Oxidant-Induced Azolation of Electron-Rich Phenol Derivatives.,Organic Letters

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Oxidant-Induced Azolation of Electron-Rich Phenol Derivatives.
Organic Letters ( IF 4.9 ) Pub Date : 2020-07-02 , DOI: 10.1021/acs.orglett.0c01796
Xiaoyu Wang ₁ , Shengchun Wang ₂ , Yiming Gao ₂ , He Sun ₂ , Xing'an Liang ₂ , Faxiang Bu ₂ , Takfaoui Abdelilah ₂ , Aiwen Lei _{1,

2}

Affiliation

Since N-arylazoles are widely present in natural products, pharmaceuticals, and functional materials, it is important to develop a simple and efficient synthetic method for the synthesis of N-arylazoles. Herein, an oxidant-induced intermolecular azolation of phenol derivatives was demonstrated under catalyst-free condition. Both monoazolation and diazolation of phenols can be successfully achieved via this practical and powerful method.

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