 82, 1285–1290. 

  21. Xu, G. F.; Yang, X. L.; Jiang, B. B; Lei, P.; Liu, X. L.; Wang, Q. M.; Zhang, X. B.; Ling, Y. Synthesis and bioactivities of novel piperazine-containing 1,5-Diphenyl-2-penten-1-one analogues from natural product lead. Bioorg. Med. Chem. Lett. 2016, 26, 1849–1853.

  22. Xu, G. F.; Yang, X. L.; Lei, P.; Liu, X. L.; Zhang, X. B.; Ling, Y. Synthesis and fungicidal activity study of novel daphneolone analogs with 2,6-dimethylmorpholine. Chin. Chem. Lett. 2016, 27, 555–558. 

  23. 徐焱, 雷鹏, 凌云, 王圣文, 杨新玲. 新型(3-取代苯基-2-丙烯-1-亚基)-苯甲酰腙类化合物的设计、合成及生物活性研究. 有机化学, 2014, 34, 1118–1123.


二、授权专利

  1. 雷鹏, 王宇佳, 高艳清, 陈光友, 蔡崇林, 马志卿, 冯俊涛. 一种噁二唑类化合物、制备方法及应用. 中国发明专利, 专利号: ZL 202210280280.0, 授权日期: 2023年10月11日.

  2. 雷鹏, 张彩霞, 马志卿, 高艳清, 李文奎, 陈光友, 闫合, 冯俊涛. 一种含异噁唑啉的酯类化合物、制备方法及应用. 中国发明专利, 专利号: ZL 202211404419.4, 授权日期: 2024年03月15日.

  3. 雷鹏, 穆雅利, 胡夏桐, 王宇佳, 马志卿, 冯俊涛, 王勇, 王艺博. 一种肟醚（酯）类化合物、制备方法及应用. 中国发明专利, 专利号: ZL 202010560725.1, 授权日期: 2023年09月1日.

  4. 雷鹏, 王艺博, 高艳清, 陈光友, 蔡崇林, 马志卿, 冯俊涛. 一种异噁唑啉类化合物、制备方法及应用. 中国发明专利, 专利号: ZL 202210031504.4, 授权日期: 2023年05月23日.

  5. 安杰, 张小河, 雷鹏, 凌云, 等. 一类新型电子盐的制备及其媒介的绿色伯奇还原反应. 中国发明专利, 专利号: ZL 201710059952.4, 授权日期: 2021年01月08日.

  6. 安杰, 雷鹏, 韩敏晖, 马晓栋, 等. 一种α, α‐二氘代醇类化合物的合成方法. 中国发明专利, 专利号: ZL 201610382079.8, 授权日期: 2020年11月03日.

  7. 凌云, 雷鹏, 杨新玲, 徐焱, 等.（1,2,3,4-四氢喹啉-1-基）（取代吡唑基）甲酮类化合物及其应用. 中国发明专利, 专利号: ZL 201510796235.0, 授权日期: 2017年12月19日.

  8. 凌云, 雷鹏, 杨新玲, 徐焱, 等. N'-取代苯亚甲基-1,2,3,4-四氢喹啉基-1-(硫代)酰肼类化合物及其制备方法和应用. 中国发明专利, 专利号: ZL 201510434634.2, 授权日期: 2017年07月18日.