Publications：

63. Sun Meng, Zhou Si-Jia, Lou Sai-Fan, Xiao Jian, Jiao Yin-Chun* and Shi Feng*, Catalytic Asymmetric (4+3) Cyclizations of In Situ Generated ortho-Quinone Methides with 2-Indolylmethanols, Angew. Chem. Int. Ed. 2019, in press. (IF = 12.1)

62. Zhang Lei, Xiang Shao-Hua, Wang Jun, Xiao Jian, Wang Junqi, Tan Bin*, Phosphoric Acid Catalyzed Atroposelective Construction of Axially Chiral Arylpyrroles, Nat. Comm. 2019, 10, 566.  (IF = 12.353)

61. Li Shuai-Shuai, Zhu Shuai, Chen Chunqi, Duan Kang, Liu Qing, Xiao Jian*. Hydride Transfer Involved Redox-Neutral Cascade Cyclizations for Construction of Spirocyclic Bisoxindoles Featuring a [3,4]-Fused Oxindole Moiety. Org. Lett. 2019, 21, 1058 . (IF = 6.579)

60. Zhu Shuai, Chen Chunqi, Duan Kang, Li Shuai-Shuai*, Liu Qing, Xiao Jian*.Cascade [1,5]-Hydride Transfer/Cyclization for Synthesis of [3,4]-Fused Oxindoles, J. Org. Chem. 2019.  (IF = 4.805)

59. Xu Lubin, Chen Haohua, Liu Jian, Zhou Lan, Lan Yu *,Xiao Jian *, Chiral Phosphoric Acid Catalyzed Asymmetric C(sp3)–H Functionalization of Biomass-Derived 2,5-Dimethylfuran via Two Sequential Cope-Type Rearrangements, Org. Chem. Front. 2019, 6,1162. (IF = 5.455)

58. Shen Yao-Bin, Li Shuai-Shuai, Sun Yun-Ming, Yu Liping, Hao Zhi-Hui*, Liu Qing, Xiao Jian*, Organocatalytic C(sp3)−H Functionalization of 5-Methyl-2,3-dihydrofuran Derivatives with Trifluoropyruvates via Sequential exo-Tautomerization/Carbonyl-Ene Process, J. Org. Chem. 2019, 84, 2779. (IF = 4.805)

57.Shen Yao-Bin, Li Shuai-Shuai, SunYun-Ming, Liu Xicheng, Yu Liping, Liu Qing, Xiao Jian*, Formal [4 + 2] Annulation of Oxindole-Embedded ortho-Quinone Methides with 1,3-Dicarbonyls: Synthesis of Spiro[Chromen-4,3'-Oxindole] Scaffolds, J. Org. Chem. 2019, 84, 3990. (IF = 4.805)

56. Shen Yao-Bin, Li Shuai-Shuai, Liu Xicheng, Yu Liping, Liu Qing,  Xiao Jian*, Dearomative [4+2] Cycloaddition of Oxindole-Embedded ortho-Quinone Methides with 2,5-Dialkylfurans, Adv. Syn. Catal. 2019, 361, 1453. (IF = 5.123)

55. Lv Xintong, Hu Fangzhi, Duan Kang, Li Shuai-Shuai, Liu Qing, Xiao Jian*, Aromatization-Driven Cascade [1, 5]-Hydride Transfer Reaction Promoted by Fluorinated Alcohols, J. Org. Chem. 2019, 84, 1833. (IF = 4.805)

54. Yu Liping, Li Shuai-Shuai, Li Weina, Yu Shitao*, Liu Qing,  Xiao Jian*, Fluorinated Alcohol Promoted Reaction of Chlorohydrocarbon with Diverse Nucleophiles for Synthesis of Triarylmethanes and Tetraarylmethanes, J. Org. Chem. 2018, 83, 15277. (IF = 4.805)

53. Wang Shuai, An Xiao-De, Li Shuai-Shuai, Liu Xicheng, Liu Qing,Xiao Jian*，Hydride Transfer Initiated Ring Expansion of Pyrrolidines toward Highly Functionalized Tetrahydro-1-benzazepines, Chem. Comm. 2018, 54, 3833. (IF = 6.290)

52. Li Shuai-Shuai, Lv Xintong, Ren Didi, Shao Chang-Lun, Liu Qing, Xiao Jian*, Redox-Triggered Cascade Dearomative Cyclizations Enabled by Hexafluoroisopropanol, Chem. Sci. 2018, 9, 8253. (IF = 9.063)

51. Shen Yao-Bin, Li Shuai-Shuai, An Xiao-De, Liu Qing，Liu Xicheng, Xiao Jian*, Organocatalytic Dearomative [4 + 2] Cycloadditions of Biomass-Derived 2,5-Dimethylfuran with ortho-Quinone Methides: Access to Multi-Substituted Chromanes, Org. Lett. 2018, 20, 6069. (IF = 6.579)

50. Li Shuai-Shuai, Zhou Lan, Wang Liang, Zhao Huaili, Yu Liping, Xiao Jian*, Carbocation-Initiated Cascade [1,5]-Hydride Transfer/Cyclization: Facile Synthesis of dibenzo[b,e]azepines， Org. Lett. 2018, 20, 138. (IF = 6.492)

49. Zhu Shuai, Chen Chunqi, Xiao Mingyan, Yu Liping, Wang Liang*, Xiao Jian*, Construction of the Tetrahydroquinoline Spiro Skeleton via Cascade [1,5]-Hydride transfer-involved C(sp3)-H Functionalization on Water, Green Chem. 2017, 19, 5653. (IF = 8.586)

48. Xiao Mingyan, Ren Didi, Xu Lubin, Yu Liping and Xiao Jian*, SN1-type Alkylation of N-Heteroaromatics with Alcohols, Org. Lett. 2017, 19, 5724. (IF = 6.492)

47. Li Shuai-Shuai, Fu Shiheng, Wang Liang, Xu Lubin and Xiao Jian*, t-BuOK-Mediated Oxidative C(sp3)-H Arylation of 2-Alkylazaarenes with Nitroarenes, J. Org. Chem. 2017, 82, 8703. (IF = 4.805)

46. Xiao Jian*, Wen Hao, Wang Liang, Xu Lubin, Hao Zhihui, Shao Chang-Lun*, Wang Chang-Yun, Catalyst-Free Dehydrative SN1-Type Reaction of Indolyl Alcohols with Diverse Nucleophiles on Water, Green Chem. 2016, 18, 1032. (IF = 8.586, Hot Paper, Highlighted by X-mol资讯网站，科技日报，中国网)

45. Wang Liang, Xiao Jian*, Hydrogen-Atom Transfer Reactions, Topics in Current Chemistry. 2016, 374, 17. (IF=4.46, Invited Review)

44. Wang Liang, Xiao Jian*, C(sp3)-H Bond Functionalization by Sequential Hydride Transfer/Cyclization: Electronic Effect and Steric Effect Controlled Regioselectivity, Org. Chem. Front. 2016, 3, 635. (IF=5.455, Inside Front Cover, Hot Articles in March 2016)

43. Zhao Huaili, Xiao Mingyan, Wang Liang * and Xiao Jian *, Bifunctional Thiourea Catalyzed Asymmetric Michael Addition of Anthrone to Methyleneindolinones, RSC Adv. 2016, 6, 38588 (IF=2.936)

42. Liu Jian, Wang Xiaoxiao, Wang Liang, Xu Lubin, Hao Zhihui and Xiao Jian*, Fluorinated Alcohol-Mediated [4+3] Cycloaddition Reaction of Indolyl Alcohols with Cyclopentadiene, Org. Biomol. Chem. 2016, 14, 11510. (IF = 3.423)

41. Dong Haoxun, Xu Lubin, Li Shuai-Shuai, Wang Liang, Shao Chang-Lun, Xiao Jian*, Facile Synthesis of Azaarene-substituted Hydroxycoumarins Possessing High Biological Activities via Three-Component C(sp3)-H Functionalization, ACS Comb. Sci. 2016, 18, 604. (IF=3.5)

40. Liu Jian, Wang Xiaoxiao, Xu Lubin, Hao Zhihui, Wang Liang* and Xiao Jian *, One Step Synthesis of 2-Alkenylchromanes via Inverse Electron-Demand Hetero-Diels-Alder Reaction of o-Quinone Methide with Unactivated Dienes, Tetrahedron. 2016, 72,7642. (IF = 2.651)

39. Zhao Huaili, Wang Xiaoxiao, Wang Liang* and Xiao Jian*, Regioselective Michael Addition of Anthrone to Methyleneindolinones, Synthesis. 2016, 48, 2112. (IF=2.650)

38. Fu Shiheng, Wang Liang, Dong Haoxun, Yu Junqiang, Xu Lubin and Xiao Jian*, Facile Synthesis of 2-Alkenylazaarenes via Dehydrative Coupling of 2-Methylazaarenes with Aldehydes on Water, Tetrahedron Lett. 2016, 57, 4533. (IF = 2.125)

37. Zhang Xianhui, Li Shuai-Shuai, Wang Liang, Xu Lubin, Xiao Jian *, Zhen-Jiang Liu*, 2-Methylquinoline Promoted Oxidative Ring-Opening of N-Sulfonyl Aziridines with DMSO: Facile Synthesis of α-Amino Aryl Ketones, Tetrahedron. 2016, 72, 8073. (IF = 2.125)

36. Zhu Shuai, Xu Lubin, Wang Liang*, Xiao Jian*, Recent Advances in Asymmetric Synthesis of Optically Active Indole Derivatives from 3-Indolylmethanols, Chin. J. Org. Chem. 2016, 36, 1229. (IF=1.852)

35. Liu Qing, Dong Xu, Li Jun, Xiao Jian, Dong Yunhui,* and Liu Hui*, Recent Advances on Palladium Radical Involved Reactions, ACS Catal. 2015, 5, 6111 (IF=11.384)

34. Wen Hao, Wang Liang, Xu Lubin, Hao Zhihui, Shao Chang-Lun,* Wang Chang-Yun, Xiao Jian*, Fluorinated Alcohol-Mediated SN1-Type Reaction of Indolyl Alcoholswith Diverse Nucleophiles, Adv. Syn. Catal. 2015, 357, 4023 (IF = 5.123) (VIP and Cover Picture, Highlighted by X-mol资讯网站，科技日报，中国网)

33. Wang Xiaoxiao, Liu Jian, Xu Lubin, Hao Zhihui, Wang Liang*, Xiao Jian*, Friedel–CraftsAlkylation of Heteroarenes and Arenes with Indolyl Alcohols for Construction of 3,3-Disubstituted Oxindoles, RSC Adv. 2015, 5, 101713. (IF=2.936)

32.  Xu Lubin, Shao Zhuzhou, Wang Liang，Xiao Jian*, Tandem sp3 C-H Activation/Decarboxylation of 2-Alkyl Azaarenes with Coumarin-3-Carboxylic Acid, Org. Lett. 2014, 16, 796. (IF = 6.492)

31.  Wang Liang, Xiao Jian*, Advancement of Cascade [1,5]-Hydrogen Transfer/Cyclization: A Method for Direct Functionalization of Inactive C(sp3)-H Bonds, Adv. Syn. Catal. 2014, 356, 1137. (IF = 5.123)

30.  Xiao Jian*, Chen Yuye, Zhu Shuai, Wang Liang, Xu Lubin, Wei Hongtao, Diversified Construction of Chromeno[3,4-c]pyridin-5-one and Benzo[c]chromen-6-one Derivatives by Domino Reaction of 4-alkynyl-2-oxo-2H-chromene-3-carbaldehydes, Adv. Syn. Catal. 2014, 356, 1835. (IF = 5.123)

29.  Wang Liang, Xiao Jian*,LohTeck-Peng*, Organocatalyticβ-Functionalization of Saturated Carbonyl Compounds---The State of the Art, Chem Cat Chem. 2014, 6, 1183.(IF = 4.674)

28.  Shao Zhuzhou, Xu Lubin, Wang Liang, Wei Hongtao, Xiao Jian,* Catalyst-free Tandem Michael Addition/Decarboxylation of (thio)coumarin-3-carboxylic Acids with Indoles: Facile Synthesis of Indole-3-substituted 3,4-dihydro(thio)coumarins, Org. Biomol.Chem. 2014, 12, 2185. (IF = 3.423)

27. Wang Liang, Chen Yuye, Xiao Jian*, AlkylideneindoleniniumIons and Alkylideneindolenine: Key Intermediates for Asymmetric Synthesis of 3-Substituted Indoles, Asian J. Org.Chem. 2014, 3, 1036. (IF = 2.496)

26. Shao Zhuzhou, Wang Liang, Xu Lubin, Zhao Huaili and Xiao Jian *, Facile Synthesis of Azaarene-2-substituted Chromanone Derivatives via Tandem sp3 C−H Functionlization/Decarboxylation of Azaarenes with 4-oxo-4H-chromene-3-carboxylic acid, RSC Advances. 2014, 4, 53188. (IF = 2.936)

25. Xu Lubin, Shao Zhuzhou, Wang Liang, Zhao Huaili and Xiao Jian *, Catalyst-Free Synthesis of (Z)-2-Alkenylquinoline Derivatives via C(sp3)-H Functionalization of 2-Methylquinolines, Tetrahedron Lett. 2014, 55, 6856. (IF = 2.125)

24. Yu Xinzhang, Yu Songjie, Xiao Jian, Wan Boshun, Li Xingwei*, Rhodium(III)-Catalyzed Azacycle-Directed Intermolecular Insertion of Arene C−H Bonds into α-Diazocarbonyl Compounds, J. Org. Chem. 2013, 78, 5444. (IF = 4.849)

23.  Xiao Jian*, Merging Organocatalysis with Transition Metal Catalysis: HighlyStereoselective Alkylation of Aldehydes, Org. Lett. 2012, 14, 1716. (IF = 6.579) (Highlighted by Synfacts 2012, 8, 0749)

22. Xiao Jian*, Oxidative Enamine Catalysis: Direct Catalytic Enantioselective β-Functionalization of Aldehydes, Chem Cat Chem. 2012, 4, 612. (IF = 4.803)

21. Liang Tao, Xiao Jian*, Xiong Zhiyi，Li Xingwei*, Organocatalytic Asymmetric 1,4 Addition of Aldehydes to Acridiniums Catalyzed by a DiarylprolinolSilyl Ether, J. Org. Chem. 2012, 77, 3583. (IF =4.805)

20. NiuRui, Xiao Jian*, Liang Tao, Li Xingwei*, Facile Synthesis of Azaarene-Substituted 3-Hydroxy-2-Oxindoles via Bronsted Acid-Catalyzed sp3C-H Functionalization, Org. Lett. 2012, 14, 676. (IF = 6.492)

19. Xiao Jian, Zhao Kai, LohTeck-Peng*, The OrganocatalyticEnantioselective Acid Free Alkylation of Aldehydes in Fluorinated Alcohols, Chem. Comm. 2012, 48, 3548. (IF = 6.29)

18. Huang Fen, Xu Lubin, Xiao Jian*, OrganocatalyticEnantioselectiveDehydrogenative α-Alkylation of Aldehydes with Benzylic Compounds, Chin. J. Chem. 2012, 30, 2721. (IF = 2.378)

(Invited Special Issue of "Asymmetric Synthesis", one of the most accessed papers from 11/2012 to 10/2013).

17. NiuRui, Yang Shiying, Xiao Jian*, Liang Tao, Li Xingwei*, Yb(OTf)3-Catalyzed Addition of 2-methylAzaarenesto Isatins via C-H Functionalization, Chin. J. Catal. 2012, 33, 1636. (IF = 2.378)

16. Wang Xiaowei, Li Xuting, Xiao Jian, Jiang Yi, Li Xingwei*, Rh(III)-Catalyzed Oxidative Olefination of N-(Naphthalen-1-yl)amides, Synlett. 2012, 1649. (IF = 2.151)

15. Xiao Jian, Zhao Kai, LohTeck-Peng*, Highly Enantioselective Intermolecular Alkylation of Aldehydes with Alcohols by Cooperative Catalysis of DiarylprolinolSilyl Ether with Brønsted Acid, Chem. Asian J. 2011, 6, 2890. (IF = 3.692)

14. Xiao Jian and Li Xingwei*, Gold a-Oxo Carbenoids in Catalysis: Catalytic O-Atom Transfer to Alkynes, Angew. Chem. Int. Ed.2011, 50, 7226. (IF = 12.102)

13. Xiao Jian, Lu Yun-Peng, Liu Yan-Ling, Wong Poh-Shen, LohTeck-Peng*, A New Class of Structurally Rigid Tricyclic Chiral Secondary Amine Organocatalyst: Highly EnantioselectiveOrganocatalytic Michael Addition of Aldehydes to Vinyl Sulfones, Org. Lett. 2011, 13, 876.(IF = 6.492)

12. Xiao Jian, Xu Feng-Xia, Lu Yun-Peng, Liu Yan-Ling, LohTeck-Peng*, Highly Efficient and Modularly Tuned Bicyclic Organocatalyst for the Enantioselective Michael Addition of Aldehydes to Nitroalkenes, Synthesis-Stuttgart. 2011, 1292. (IF = 2.650)

11. Xiao Jian, Xu Feng-Xia, Lu Yun-Peng, LohTeck-Peng*, Chemzymes: A New Class of Structurally Rigid Tricyclic Amphibian Organocatalyst Inspired by Natural Product, Org. Lett. 2010,12, 1220. (IF = 6.492) (Highlighted by Synfacts 2011, 5, 0561)

10. Xiao Jian, Wong Zhen-Zhou, Lu Yun-Peng, LohTeck-Peng*, Hexahydropyrrolo[2,3-b]indoles: A New Class of Structurally Rigid Tricyclic Skeleton for Oxazaborolidine-Catalyzed Asymmetric Borane Reduction, Adv. Synth. Catal. 2010, 352, 1107. (IF = 5.123)

9. Xiao Jian and Loh Teck-Peng*, The Organocatalytic Enantioselective Michael Addition of Aldehydes to Vinyl Sulfones in Water, Synlett. 2010, 2029. (IF = 2.151)

8. Xiao Jian and Loh Teck-Peng*, Design, Synthesis and Optical Resolution of New Bifunctional Ligand: 1,1′-Dimethyl-octahydro-8,8′-Biquinoline-7,7′-diol, Org. Lett. 2009, 11, 2876. (IF = 6.492)

7. Xiao Jian and Loh Teck-Peng*, Unexpected Domino Ring Closure: Highly Stereoselective Construction of a Tetracyclic Indole Alkaloid Ring System, Tetrahedron Lett. 2008, 49, 7184. (IF = 2.125)

6. Xiao Jian and Loh Teck-Peng*, Design and Synthesis of a Water-Tolerant Chiral Indium Complex: Application to One-Pot Three-Component Mannich-Type Reactions in Water, Synlett. 2007, 815. (IF = 2.151)

5. Xiao Jian, Lu Yong-Na, Wang Guo-Cang, Li Jin-Shan et al., 3-(3H-Inden-1-ylmethyl)-2,2'-bis(methoxymethoxy)1,1'-binaphthalenyl, Acta Crystallographica Section E. 2005, 61, O1501.

4.Wang Guo-Cang, Xiao Jian, Lu Yong-Na, et al., Synthesis, Crystal Structures and in Vitro Antitumor Activities of Some Arylantimony Derivatives of Analogues of Demethylcantharimide, J. Organomet. Chem. 2004, 689, 1631. (IF = 2.184)

3.Wang Guo-Cang, Xiao Jian, Lu Yong-Na, Li Jin-Shan, Synthesis, Characterization and in Vitro Cytotoxicity Screening of Some Triarylbismuth(V) di(N-salicylidene) Amino Carboxylates and the Crystal Structure of (2-HOC6H4CH=NCH2CO2)2Bi(C6H5)3, Appl. Organomet. Chem. 2005, 19, 113. (IF = 2.4)

2.Wang Guo-Cang, Lu Yong-Na, Xiao Jian, Li Jin-Shan, Synthesis, Crystal Structures and in Vitro Antitumor Activities of Some Organoantimony Arylhydroxamates, J. Organomet. Chem. 2005, 690, 151. (IF = 2.184)

1. Guo Qun-Sheng, Lu Yong-Na, Liu Bing, Xiao Jian, Li Jin-Shan, A Facile Synthesis of 3 or 3,3′-Substituted Binaphthols and Their Applications in the Asymmetric Addition of Diethylzinc to Aldehydes, J. Organomet. Chem. 2006, 691, 1282. (IF = 2.184)

Patents

7. 肖建， 朱帅， 王亮，“一种无催化剂条件下构建三芳基和四芳基甲烷的方法”

申请号：201710504410.3

6. 肖建， 朱帅， 王亮，“一种合成吲哚取代或二茂铁取代氮杂芳烃的方法”

申请号：201710442072.5

5. 肖建，朱帅，“一种在无催化剂条件下构建四氢喹啉螺环骨架的方法”

申请号：201611038032.6

4. 肖建， 朱帅， 王亮，“一种氮杂芳烃苄位与缺电子芳环偶联的方法”

申请号：201611188837.9

3. 肖建，徐鲁斌，邵朱宙，“3-(1-芳基-2-(2-氮杂芳烃)乙基)-4-羟基香豆素及其制备方法”申请号：201510679157.6

2. Loh Teck-Peng* and Xiao Jian “Process for Preparation of Octahydrobiquinoline Compounds”, PCT International Patent Application, 2010, 59pp. Patent Number: WO 2010132029

1. Loh Teck-Peng* and Xiao Jian “Preparation of Tricyclic Chiral Compounds and Their Use in Asymmetric Catalysis”, PCT International Patent Application, 2010, 141pp. Patent number: WO2010027334